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3IQH
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Structure of O-Acetylserine Sulfhydrylase in Complex with Peptide MNYDI
分子名称: Cysteine synthase, MNYDI, SULFATE ION
著者Roderick, S.L.
登録日2009-08-20
公開日2009-11-17
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Design of o-acetylserine sulfhydrylase inhibitors by mimicking nature.
J.Med.Chem., 53, 2010
5VR9
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CH1/Ckappa Fab based on Matuzumab
分子名称: CH1/Ckappa Fab heavy chain, CH1/Ckappa Fab light chain
著者Hendle, J.
登録日2017-05-10
公開日2017-08-02
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Computational design of a specific heavy chain/ kappa light chain interface for expressing fully IgG bispecific antibodies.
Protein Sci., 26, 2017
3IWR
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Crystal structure of class I chitinase from Oryza sativa L. japonica
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, Chitinase
著者Kezuka, Y, Watanabe, T, Nonaka, T.
登録日2009-09-03
公開日2010-04-21
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献Structure of full-length class I chitinase from rice revealed by X-ray crystallography and small-angle X-ray scattering.
Proteins, 78, 2010
4ZFU
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BU of 4zfu by Molmil
Structural studies on a non-toxic homologue of type II RIPs from Momordica charantia (bitter gourd) in complex with N-acetyl D galactosamine
分子名称: 2-acetamido-2-deoxy-alpha-D-galactopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Chandran, T, Sharma, A, Vijayan, M.
登録日2015-04-21
公開日2016-03-23
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.53 Å)
主引用文献Structural studies on a non-toxic homologue of type II RIPs from bitter gourd: Molecular basis of non-toxicity, conformational selection and glycan structure.
J.Biosci., 40, 2015
6KDJ
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BU of 6kdj by Molmil
HIV-1 reverse transcriptase with Q151M/Y115F/F116Y:DNA:lamivudine 5'-triphosphate ternary complex
分子名称: DNA/RNA (38-MER), GLYCEROL, HIV-1 RT p51 subunit, ...
著者Yasutake, Y, Hattori, S.I, Tamura, N, Maeda, K.
登録日2019-07-02
公開日2020-03-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.51 Å)
主引用文献Structural features in common of HBV and HIV-1 resistance against chirally-distinct nucleoside analogues entecavir and lamivudine.
Sci Rep, 10, 2020
1AQV
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GLUTATHIONE S-TRANSFERASE IN COMPLEX WITH P-BROMOBENZYLGLUTATHIONE
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, GLUTATHIONE S-TRANSFERASE, N-[(4S)-4-ammonio-4-carboxybutanoyl]-S-(4-bromobenzyl)-L-cysteinylglycine
著者Prade, L, Huber, R, Manoharan, T.H, Fahl, W.E, Reuter, W.
登録日1997-08-01
公開日1997-12-24
最終更新日2024-02-07
実験手法X-RAY DIFFRACTION (1.94 Å)
主引用文献Structures of class pi glutathione S-transferase from human placenta in complex with substrate, transition-state analogue and inhibitor.
Structure, 5, 1997
5W4R
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BU of 5w4r by Molmil
Structure of RORgt bound to a tertiary alcohol
分子名称: 1-{4-[(R)-(4-chloro-2-methoxy-3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}quinolin-6-yl)(hydroxy)(1-methyl-1H-imidazol-5-yl)methyl]piperidin-1-yl}ethan-1-one, Nuclear receptor ROR-gamma
著者Spurlino, J.
登録日2017-06-12
公開日2017-12-27
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (3.002 Å)
主引用文献6-Substituted quinolines as ROR gamma t inverse agonists.
Bioorg. Med. Chem. Lett., 27, 2017
5VXH
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Crystal structure of Xanthomonas campestris OleA E117D
分子名称: 3-oxoacyl-[ACP] synthase III, GLYCEROL, PHOSPHATE ION
著者Jensen, M.R, Wilmot, C.M.
登録日2017-05-23
公開日2017-10-25
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.84 Å)
主引用文献OleA Glu117 is key to condensation of two fatty-acyl coenzyme A substrates in long-chain olefin biosynthesis.
Biochem. J., 474, 2017
3KQ0
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BU of 3kq0 by Molmil
Crystal structure of human alpha1-acid glycoprotein
分子名称: (2R)-2,3-dihydroxypropyl acetate, Alpha-1-acid glycoprotein 1, CHLORIDE ION
著者Schiefner, A, Schonfeld, D.L, Ravelli, R.B.G, Mueller, U, Skerra, A.
登録日2009-11-17
公開日2010-02-02
最終更新日2019-12-25
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献The 1.8-A crystal structure of alpha1-acid glycoprotein (Orosomucoid) solved by UV RIP reveals the broad drug-binding activity of this human plasma lipocalin.
