Entry Database : PDB / ID : 6d1s Structure visualization Downloads & linksTitle Crystal structure of an apo chimeric human alpha1GABAA receptor Componentschimeric alpha1GABAA receptor Details Keywords PROTEIN TRANSPORT / GABAA receptor / anesthetics / alphaxalone / neurosteroidsFunction / homology Function and homology informationFunction Domain/homology Component
GABA receptor complex / inhibitory extracellular ligand-gated monoatomic ion channel activity / GABA receptor activation / GABA-gated chloride ion channel activity / inhibitory synapse assembly / GABA-A receptor activity / GABA-A receptor complex / synaptic transmission, GABAergic / gamma-aminobutyric acid signaling pathway / Signaling by ERBB4 ... GABA receptor complex / inhibitory extracellular ligand-gated monoatomic ion channel activity / GABA receptor activation / GABA-gated chloride ion channel activity / inhibitory synapse assembly / GABA-A receptor activity / GABA-A receptor complex / synaptic transmission, GABAergic / gamma-aminobutyric acid signaling pathway / Signaling by ERBB4 / extracellular ligand-gated monoatomic ion channel activity / chloride channel complex / GABA-ergic synapse / regulation of postsynaptic membrane potential / chloride transmembrane transport / dendrite membrane / transmitter-gated monoatomic ion channel activity involved in regulation of postsynaptic membrane potential / cytoplasmic vesicle membrane / transmembrane signaling receptor activity / postsynapse / postsynaptic membrane / neuron projection / synapse / membrane / identical protein binding / plasma membrane Similarity search - Function : / Gamma-aminobutyric-acid A receptor, alpha 1 subunit / : / Gamma-aminobutyric-acid A receptor, alpha subunit / Acetylcholine Binding Protein; Chain: A, / Neurotransmitter-gated ion-channel ligand-binding domain / Gamma-aminobutyric acid A receptor/Glycine receptor alpha / Neurotransmitter-gated ion-channel, conserved site / Neurotransmitter-gated ion-channels signature. / Neurotransmitter-gated ion-channel transmembrane domain ... : / Gamma-aminobutyric-acid A receptor, alpha 1 subunit / : / Gamma-aminobutyric-acid A receptor, alpha subunit / Acetylcholine Binding Protein; Chain: A, / Neurotransmitter-gated ion-channel ligand-binding domain / Gamma-aminobutyric acid A receptor/Glycine receptor alpha / Neurotransmitter-gated ion-channel, conserved site / Neurotransmitter-gated ion-channels signature. / Neurotransmitter-gated ion-channel transmembrane domain / Neurotransmitter-gated ion-channel transmembrane region / Neurotransmitter-gated ion-channel transmembrane domain superfamily / Neuronal acetylcholine receptor / Neurotransmitter-gated ion-channel / Neurotransmitter-gated ion-channel ligand-binding domain / Neurotransmitter-gated ion-channel ligand-binding domain superfamily / Neurotransmitter-gated ion-channel ligand binding domain / Distorted Sandwich / Mainly Beta Similarity search - Domain/homologyBiological species Dickeya dadantii (bacteria)Homo sapiens (human)Method X-RAY DIFFRACTION / SYNCHROTRON / MOLECULAR REPLACEMENT / Resolution : 3.2 Å DetailsAuthors Chen, Q. / Arjunan, P. / Cohen, A.E. / Xu, Y. / Tang, P. Funding support United States, 1items Details Hide detailsOrganization Grant number Country National Institutes of Health/National Human Genome Research Institute (NIH/NHGRI) R01GM056257 United States
CitationJournal : Nat Commun / Year : 2018Title : Structural basis of neurosteroid anesthetic action on GABAAreceptors.Authors : Chen, Q. / Wells, M.M. / Arjunan, P. / Tillman, T.S. / Cohen, A.E. / Xu, Y. / Tang, P. History Deposition Apr 12, 2018 Deposition site : RCSB / Processing site : RCSBRevision 1.0 Aug 22, 2018 Provider : repository / Type : Initial releaseRevision 1.1 Oct 3, 2018 Group : Data collection / Database references / Category : citationItem : _citation.country / _citation.journal_abbrev ... _citation.country / _citation.journal_abbrev / _citation.journal_id_CSD / _citation.journal_id_ISSN / _citation.pdbx_database_id_DOI / _citation.title / _citation.year Revision 1.2 Oct 10, 2018 Group : Data collection / Database references / Structure summaryCategory : citation / citation_author / entityItem : _citation.journal_volume / _citation.page_first ... _citation.journal_volume / _citation.page_first / _citation.page_last / _citation.pdbx_database_id_DOI / _citation.pdbx_database_id_PubMed / _citation.title / _citation.year / _entity.formula_weight Revision 1.3 Oct 24, 2018 Group : Data collection / Database references / Structure summaryCategory : citation / citation_author / entityItem : _citation.journal_volume / _citation.page_first ... _citation.journal_volume / _citation.page_first / _citation.page_last / _citation.pdbx_database_id_DOI / _citation.pdbx_database_id_PubMed / _citation.title / _citation.year / _entity.formula_weight Revision 1.4 Dec 18, 2019 Group : Author supporting evidence / Category : pdbx_audit_support / Item : _pdbx_audit_support.funding_organizationRevision 1.5 Mar 13, 2024 Group : Data collection / Database references / Category : chem_comp_atom / chem_comp_bond / database_2Item : _database_2.pdbx_DOI / _database_2.pdbx_database_accession
Show all Show less