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5OQJ
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BU of 5oqj by Molmil
STRUCTURE OF YEAST TRANSCRIPTION PRE-INITIATION COMPLEX WITH TFIIH
分子名称: DNA repair helicase RAD25, DNA repair helicase RAD3, DNA-directed RNA polymerase II subunit RPB1, ...
著者Schilbach, S, Hantsche, M, Tegunov, D, Dienemann, C, Wigge, C, Henning, U, Cramer, P.
登録日2017-08-11
公開日2018-04-25
最終更新日2024-05-15
実験手法ELECTRON MICROSCOPY (4.7 Å)
主引用文献Structures of transcription pre-initiation complex with TFIIH and Mediator.
Nature, 551, 2017
5OWA
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BU of 5owa by Molmil
Crystal structure of the human BRPF1 bromodomain in complex with BZ054
分子名称: Peregrin, ~{N}-[4-[[(3~{S},5~{R})-3,5-dimethylpiperidin-1-yl]methyl]-1,3-thiazol-2-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
著者Zhu, J, Caflisch, A.
登録日2017-08-31
公開日2018-06-27
最終更新日2024-01-17
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献Structure-based discovery of selective BRPF1 bromodomain inhibitors.
Eur J Med Chem, 155, 2018
5OX2
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BU of 5ox2 by Molmil
Crystal structure of thymoligase, a substrate-tailored peptiligase variant
分子名称: Fragment of prodomain, SULFATE ION, Subtilisin BPN'
著者Rozeboom, H.J, Janssen, D.B.
登録日2017-09-05
公開日2018-01-10
最終更新日2018-04-18
実験手法X-RAY DIFFRACTION (2.24 Å)
主引用文献Design of a substrate-tailored peptiligase variant for the efficient synthesis of thymosin-alpha1.
Org. Biomol. Chem., 16, 2018
5SIC
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BU of 5sic by Molmil
MOLECULAR RECOGNITION AT THE ACTIVE SITE OF SUBTILISIN BPN': CRYSTALLOGRAPHIC STUDIES USING GENETICALLY ENGINEERED PROTEINACEOUS INHIBITOR SSI (STREPTOMYCES SUBTILISIN INHIBITOR)
分子名称: CALCIUM ION, SUBTILISIN BPN', SUBTILISIN INHIBITOR (SSI)
著者Mitsui, Y, Takeuchi, Y, Nakamura, K.T.
登録日1991-11-18
公開日1994-01-31
最終更新日2017-11-29
実験手法X-RAY DIFFRACTION (2.2 Å)
主引用文献Molecular recognition at the active site of subtilisin BPN': crystallographic studies using genetically engineered proteinaceous inhibitor SSI (Streptomyces subtilisin inhibitor).
Protein Eng., 4, 1991

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件を2024-09-25に公開中

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