9R3I
 
 | | Structure of liver pyruvate kinase in complex with fluorescent probe 4c | | Descriptor: | 1,6-di-O-phosphono-beta-D-fructofuranose, 4-[4-[[7-(dimethylamino)-2,1,3-benzoxadiazol-4-yl]sulfonyl]piperazin-1-yl]sulfonyl-5-pyridin-3-yl-benzene-1,2-diol, Isoform L-type of Pyruvate kinase PKLR | | Authors: | Bogucka, A, Nilsson, O, Grotli, M, Hyvonen, M. | | Deposit date: | 2025-05-05 | | Release date: | 2025-08-13 | | Method: | X-RAY DIFFRACTION (2.579 Å) | | Cite: | Fluorescent binding assay for allosteric ligands of liver pyruvate kinase.
Eur.J.Med.Chem., 298, 2025
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9R3L
 | | Structure of liver pyruvate kinase in complex with fluorescent probe 4d | | Descriptor: | 1,6-di-O-phosphono-beta-D-fructofuranose, 4-[4-[[7-(azetidin-1-yl)-2,1,3-benzoxadiazol-4-yl]sulfonyl]piperazin-1-yl]sulfonylbenzene-1,2-diol, Isoform L-type of Pyruvate kinase PKLR, ... | | Authors: | Bogucka, A, Nilsson, O, Grotli, M, Hyvonen, M. | | Deposit date: | 2025-05-05 | | Release date: | 2025-08-13 | | Method: | X-RAY DIFFRACTION (2.158 Å) | | Cite: | Fluorescent binding assay for allosteric ligands of liver pyruvate kinase.
Eur.J.Med.Chem., 298, 2025
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9R3H
 | | Structure of liver pyruvate kinase in complex with fluorescent probe 4b | | Descriptor: | 1,6-di-O-phosphono-beta-D-fructofuranose, 4-[4-[(7-azanyl-2,1,3-benzoxadiazol-4-yl)sulfonyl]piperazin-1-yl]sulfonylbenzene-1,2-diol, Isoform L-type of Pyruvate kinase PKLR, ... | | Authors: | Bogucka, A, Nilsson, O, Grotli, M, Hyvonen, M. | | Deposit date: | 2025-05-05 | | Release date: | 2025-08-13 | | Method: | X-RAY DIFFRACTION (2.1 Å) | | Cite: | Fluorescent binding assay for allosteric ligands of liver pyruvate kinase.
Eur.J.Med.Chem., 298, 2025
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9R3M
 | | Structure of liver pyruvate kinase in complex with fluorescent probe 8a | | Descriptor: | 1,6-di-O-phosphono-beta-D-fructofuranose, 4-[4-[(7-piperidin-1-yl-2,1,3-benzoxadiazol-4-yl)sulfonyl]piperazin-1-yl]sulfonylbenzene-1,2-diol, Isoform L-type of Pyruvate kinase PKLR, ... | | Authors: | Bogucka, A, Nilsson, O, Grotli, M, Hyvonen, M. | | Deposit date: | 2025-05-05 | | Release date: | 2025-08-13 | | Method: | X-RAY DIFFRACTION (2.062 Å) | | Cite: | Fluorescent binding assay for allosteric ligands of liver pyruvate kinase.
Eur.J.Med.Chem., 298, 2025
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9R3O
 | | Structure of liver pyruvate kinase in complex with fluorescent probe 4a | | Descriptor: | 1,6-di-O-phosphono-beta-D-fructofuranose, 4-[4-[[7-(dimethylamino)-2,1,3-benzoxadiazol-4-yl]sulfonyl]piperazin-1-yl]sulfonylbenzene-1,2-diol, Isoform L-type of Pyruvate kinase PKLR, ... | | Authors: | Bogucka, A, Nilsson, O, Grotli, M, Hyvonen, M. | | Deposit date: | 2025-05-05 | | Release date: | 2025-08-13 | | Method: | X-RAY DIFFRACTION (2.045 Å) | | Cite: | Fluorescent binding assay for allosteric ligands of liver pyruvate kinase.
Eur.J.Med.Chem., 298, 2025
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