6SN3
| BamABCDE in MSP1D1 nanodisc ensemble 0-3 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (8.4 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-3 To Be Published
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6SN2
| BamABCDE in MSP1D1 nanodisc ensemble 0-2 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (9.5 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-2 To Be Published
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7AL0
| Crystal Structure of Heymonin, a Novel Frog-derived Peptide | 分子名称: | CHLORIDE ION, Heymonin | 著者 | Kascakova, B, Prudnikova, T, Kuta Smatanova, I, Xu, X. | 登録日 | 2020-10-03 | 公開日 | 2021-04-21 | 最終更新日 | 2021-05-05 | 実験手法 | X-RAY DIFFRACTION (2.2 Å) | 主引用文献 | Characterization and functional analysis of cathelicidin-MH, a novel frog-derived peptide with anti-septicemic properties. Elife, 10, 2021
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4ZSP
| BACE crystal structure with bicyclic aminothiazine inhibitor | 分子名称: | Beta-secretase 1, GLYCEROL, N-[(4aS,6S,8aR)-2-amino-4a,5,6,7,8,8a-hexahydro-4H-3,1-benzothiazin-6-yl]-3-chlorobenzamide | 著者 | Timm, D.E. | 登録日 | 2015-05-13 | 公開日 | 2015-06-10 | 最終更新日 | 2015-06-17 | 実験手法 | X-RAY DIFFRACTION (1.91 Å) | 主引用文献 | Preparation and biological evaluation of conformationally constrained BACE1 inhibitors. Bioorg.Med.Chem., 23, 2015
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6SN5
| BamABCDE in MSP1D1 nanodisc ensemble 0-5 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (9.8 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-5 To Be Published
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5AI0
| Ligand complex structure of soluble epoxide hydrolase | 分子名称: | 4-PHENYL-1,2,5-OXADIAZOL-3-AMINE, BIFUNCTIONAL EPOXIDE HYDROLASE 2, DI(HYDROXYETHYL)ETHER, ... | 著者 | Oster, L, Tapani, S, Xue, Y, Kack, H. | 登録日 | 2015-02-11 | 公開日 | 2015-05-13 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (1.75 Å) | 主引用文献 | Successful Generation of Structural Information for Fragment-Based Drug Discovery. Drug Discov Today, 20, 2015
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6SO8
| BamABCDE in MSP1D1 nanodisc ensemble 1-3 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-29 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (9.8 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 1-3 To Be Published
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6SN4
| BamABCDE in MSP1D1 nanodisc ensemble 0-4 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (9.5 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-4 To Be Published
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7B62
| Crystal structure of SARS-CoV-2 spike protein N-terminal domain in complex with biliverdin | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, BILIVERDINE IX ALPHA, DI(HYDROXYETHYL)ETHER, ... | 著者 | Pye, V.E, Rosa, A, Roustan, C, Cherepanov, P. | 登録日 | 2020-12-07 | 公開日 | 2021-04-28 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.82 Å) | 主引用文献 | SARS-CoV-2 can recruit a heme metabolite to evade antibody immunity. Sci Adv, 7, 2021
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6SOC
| BamABCDE in MSP1D1 nanodisc ensemble 1-5 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-29 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (9 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 1-5 To Be Published
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6SN7
| BamABCDE in MSP1D1 nanodisc ensemble 0-6 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (8.9 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-6 To Be Published
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7AUE
| Melanocortin receptor 4 (MC4R) Gs protein complex | 分子名称: | AMINOSERINE, CALCIUM ION, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ... | 著者 | Degtjarik, O, Israeli, H, Prabahar, V, Shalev-Benami, M. | 登録日 | 2020-11-02 | 公開日 | 2021-04-28 | 最終更新日 | 2023-03-15 | 実験手法 | ELECTRON MICROSCOPY (2.97 Å) | 主引用文献 | Structure reveals the activation mechanism of the MC4 receptor to initiate satiation signaling. Science, 372, 2021
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4ZU0
| Structure of the complex of type 1 ribosome inactivating protein from Momordica balsamina with a nucleotide, cytidine monophosphate at 1.80 A resolution | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, CYTIDINE-5'-MONOPHOSPHATE, GLYCEROL, ... | 著者 | Yamin, S, Pandey, S, Kaur, P, Sharma, S, Singh, T.P. | 登録日 | 2015-05-15 | 公開日 | 2015-06-03 | 最終更新日 | 2023-11-08 | 実験手法 | X-RAY DIFFRACTION (1.8 Å) | 主引用文献 | Binding and structural studies of the complexes of type 1 ribosome inactivating protein fromMomordica balsaminawith cytosine, cytidine, and cytidine diphosphate. Biochem Biophys Rep, 4, 2015
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6SMX
| BamABCDE in MSP1D1 nanodisc | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-23 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (6.65 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc To Be Published