J.Mol.Biol., 384, 2008
5VSK
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Structure of DUB complex
分子名称: 7-chloro-3-({4-hydroxy-1-[(3S)-3-phenylbutanoyl]piperidin-4-yl}methyl)quinazolin-4(3H)-one, Ubiquitin carboxyl-terminal hydrolase 7, ZINC ION
著者Seo, H.-Y, Dhe-Paganon, S.
登録日2017-05-11
公開日2017-12-20
最終更新日2018-01-03
実験手法X-RAY DIFFRACTION (3.33 Å)
主引用文献Structure-Guided Development of a Potent and Selective Non-covalent Active-Site Inhibitor of USP7.
Cell Chem Biol, 24, 2017
2G8A
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BU of 2g8a by Molmil
Lactobacillus casei Y261M in complex with substrate, dUMP
分子名称: 2'-DEOXYURIDINE 5'-MONOPHOSPHATE, thymidylate synthase
著者Finer-Moore, J.S, Stroud, R.M.
登録日2006-03-02
公開日2006-03-14
最終更新日2024-02-14
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献The role of protein dynamics in thymidylate synthase catalysis: variants of conserved 2'-deoxyuridine 5'-monophosphate (dUMP)-binding Tyr-261
Biochemistry, 45, 2006
5VXF
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BU of 5vxf by Molmil
Crystal structure of Xanthomonas campestris OleA E117Q
分子名称: 3-oxoacyl-[ACP] synthase III, GLYCEROL
著者Jensen, M.R, Wilmot, C.M.
登録日2017-05-23
公開日2017-10-25
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献OleA Glu117 is key to condensation of two fatty-acyl coenzyme A substrates in long-chain olefin biosynthesis.
Biochem. J., 474, 2017
3BS2
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BU of 3bs2 by Molmil
Crystal Structure of Monomine
分子名称: GLYCEROL, Lipocalin
著者Mans, B.J, Ribeiro, J.M, Andersen, J.F.
登録日2007-12-21
公開日2008-04-01
最終更新日2017-10-25
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Structure, function, and evolution of biogenic amine-binding proteins in soft ticks.
J.Biol.Chem., 283, 2008
5T8Q
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Crystal structure of murine NF-kappaB inducing kinase (NIK) bound to aryl pyrrole fragment 17
分子名称: 1-[(2-chlorophenyl)methyl]pyrrole-2-carboxamide, Mitogen-activated protein kinase kinase kinase 14, SULFATE ION
著者Smith, M.A, McEwan, P.A, Hymowitz, S.G.
登録日2016-09-08
公開日2017-01-11
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.63 Å)
主引用文献Structure-Based Design of Tricyclic NF-kappa B Inducing Kinase (NIK) Inhibitors That Have High Selectivity over Phosphoinositide-3-kinase (PI3K).
J. Med. Chem., 60, 2017
3L27
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BU of 3l27 by Molmil
Crystal structure of Zaire Ebola VP35 interferon inhibitory domain R312A mutant
分子名称: CHLORIDE ION, GLYCEROL, PHOSPHATE ION, ...
著者Leung, D.W, Prins, K.C, Borek, D.M, Farahbakhsh, M, Tufariello, J.M, Ramanan, P, Nix, J.C, Helgeson, L.A, Otwinowski, Z, Honzatko, R.B, Basler, C.F, Amarasinghe, G.K.
登録日2009-12-14
公開日2010-01-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structural basis for dsRNA recognition and interferon antagonism by Ebola VP35.
Nat.Struct.Mol.Biol., 17, 2010
3L26
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Crystal structure of Zaire Ebola VP35 interferon inhibitory domain bound to 8 bp dsRNA
分子名称: CHLORIDE ION, MAGNESIUM ION, Polymerase cofactor VP35, ...
著者Leung, D.W, Prins, K.C, Borek, D.M, Farahbakhsh, M, Tufariello, J.M, Ramanan, P, Nix, J.C, Helgeson, L.A, Otwinowski, Z, Honzatko, R.B, Basler, C.F, Amarasinghe, G.K.
登録日2009-12-14
公開日2010-01-26
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Structural basis for dsRNA recognition and interferon antagonism by Ebola VP35.
Nat.Struct.Mol.Biol., 17, 2010
1I6G
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BU of 1i6g by Molmil
NMR SOLUTION STRUCTURE OF THE INSECT-SPECIFIC NEUROTOXIN VARIANT 5 (CSE-V5) FROM THE SCORPION CENTRUROIDES SCULPTURATUS EWING
分子名称: NEUROTOXIN V-5
著者Jablonsky, M.J, Jackson, P.L, Krishna, N.R.
登録日2001-03-02
公開日2001-08-01
最終更新日2022-02-23
実験手法SOLUTION NMR
主引用文献Solution structure of an insect-specific neurotoxin from the New World scorpion Centruroides sculpturatus Ewing.
Biochemistry, 40, 2001
6KDK
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BU of 6kdk by Molmil
HIV-1 reverse transcriptase with Q151M/Y115F/F116Y:DNA:dCTP ternary complex
分子名称: 2'-DEOXYCYTIDINE-5'-TRIPHOSPHATE, DNA/RNA (38-MER), GLYCEROL, ...
