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7P4W
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Crystal structure of alpha-amylase from Aspergillus oryzae in space group I222
分子名称: 2-(N-MORPHOLINO)-ETHANESULFONIC ACID, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-amylase, ...
著者Bellini, D, Gorrec, F.
登録日2021-07-13
公開日2021-08-25
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.28 Å)
主引用文献The FUSION protein crystallization screen.
J.Appl.Crystallogr., 55, 2022
6NO6
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BU of 6no6 by Molmil
K46bE&K114bD mutant ATP-grasp fold of Blastocystis hominis succinyl-CoA synthetase
分子名称: Succinate--CoA ligase [ADP-forming] subunit beta
著者Huang, J, Fraser, M.E.
登録日2019-01-15
公開日2019-07-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (1.911 Å)
主引用文献ATP-specificity of succinyl-CoA synthetase from Blastocystis hominis.
Acta Crystallogr D Struct Biol, 75, 2019
3FHW
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BU of 3fhw by Molmil
Crystal structure of the protein priB from Bordetella parapertussis. Northeast Structural Genomics Consortium target BpR162.
分子名称: DI(HYDROXYETHYL)ETHER, Primosomal replication protein n, SODIUM ION
著者Kuzin, A.P, Neely, H, Seetharaman, J, Forouhar, F, Wang, D, Mao, L, Maglaqui, M, Xiao, R, Liu, J, Baran, M.C, Acton, T.B, Rost, B, Montelione, G.T, Hunt, J.F, Tong, L, Northeast Structural Genomics Consortium (NESG)
登録日2008-12-10
公開日2008-12-30
最終更新日2017-11-01
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Crystal structure of the protein priB from Bordetella parapertussis. Northeast Structural Genomics Consortium target BpR162.
To be Published
6NO1
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BU of 6no1 by Molmil
ADP bound to K46bE mutant ATP-grasp fold of Blastocystis hominis succinyl-CoA synthetase
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Succinate--CoA ligase [ADP-forming] subunit beta
著者Huang, J, Fraser, M.E.
登録日2019-01-15
公開日2019-07-17
最終更新日2020-01-08
実験手法X-RAY DIFFRACTION (2.44 Å)
主引用文献ATP-specificity of succinyl-CoA synthetase from Blastocystis hominis.
Acta Crystallogr D Struct Biol, 75, 2019
6H0C
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BU of 6h0c by Molmil
Flv1 flavodiiron core from Synechocystis sp. PCC6803
分子名称: CHLORIDE ION, CITRATE ANION, Putative diflavin flavoprotein A 3
著者Borges, P.T, Romao, C.V, Saraiva, L, Goncalves, V.L, Carrondo, M.A, Teixeira, M, Frazao, C.
登録日2018-07-08
公開日2019-01-30
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.592 Å)
主引用文献Analysis of a new flavodiiron core structural arrangement in Flv1-Delta FlR protein from Synechocystis sp. PCC6803.
J. Struct. Biol., 205, 2019
7CGC
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BU of 7cgc by Molmil
Silver-bound E. coli Malate dehydrogenase (C113 and C251)
分子名称: Malate dehydrogenase, SILVER ION
著者Wang, H, Wang, M, Sun, H.
登録日2020-07-01
公開日2020-09-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.548 Å)
主引用文献Atomic differentiation of silver binding preference in protein targets: Escherichia coli malate dehydrogenase as a paradigm.
Chem Sci, 11, 2020
6NO4
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BU of 6no4 by Molmil
ADP bound to L227bF mutant ATP-grasp fold of Blastocystis hominis succinyl-CoA synthetase
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Succinate--CoA ligase [ADP-forming] subunit beta
著者Huang, J, Fraser, M.E.
登録日2019-01-15
公開日2019-07-17
最終更新日2020-01-08
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献ATP-specificity of succinyl-CoA synthetase from Blastocystis hominis.
Acta Crystallogr D Struct Biol, 75, 2019
7CGD
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BU of 7cgd by Molmil
Silver-bound E.coli malate dehydrogenase
分子名称: Malate dehydrogenase, SILVER ION
著者Wang, H, Wang, M, Sun, H.
登録日2020-07-01
公開日2020-09-23
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.06 Å)
主引用文献Atomic differentiation of silver binding preference in protein targets: Escherichia coli malate dehydrogenase as a paradigm.
Chem Sci, 11, 2020
7CGV
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BU of 7cgv by Molmil
Full consensus L-threonine 3-dehydrogenase, FcTDH-IIYM (NAD+ bound form)
分子名称: Artificial L-threonine 3-dehydrogenase, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
著者Motoyama, T, Hiramatsu, N, Asano, Y, Nakano, S, Ito, S.
登録日2020-07-02
公開日2020-10-28
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Protein Sequence Selection Method That Enables Full Consensus Design of Artificial l-Threonine 3-Dehydrogenases with Unique Enzymatic Properties.
