登録情報 | データベース: PDB / ID: 3gqy |
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タイトル | Activator-Bound Structure of Human Pyruvate Kinase M2 |
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要素 | Pyruvate kinase isozymes M1/M2 |
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キーワード | TRANSFERASE (転移酵素) / activator / Acetylation (アセチル化) / Allosteric enzyme / Alternative splicing (選択的スプライシング) / Glycolysis (解糖系) / Kinase (キナーゼ) / Magnesium (マグネシウム) / Metal-binding / Phosphoprotein / Polymorphism / Pyruvate (ピルビン酸) / Structural Genomics (構造ゲノミクス) / Structural Genomics Consortium / SGC |
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機能・相同性 | 機能・相同性情報
ピルビン酸キナーゼ / pyruvate kinase activity / positive regulation of cytoplasmic translation / プログラム細胞死 / histone H3T11 kinase activity / canonical glycolysis / 解糖系 / positive regulation of sprouting angiogenesis / potassium ion binding / 小胞体 ...ピルビン酸キナーゼ / pyruvate kinase activity / positive regulation of cytoplasmic translation / プログラム細胞死 / histone H3T11 kinase activity / canonical glycolysis / 解糖系 / positive regulation of sprouting angiogenesis / potassium ion binding / 小胞体 / glycolytic process / non-specific protein-tyrosine kinase / 繊毛 / cellular response to insulin stimulus / extracellular vesicle / MHC class II protein complex binding / protein tyrosine kinase activity / secretory granule lumen / collagen-containing extracellular matrix / vesicle / ficolin-1-rich granule lumen / transcription coactivator activity / non-specific serine/threonine protein kinase / cadherin binding / リン酸化 / mRNA binding / Neutrophil degranulation / magnesium ion binding / protein homodimerization activity / positive regulation of transcription by RNA polymerase II / ミトコンドリア / RNA binding / extracellular exosome / extracellular region / ATP binding / 細胞核 / 細胞質基質 / 細胞質類似検索 - 分子機能 PK beta-barrel domain-like / M1 Pyruvate Kinase; Domain 3 / Pyruvate kinase, C-terminal domain / Pyruvate Kinase; Chain: A, domain 1 / Pyruvate kinase, active site / Pyruvate kinase active site signature. / ピルビン酸キナーゼ / Pyruvate kinase, barrel / Pyruvate kinase, insert domain superfamily / Pyruvate kinase, barrel domain ...PK beta-barrel domain-like / M1 Pyruvate Kinase; Domain 3 / Pyruvate kinase, C-terminal domain / Pyruvate Kinase; Chain: A, domain 1 / Pyruvate kinase, active site / Pyruvate kinase active site signature. / ピルビン酸キナーゼ / Pyruvate kinase, barrel / Pyruvate kinase, insert domain superfamily / Pyruvate kinase, barrel domain / Pyruvate kinase, C-terminal / Pyruvate kinase, C-terminal domain superfamily / Pyruvate kinase, alpha/beta domain / Pyruvate kinase-like, insert domain superfamily / Phosphoenolpyruvate-binding domains / Pyruvate kinase-like domain superfamily / Pyruvate/Phosphoenolpyruvate kinase-like domain superfamily / TIMバレル / Alpha-Beta Barrel / Βバレル / 3-Layer(aba) Sandwich / Mainly Beta / Alpha Beta類似検索 - ドメイン・相同性 Chem-DZG / 1,6-di-O-phosphono-beta-D-fructofuranose / L(+)-TARTARIC ACID / Pyruvate kinase PKM類似検索 - 構成要素 |
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生物種 | Homo sapiens (ヒト) |
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手法 | X線回折 / 分子置換 / 解像度: 1.85 Å |
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データ登録者 | Hong, B. / Dimov, S. / Tempel, W. / Auld, D. / Thomas, C. / Boxer, M. / Jianq, J.-K. / Skoumbourdis, A. / Min, S. / Southall, N. ...Hong, B. / Dimov, S. / Tempel, W. / Auld, D. / Thomas, C. / Boxer, M. / Jianq, J.-K. / Skoumbourdis, A. / Min, S. / Southall, N. / Arrowsmith, C.H. / Edwards, A.M. / Bountra, C. / Weigelt, J. / Bochkarev, A. / Inglese, J. / Park, H. / Structural Genomics Consortium (SGC) |
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引用 | ジャーナル: to be published タイトル: Activator-Bound Structures of Human Pyruvate Kinase M2 著者: Hong, B. / Dimov, S. / Tempel, W. / Auld, D. / Thomas, C. / Boxer, M. / Jianq, J.-K. / Skoumbourdis, A. / Min, S. / Southall, N. / Arrowsmith, C.H. / Edwards, A.M. / Bountra, C. / Weigelt, J. ...著者: Hong, B. / Dimov, S. / Tempel, W. / Auld, D. / Thomas, C. / Boxer, M. / Jianq, J.-K. / Skoumbourdis, A. / Min, S. / Southall, N. / Arrowsmith, C.H. / Edwards, A.M. / Bountra, C. / Weigelt, J. / Bochkarev, A. / Inglese, J. / Park, H. |
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履歴 | 登録 | 2009年3月24日 | 登録サイト: RCSB / 処理サイト: RCSB |
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改定 1.0 | 2009年4月7日 | Provider: repository / タイプ: Initial release |
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改定 1.1 | 2011年7月13日 | Group: Version format compliance |
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改定 1.2 | 2017年11月1日 | Group: Refinement description / カテゴリ: software |
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改定 1.3 | 2020年7月29日 | Group: Data collection / Database references ...Data collection / Database references / Derived calculations / Structure summary カテゴリ: chem_comp / diffrn_source ...chem_comp / diffrn_source / entity / pdbx_chem_comp_identifier / pdbx_entity_nonpoly / struct_ref_seq_dif / struct_site / struct_site_gen Item: _chem_comp.mon_nstd_flag / _chem_comp.name ..._chem_comp.mon_nstd_flag / _chem_comp.name / _chem_comp.type / _diffrn_source.type / _entity.pdbx_description / _pdbx_entity_nonpoly.name / _struct_ref_seq_dif.details 解説: Carbohydrate remediation / Provider: repository / タイプ: Remediation |
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改定 1.4 | 2023年9月6日 | Group: Data collection / Database references ...Data collection / Database references / Refinement description / Structure summary カテゴリ: chem_comp / chem_comp_atom ...chem_comp / chem_comp_atom / chem_comp_bond / database_2 / pdbx_initial_refinement_model Item: _chem_comp.pdbx_synonyms / _database_2.pdbx_DOI / _database_2.pdbx_database_accession |
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