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6SN3
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BU of 6sn3 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-3
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (8.4 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-3
To Be Published
6SN2
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BU of 6sn2 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-2
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (9.5 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-2
To Be Published
7AL0
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BU of 7al0 by Molmil
Crystal Structure of Heymonin, a Novel Frog-derived Peptide
分子名称: CHLORIDE ION, Heymonin
著者Kascakova, B, Prudnikova, T, Kuta Smatanova, I, Xu, X.
登録日2020-10-03
公開日2021-04-21
最終更新日2021-05-05
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Characterization and functional analysis of cathelicidin-MH, a novel frog-derived peptide with anti-septicemic properties.
Elife, 10, 2021
4ZSP
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BU of 4zsp by Molmil
BACE crystal structure with bicyclic aminothiazine inhibitor
分子名称: Beta-secretase 1, GLYCEROL, N-[(4aS,6S,8aR)-2-amino-4a,5,6,7,8,8a-hexahydro-4H-3,1-benzothiazin-6-yl]-3-chlorobenzamide
著者Timm, D.E.
登録日2015-05-13
公開日2015-06-10
最終更新日2015-06-17
実験手法X-RAY DIFFRACTION (1.91 Å)
主引用文献Preparation and biological evaluation of conformationally constrained BACE1 inhibitors.
Bioorg.Med.Chem., 23, 2015
6SN5
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BU of 6sn5 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-5
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (9.8 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-5
To Be Published
5AI0
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BU of 5ai0 by Molmil
Ligand complex structure of soluble epoxide hydrolase
分子名称: 4-PHENYL-1,2,5-OXADIAZOL-3-AMINE, BIFUNCTIONAL EPOXIDE HYDROLASE 2, DI(HYDROXYETHYL)ETHER, ...
著者Oster, L, Tapani, S, Xue, Y, Kack, H.
登録日2015-02-11
公開日2015-05-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献Successful Generation of Structural Information for Fragment-Based Drug Discovery.
Drug Discov Today, 20, 2015
6SO8
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BU of 6so8 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 1-3
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-29
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (9.8 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 1-3
To Be Published
6SN4
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BU of 6sn4 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-4
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (9.5 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-4
To Be Published
7B62
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BU of 7b62 by Molmil
Crystal structure of SARS-CoV-2 spike protein N-terminal domain in complex with biliverdin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, BILIVERDINE IX ALPHA, DI(HYDROXYETHYL)ETHER, ...
著者Pye, V.E, Rosa, A, Roustan, C, Cherepanov, P.
登録日2020-12-07
公開日2021-04-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.82 Å)
主引用文献SARS-CoV-2 can recruit a heme metabolite to evade antibody immunity.
Sci Adv, 7, 2021
6SOC
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BU of 6soc by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 1-5
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-29
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (9 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 1-5
To Be Published
6SN7
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BU of 6sn7 by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-6
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (8.9 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-6
To Be Published
7AUE
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BU of 7aue by Molmil
Melanocortin receptor 4 (MC4R) Gs protein complex
分子名称: AMINOSERINE, CALCIUM ION, Guanine nucleotide-binding protein G(I)/G(S)/G(O) subunit gamma-2, ...
著者Degtjarik, O, Israeli, H, Prabahar, V, Shalev-Benami, M.
登録日2020-11-02
公開日2021-04-28
最終更新日2023-03-15
実験手法ELECTRON MICROSCOPY (2.97 Å)
主引用文献Structure reveals the activation mechanism of the MC4 receptor to initiate satiation signaling.
Science, 372, 2021
4ZU0
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BU of 4zu0 by Molmil
Structure of the complex of type 1 ribosome inactivating protein from Momordica balsamina with a nucleotide, cytidine monophosphate at 1.80 A resolution
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CYTIDINE-5'-MONOPHOSPHATE, GLYCEROL, ...
著者Yamin, S, Pandey, S, Kaur, P, Sharma, S, Singh, T.P.