Biochemistry, 59, 2020
6H8S
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BU of 6h8s by Molmil
CRYSTAL STRUCTURE OF THE MOUSE PROTEIN TYROSINE PHOSPHATASE PTPN5 (STEP) IN COMPLEX WITH COMPOUND BI-0314
分子名称: 1-[3-piperidin-4-yl-5-(trifluoromethyl)phenyl]guanidine, Tyrosine-protein phosphatase non-receptor type 5
著者Fiegen, D, Schnapp, G.
登録日2018-08-03
公開日2018-09-26
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.771 Å)
主引用文献Allosteric Activation of Striatal-Enriched Protein Tyrosine Phosphatase (STEP, PTPN5) by a Fragment-like Molecule.
J. Med. Chem., 62, 2019
6NO5
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BU of 6no5 by Molmil
ADP bound to K46bE&K114bD mutant ATP-grasp fold of Blastocystis hominis succinyl-CoA synthetase
分子名称: ADENOSINE-5'-DIPHOSPHATE, AMMONIUM ION, MAGNESIUM ION, ...
著者Huang, J, Fraser, M.E.
登録日2019-01-15
公開日2019-07-17
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.069 Å)
主引用文献ATP-specificity of succinyl-CoA synthetase from Blastocystis hominis.
Acta Crystallogr D Struct Biol, 75, 2019
6NO0
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BU of 6no0 by Molmil
ADP bound to ATP-grasp fold of Blastocystis hominis succinyl-CoA synthetase
分子名称: ADENOSINE-5'-DIPHOSPHATE, CHLORIDE ION, MAGNESIUM ION, ...
著者Huang, J, Fraser, M.E.
登録日2019-01-15
公開日2019-07-17
最終更新日2020-01-08
実験手法X-RAY DIFFRACTION (2.209 Å)
主引用文献ATP-specificity of succinyl-CoA synthetase from Blastocystis hominis.
Acta Crystallogr D Struct Biol, 75, 2019
7CND
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BU of 7cnd by Molmil
NCI-1 in complex with CRM1-Ran-RanBP1
分子名称: 3[N-MORPHOLINO]PROPANE SULFONIC ACID, CHLORIDE ION, CRM1 isoform 1, ...
著者Sun, Q, Lei, Y.
登録日2020-07-31
公開日2021-06-09
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Structure-Guided Design of the First Noncovalent Small-Molecule Inhibitor of CRM1.
J.Med.Chem., 64, 2021
7OWQ
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BU of 7owq by Molmil
HsNMT1 in complex with both MyrCoA and peptide N-Methylated-GNCFSKPR
分子名称: Glycylpeptide N-tetradecanoyltransferase 1, MGY-ASN-CYS-PHE-SER-LYS-PRO-ARG, TETRADECANOYL-COA
著者Dian, C, Giglione, C, Meinnel, T.
登録日2021-06-18
公開日2022-12-21
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural and Large-scale Analysis Unveil the Intertwined Paths Promoting NMT-catalyzed Lysine and Glycine Myristoylation.
J.Mol.Biol., 434, 2022
7OWR
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BU of 7owr by Molmil
HsNMT1 in complex with both MyrCoA and peptide GGKSFSKPR
分子名称: GLY-GLY-LYS-SER-PHE-SER-LYS-PRO-ARG, GLYCEROL, Glycylpeptide N-tetradecanoyltransferase 1, ...
著者Dian, C, Giglione, C, Meinnel, T.
登録日2021-06-18
公開日2022-12-21
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.39 Å)
主引用文献Structural and Large-scale Analysis Unveil the Intertwined Paths Promoting NMT-catalyzed Lysine and Glycine Myristoylation.
J.Mol.Biol., 434, 2022
7PHP
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BU of 7php by Molmil
Structure of Multidrug and Toxin Compound Extrusion (MATE) transporter NorM by NabFab-fiducial assisted cryo-EM
分子名称: Anti-Fab nanobody, Multidrug resistance protein NorM, NabFab HC, ...
著者Bloch, J.S, Mukherjee, S, Kowal, J, Niederer, M, Pardon, E, Steyaert, J, Kossiakoff, A.A, Locher, K.P.
登録日2021-08-18
公開日2021-09-01
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (3.47 Å)
主引用文献Development of a universal nanobody-binding Fab module for fiducial-assisted cryo-EM studies of membrane proteins.
Proc.Natl.Acad.Sci.USA, 118, 2021
7PIJ
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BU of 7pij by Molmil
Structure of Staphylococcus capitis divalent metal ion transporter (DMT) by NabFab-fiducial assisted cryo-EM
分子名称: Anti-Fab nanobody, DMTNb16_4, Divalent metal cation transporter MntH, ...
著者Bloch, J.S, Mukherjee, S, Kowal, J, Kossiakoff, A.A, Locher, K.P.
登録日2021-08-20
公開日2021-09-01
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (3.78 Å)
主引用文献Development of a universal nanobody-binding Fab module for fiducial-assisted cryo-EM studies of membrane proteins.