著者Yasutake, Y, Hattori, S.I, Tamura, N, Maeda, K.
登録日2019-07-02
公開日2020-03-04
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (2.56 Å)
主引用文献Structural features in common of HBV and HIV-1 resistance against chirally-distinct nucleoside analogues entecavir and lamivudine.
Sci Rep, 10, 2020
3L9W
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BU of 3l9w by Molmil
KefC C-terminal domain in complex with KefF and GSH
分子名称: ADENOSINE MONOPHOSPHATE, FLAVIN MONONUCLEOTIDE, GLUTATHIONE, ...
著者Roosild, T.P.
登録日2010-01-05
公開日2010-11-17
最終更新日2023-09-06
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Mechanism of ligand-gated potassium efflux in bacterial pathogens.
Proc.Natl.Acad.Sci.USA, 107, 2010
5TIE
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BU of 5tie by Molmil
x-ray structure of acyl-CoA thioesterase I, TesA, mutant M141L/Y145K/L146K at pH 7.5 in complex with octanoic acid
分子名称: Acyl-CoA thioesterase I, OCTANOIC ACID (CAPRYLIC ACID)
著者Thoden, J.B, Holden, H.M, Grisewood, M.J, Hernandez Lozada, N.J, Gifford, N.P, Mendez-Perez, D, Schoenberger, H.A, Allan, M.F, Pfleger, B.F, Marines, C.D.
登録日2016-10-02
公開日2017-04-26
最終更新日2023-10-04
実験手法X-RAY DIFFRACTION (1.15 Å)
主引用文献Computational Redesign of Acyl-ACP Thioesterase with Improved Selectivity toward Medium-Chain-Length Fatty Acids.
ACS Catal, 7, 2017
3LDY
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BU of 3ldy by Molmil
An extraordinary mechanism of DNA perturbation exhibited by the rare-cutting HNH restriction endonuclease PacI
分子名称: CALCIUM ION, DNA (5'-D(*GP*AP*GP*GP*CP*TP*TP*A)-3'), DNA (5'-D(P*AP*TP*TP*AP*AP*GP*CP*CP*TP*C)-3'), ...
著者Shen, B.W, Heiter, D, Chan, S.-H, Xu, S.-Y, Wilson, G, Stoddard, B.L.
登録日2010-01-13
公開日2010-04-21
最終更新日2024-02-21
実験手法X-RAY DIFFRACTION (1.97 Å)
主引用文献Unusual target site disruption by the rare-cutting HNH restriction endonuclease PacI.
Structure, 18, 2010
2Q4W
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Ensemble refinement of the protein crystal structure of cytokinin oxidase/dehydrogenase (CKX) from Arabidopsis thaliana At5g21482
分子名称: Cytokinin dehydrogenase 7, FLAVIN-ADENINE DINUCLEOTIDE
著者Levin, E.J, Kondrashov, D.A, Wesenberg, G.E, Phillips Jr, G.N, Center for Eukaryotic Structural Genomics (CESG)
登録日2007-05-31
公開日2007-06-19
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Crystal structure of Arabidopsis thaliana cytokinin dehydrogenase.
Proteins, 70, 2008
5U92
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Crystal Structure of arginine kinase from the spider Polybetes pythagoricus in complex with arginine
分子名称: ARGININE, SODIUM ION, arginine kinase
著者Lopez-zavala, A.A, Garcia, C.F, Paredes-Hernandez, J, Stojanoff, V, Sotelo-Mundo, R.R.
登録日2016-12-15
公開日2017-09-06
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Biochemical and structural characterization of a novel arginine kinase from the spider Polybetes pythagoricus.
PeerJ, 5, 2017
1DE7
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INTERACTION OF FACTOR XIII ACTIVATION PEPTIDE WITH ALPHA-THROMBIN: CRYSTAL STRUCTURE OF THE ENZYME-SUBSTRATE COMPLEX
分子名称: ALPHA-THROMBIN (HEAVY CHAIN), ALPHA-THROMBIN (LIGHT CHAIN), FACTOR XIII ACTIVATION PEPTIDE (28-37), ...
著者Sadasivan, C, Yee, V.C.
登録日1999-11-13
公開日2000-12-13
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Interaction of the factor XIII activation peptide with alpha -thrombin. Crystal structure of its enzyme-substrate analog complex.
J.Biol.Chem., 275, 2000
5TQQ
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Cryo-electron microscopy structure of a bovine CLC-K chloride channel, main (class 1) conformation
分子名称: Chloride channel protein, Monoclonal antibody, Fab fragment, ...
著者Park, E, MacKinnon, R.
登録日2016-10-24
公開日2017-01-04
最終更新日2019-11-20
実験手法ELECTRON MICROSCOPY (3.76 Å)
主引用文献Structure of a CLC chloride ion channel by cryo-electron microscopy.
Nature, 541, 2017

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