登録日2015-05-15
公開日2015-06-03
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Binding and structural studies of the complexes of type 1 ribosome inactivating protein fromMomordica balsaminawith cytosine, cytidine, and cytidine diphosphate.
Biochem Biophys Rep, 4, 2015
6SMX
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BU of 6smx by Molmil
BamABCDE in MSP1D1 nanodisc
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-23
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (6.65 Å)
主引用文献BamABCDE in MSP1D1 nanodisc
To Be Published
6SOA
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BU of 6soa by Molmil
BamABCDE in MSP1D1 nanodisc ensemble 0-9
分子名称: Outer membrane protein assembly factor BamA, Outer membrane protein assembly factor BamB, Outer membrane protein assembly factor BamC, ...
著者Iadanza, M.G, Ranson, N.A, Radford, S.E, Higgins, A.J, Calabrese, A.N, Schiffrin, B, White, P.
登録日2019-08-29
公開日2021-03-31
最終更新日2024-05-22
実験手法ELECTRON MICROSCOPY (10.8 Å)
主引用文献BamABCDE in MSP1D1 nanodisc ensemble 0-9
To Be Published
7AYG
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BU of 7ayg by Molmil
oxalyl-CoA decarboxylase from Methylorubrum extorquens with bound TPP and ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Putative oxalyl-CoA decarboxylase (Oxc, ...
著者Pfister, P, Burgener, S, Nattermann, M, Zarzycki, J, Erb, T.J.
登録日2020-11-12
公開日2021-04-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献Engineering a Highly Efficient Carboligase for Synthetic One-Carbon Metabolism.
Acs Catalysis, 11, 2021
7B2E
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BU of 7b2e by Molmil
quadruple mutant of oxalyl-CoA decarboxylase from Methylorubrum extorquens with bound TPP and ADP
分子名称: ADENOSINE-5'-DIPHOSPHATE, MAGNESIUM ION, Putative oxalyl-CoA decarboxylase (Oxc, ...
著者Pfister, P, Burgener, S, Nattermann, M, Zarzycki, J, Erb, T.J.
登録日2020-11-26
公開日2021-04-28
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.8 Å)
主引用文献Engineering a Highly Efficient Carboligase for Synthetic One-Carbon Metabolism.
Acs Catalysis, 11, 2021
6JBQ
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BU of 6jbq by Molmil
CryoEM structure of Escherichia coli sigmaE transcription initiation complex containing 5nt of RNA
分子名称: DNA (48-MER), DNA-directed RNA polymerase subunit alpha, DNA-directed RNA polymerase subunit beta, ...
著者Fang, C.L, Zhang, Y.
登録日2019-01-26
公開日2019-05-29
最終更新日2024-03-27
実験手法ELECTRON MICROSCOPY (4.02 Å)
主引用文献Structures and mechanism of transcription initiation by bacterial ECF factors.
Nucleic Acids Res., 47, 2019
5A4L
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BU of 5a4l by Molmil
DYRK1A IN COMPLEX WITH FLUORO BENZOTHIAZOLE FRAGMENT
分子名称: DUAL SPECIFICITY TYROSINE-PHOSPHORYLATION- REGULATED KINASE 1A, N-(5-FLUORANYL-1,3-BENZOTHIAZOL-2-YL)ETHANAMIDE
著者Rothweiler, U.
登録日2015-06-10
公開日2016-06-29
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.73 Å)
主引用文献Probing the ATP-Binding Pocket of Protein Kinase Dyrk1A with Benzothiazole Fragment Molecules
J.Med.Chem., 59, 2016
7B2L
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BU of 7b2l by Molmil
Structure of the endocytic adaptor complex AENTH
分子名称: ANTH domain of Sla2, ENTH domain of epsin Ent1, [(2R)-2-octanoyloxy-3-[oxidanyl-[(1R,2R,3S,4R,5R,6S)-2,3,6-tris(oxidanyl)-4,5-diphosphonooxy-cyclohexyl]oxy-phosphoryl]oxy-propyl] octanoate
著者Klebl, D.P, Lizarrondo, J, Sobott, F, Garcia-Alai, M, Muench, S.P.