Proc.Natl.Acad.Sci.USA, 118, 2021
7PHQ
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BU of 7phq by Molmil
Structure of homo-dimeric Staphylococcus capitis divalent metal ion transporter (DMT) by NabFab-fiducial assisted cryo-EM
分子名称: Anti-Fab nanobody, DMT-Nb16_4, Divalent metal cation transporter MntH, ...
著者Bloch, J.S, Mukherjee, S, Kowal, J, Kossiakoff, A.A, Locher, K.P.
登録日2021-08-18
公開日2021-09-01
最終更新日2021-12-01
実験手法ELECTRON MICROSCOPY (8.45 Å)
主引用文献Development of a universal nanobody-binding Fab module for fiducial-assisted cryo-EM studies of membrane proteins.
Proc.Natl.Acad.Sci.USA, 118, 2021
7PDC
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BU of 7pdc by Molmil
The structure of the human tetrameric LL-37 peptide in a channel conformation
分子名称: CHLORIDE ION, Cathelicidin antimicrobial peptide
著者Zeth, K, Sancho-Vaello, E.
登録日2021-08-05
公開日2021-09-08
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.83 Å)
主引用文献The structure of the antimicrobial human cathelicidin LL-37 shows oligomerization and channel formation in the presence of membrane mimics.
Sci Rep, 10, 2020
6O9U
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BU of 6o9u by Molmil
KirBac3.1 at a resolution of 2 Angstroms
分子名称: 1,2-DIOLEOYL-SN-GLYCERO-3-PHOSPHOCHOLINE, 3,3',3''-phosphoryltripropanoic acid, BARIUM ION, ...
著者Gulbis, J.M, Clarke, O.B.
登録日2019-03-15
公開日2020-05-27
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献A constricted opening in Kir channels does not impede potassium conduction.
Nat Commun, 11, 2020
6O5D
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PYOCHELIN
分子名称: GLYCEROL, Neutrophil gelatinase-associated lipocalin, SULFATE ION
著者Rupert, P.B, Strong, R.K, Clifton, M.C, Edwards, T.E, Seattle Structural Genomics Center for Infectious Disease (SSGCID)
登録日2019-03-01
公開日2019-09-11
最終更新日2020-07-29
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Parsing the functional specificity of Siderocalin/Lipocalin 2/NGAL for siderophores and related small-molecule ligands.
J Struct Biol X, 2, 2019
7PKX
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BU of 7pkx by Molmil
Crystal structure of a DyP-type peroxidase from Bacillus subtilis in P3121 space group
分子名称: Deferrochelatase/peroxidase, PROTOPORPHYRIN IX CONTAINING FE
著者Borges, P.T, Rodrigues, C, Silva, D, Taborda, A, Brissos, V, Frazao, C, Martins, L.O.
登録日2021-08-27
公開日2021-10-27
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.491 Å)
主引用文献Loops around the Heme Pocket Have a Critical Role in the Function and Stability of Bs DyP from Bacillus subtilis .
Int J Mol Sci, 22, 2021
6H0D
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BU of 6h0d by Molmil
Metal soaked Flv1 flavodiiron core from Synechocystis sp. PCC6803
分子名称: CHLORIDE ION, Putative diflavin flavoprotein A 3, SULFATE ION
著者Borges, P.T, Romao, C.V, Saraiva, L, Goncalves, V.L, Carrondo, M.A, Teixeira, M, Frazao, C.
登録日2018-07-08
公開日2019-01-30
最終更新日2024-05-15
実験手法X-RAY DIFFRACTION (1.598 Å)
主引用文献Analysis of a new flavodiiron core structural arrangement in Flv1-Delta FlR protein from Synechocystis sp. PCC6803.
J. Struct. Biol., 205, 2019
8BSU
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BU of 8bsu by Molmil
Crystal structure of the kainate receptor GluK3-H523A ligand binding domain in complex with kainate and the positive allosteric modulator BPAM344 at 2.9A resolution
分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, 4-cyclopropyl-7-fluoro-3,4-dihydro-2H-1,2,4-benzothiadiazine 1,1-dioxide, ACETATE ION, ...
著者Venskutonyte, R, Frydenvang, K, Kastrup, J.S.
登録日2022-11-26
公開日2023-12-13
最終更新日2024-07-03
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure.
Febs J., 291, 2024
8BST
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BU of 8bst by Molmil
Crystal structure of the kainate receptor GluK3-H523A ligand binding domain in complex with kainate at 2.7A resolution
分子名称: 3-(CARBOXYMETHYL)-4-ISOPROPENYLPROLINE, ACETATE ION, CHLORIDE ION, ...
著者Venskutonyte, R, Frydenvang, K, Kastrup, J.S.
登録日2022-11-26
公開日2023-12-13
最終更新日2024-04-10
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Small-molecule positive allosteric modulation of homomeric kainate receptors GluK1-3: development of screening assays and insight into GluK3 structure.
Febs J., 291, 2024

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