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-Structure paper
Title | A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases. |
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Journal, issue, pages | Acs Chem. Biol., Vol. 11, Page 772-781, Year 2016 |
Publish date | Oct 14, 2015 (structure data deposition date) |
Authors | Eram, M.S. / Shen, Y. / Szewczyk, M.M. / Wu, H. / Senisterra, G. / Li, F. / Butler, K.V. / Kaniskan, H.U. / Speed, B.A. / Dela Sena, C. ...Eram, M.S. / Shen, Y. / Szewczyk, M.M. / Wu, H. / Senisterra, G. / Li, F. / Butler, K.V. / Kaniskan, H.U. / Speed, B.A. / Dela Sena, C. / Dong, A. / Zeng, H. / Schapira, M. / Brown, P.J. / Arrowsmith, C.H. / Barsyte-Lovejoy, D. / Liu, J. / Vedadi, M. / Jin, J. |
External links | Acs Chem. Biol. / PubMed:26598975 |
Methods | X-ray diffraction |
Resolution | 2.55 Å |
Structure data | PDB-5e8r: |
Chemicals | ChemComp-SAH: ChemComp-5L6: ChemComp-CL: ChemComp-UNX: ChemComp-HOH: |
Source |
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Keywords | TRANSFERASE / HRMT1L6 / MS-023 / Structural Genomics / Structural Genomics Consortium / SGC |