登録日2020-11-27
公開日2021-05-05
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.9 Å)
主引用文献Structure of the endocytic adaptor complex reveals the basis for efficient membrane anchoring during clathrin-mediated endocytosis.
Nat Commun, 12, 2021
6JQA
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BU of 6jqa by Molmil
Crystal structure of phyllogen, a phyllody inducing effector protein of phytoplasma.
分子名称: IODIDE ION, Phytoplasmal effector causing phyllody 1
著者Miyatake, H, Maejima, K.
登録日2019-03-29
公開日2019-05-15
最終更新日2019-05-29
実験手法X-RAY DIFFRACTION (2.402 Å)
主引用文献Crystal structure of phyllogen, a phyllody-inducing effector protein of phytoplasma.
Biochem.Biophys.Res.Commun., 513, 2019
6SWU
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BU of 6swu by Molmil
Crystal structure of the TPR domain of KLC1 in complex with an engineered high-affinity cargo peptide.
分子名称: 1,2-ETHANEDIOL, DI(HYDROXYETHYL)ETHER, Kinesin light chain 1,Kinesin light chain 1,TPR domain of kinesin light chain 1 in complex with an engineered high-affinity cargo peptide of sequence TVFTTEDIYEWDDSAI
著者Chegkazi, M.S, Steiner, R.A.
登録日2019-09-23
公開日2020-09-30
最終更新日2024-01-24
実験手法X-RAY DIFFRACTION (2.849 Å)
主引用文献Fragment-linking peptide design yields a high-affinity ligand for microtubule-based transport.
Cell Chem Biol, 28, 2021
7ASW
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BU of 7asw by Molmil
Crystal structure of chloroplastic thioredoxin z defines a novel type-specific target recognition
分子名称: Thioredoxin-related protein CITRX
著者Le Moigne, T, Gurrieri, L, Crozet, P, Marchand, C.H, Zaffagnini, M, Sparla, F, Lemaire, S.D, Henri, J.
登録日2020-10-28
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.444 Å)
主引用文献Crystal structure of chloroplastic thioredoxin z defines a type-specific target recognition.
Plant J., 107, 2021
5A4C
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BU of 5a4c by Molmil
FGFR1 ligand complex
分子名称: 1,2-ETHANEDIOL, 1-tert-butyl-3-[2-[3-(diethylamino)propylamino]-6-(3,5-dimethoxyphenyl)pyrido[2,3-d]pyrimidin-7-yl]urea, FIBROBLAST GROWTH FACTOR RECEPTOR 1 (FMS-RELATED TYROSINE KINASE 2, ...
著者Klein, T, Vajpai, N, Phillips, J.J, Davies, G, Holdgate, G.A, Phillips, C, Tucker, J.A, Norman, R.A, Scott, A.S, Higazi, D.R, Lowe, D, Thompson, G.S, Breeze, A.L.
登録日2015-06-05
公開日2015-08-05
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (2.09 Å)
主引用文献Structural and Dynamic Insights Into the Energetics of Activation Loop Rearrangement in Fgfr1 Kinase.
Nat.Commun., 6, 2015
5AGO
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BU of 5ago by Molmil
Structure of rat neuronal nitric oxide synthase heme domain in complex with (S)-2-Amino-5-(2-mercaptoacetimidamido)pentanoic acid
分子名称: (S)-2-AMINO-5-(2-MERCAPTOACETIMIDAMIDO)PENTANOIC ACID, 5,6,7,8-TETRAHYDROBIOPTERIN, ACETATE ION, ...
著者Li, H, Poulos, T.L.
登録日2015-02-02
公開日2015-04-29
最終更新日2024-05-08
実験手法X-RAY DIFFRACTION (1.902 Å)
主引用文献Mechanism of Inactivation of Neuronal Nitric Oxide Synthase by (S)-2-Amino-5-(2-(Methylthio)Acetimidamido)Pentanoic Acid.
J.Am.Chem.Soc., 137, 2015

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件を2024-09-25に公開中

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