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6SOA
| BamABCDE in MSP1D1 nanodisc ensemble 0-9 | 分子名称: | Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ... | 著者 | Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P. | 登録日 | 2019-08-29 | 公開日 | 2021-03-31 | 最終更新日 | 2024-05-22 | 実験手法 | ELECTRON MICROSCOPY (10.8 Å) | 主引用文献 | BamABCDE in MSP1D1 nanodisc ensemble 0-9 To Be Published
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7AYG
| oxalyl-CoA decarboxylase from Methylorubrum extorquens with bound TPP and ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Putative oxalyl-CoA decarboxylase (Oxc, ... | 著者 | Pfister, P, Burgener, S, Nattermann, M, Zarzycki, J, Erb, T.J. | 登録日 | 2020-11-12 | 公開日 | 2021-04-28 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (1.9 Å) | 主引用文献 | Engineering a Highly Efficient Carboligase for Synthetic One-Carbon Metabolism. Acs Catalysis, 11, 2021
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7B2E
| quadruple mutant of oxalyl-CoA decarboxylase from Methylorubrum extorquens with bound TPP and ADP | 分子名称: | ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Putative oxalyl-CoA decarboxylase (Oxc, ... | 著者 | Pfister, P, Burgener, S, Nattermann, M, Zarzycki, J, Erb, T.J. | 登録日 | 2020-11-26 | 公開日 | 2021-04-28 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | Engineering a Highly Efficient Carboligase for Synthetic One-Carbon Metabolism. Acs Catalysis, 11, 2021
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6JBQ
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5A4L
| DYRK1A IN COMPLEX WITH FLUORO BENZOTHIAZOLE FRAGMENT | 分子名称: | DUAL SPECIFICITY TYROSINE-PHOSPHORYLATION- REGULATED KINASE 1A, N-(5-FLUORANYL-1,3-BENZOTHIAZOL-2-YL)ETHANAMIDE | 著者 | Rothweiler, U. | 登録日 | 2015-06-10 | 公開日 | 2016-06-29 | 最終更新日 | 2024-01-10 | 実験手法 | X-RAY DIFFRACTION (2.73 Å) | 主引用文献 | Probing the ATP-Binding Pocket of Protein Kinase Dyrk1A with Benzothiazole Fragment Molecules J.Med.Chem., 59, 2016
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7B2L
| Structure of the endocytic adaptor complex AENTH | 分子名称: | ANTH domain of Sla2, ENTH domain of epsin Ent1, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate | 著者 | Klebl, D.P, Lizarrondo, J, Sobott, F, Garcia-Alai, M, Muench, S.P. | 登録日 | 2020-11-27 | 公開日 | 2021-05-05 | 最終更新日 | 2024-05-01 | 実験手法 | ELECTRON MICROSCOPY (3.9 Å) | 主引用文献 | Structure of the endocytic adaptor complex reveals the basis for efficient membrane anchoring during clathrin-mediated endocytosis. Nat Commun, 12, 2021
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6JQA
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6SWU
| Crystal structure of the TPR domain of KLC1 in complex with an engineered high-affinity cargo peptide. | 分子名称: | 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Kinesin light chain 1,Kinesin light chain 1,TPR domain of kinesin light chain 1 in complex with an engineered high-affinity cargo peptide of sequence TVFTTEDIYEWDDSAI | 著者 | Chegkazi, M.S, Steiner, R.A. | 登録日 | 2019-09-23 | 公開日 | 2020-09-30 | 最終更新日 | 2024-01-24 | 実験手法 | X-RAY DIFFRACTION (2.849 Å) | 主引用文献 | Fragment-linking peptide design yields a high-affinity ligand for microtubule-based transport. Cell Chem Biol, 28, 2021
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7ASW
| Crystal structure of chloroplastic thioredoxin z defines a novel type-specific target recognition | 分子名称: | Thioredoxin-related protein CITRX | 著者 | Le Moigne, T, Gurrieri, L, Crozet, P, Marchand, C.H, Zaffagnini, M, Sparla, F, Lemaire, S.D, Henri, J. | 登録日 | 2020-10-28 | 公開日 | 2021-05-19 | 最終更新日 | 2024-01-31 | 実験手法 | X-RAY DIFFRACTION (2.444 Å) | 主引用文献 | Crystal structure of chloroplastic thioredoxin z defines a type-specific target recognition. Plant J., 107, 2021
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5A4C
| FGFR1 ligand complex | 分子名称: | 1,2-ETHANEDIOL, 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, FIBROBLAST GROWTH FACTOR RECEPTOR 1 (FMS-RELATED TYROSINE KINASE 2, ... | 著者 | Klein, T, Vajpai, N, Phillips, J.J, Davies, G, Holdgate, G.A, Phillips, C, Tucker, J.A, Norman, R.A, Scott, A.S, Higazi, D.R, Lowe, D, Thompson, G.S, Breeze, A.L. | 登録日 | 2015-06-05 | 公開日 | 2015-08-05 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (2.09 Å) | 主引用文献 | Structural and Dynamic Insights Into the Energetics of Activation Loop Rearrangement in Fgfr1 Kinase. Nat.Commun., 6, 2015
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5AGO
| Structure of rat neuronal nitric oxide synthase heme domain in complex with (S)-2-Amino-5-(2-mercaptoacetimidamido)pentanoic acid | 分子名称: | (S)-2-AMINO-5-(2-MERCAPTOACETIMIDAMIDO)PENTANOIC ACID, 5,6,7,8-TETRAHYDROBIOPTERIN, ACETATE ION, ... | 著者 | Li, H, Poulos, T.L. | 登録日 | 2015-02-02 | 公開日 | 2015-04-29 | 最終更新日 | 2024-05-08 | 実験手法 | X-RAY DIFFRACTION (1.902 Å) | 主引用文献 | Mechanism of Inactivation of Neuronal Nitric Oxide Synthase by (S)-2-Amino-5-(2-(Methylthio)Acetimidamido)Pentanoic Acid. J.Am.Chem.Soc., 137, 2015
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