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3U36
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Crystal Structure of PG9 Fab
分子名称: PG9 Fab heavy chain, PG9 Fab light chain, SULFATE ION
著者McLellan, J.S, Kwong, P.D.
登録日2011-10-04
公開日2011-11-30
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (3.281 Å)
主引用文献Structure of HIV-1 gp120 V1/V2 domain with broadly neutralizing antibody PG9.
Nature, 480, 2011
3U4B
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CH04H/CH02L Fab P4
分子名称: CH02 Light chain, CH04 Heavy chain
著者Pancera, M, Louder, R, Mclellan, J.S, KWong, P.D.
登録日2011-10-07
公開日2011-11-30
最終更新日2011-12-21
実験手法X-RAY DIFFRACTION (2.893 Å)
主引用文献Structure of HIV-1 gp120 V1/V2 domain with broadly neutralizing antibody PG9.
Nature, 480, 2011
3B21
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Crystal structure of OspI from Shigella flexineri
分子名称: ORF169b
著者Sanada, T, Kim, M, Sasakawa, C, Mizushima, T.
登録日2011-07-19
公開日2012-02-22
最終更新日2012-04-04
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献The Shigella flexneri effector OspI deamidates UBC13 to dampen the inflammatory response
Nature, 483, 2012
3B1M
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Crystal structure of the PPARgamma-LBD complexed with a cercosporamide derivative modulator Cerco-A
分子名称: (9aS)-8-acetyl-N-[(2-ethylnaphthalen-1-yl)methyl]-1,7-dihydroxy-3-methoxy-9a-methyl-9-oxo-9,9a-dihydrodibenzo[b,d]furan-4-carboxamide, Peroxisome proliferator-activated receptor gamma, Peroxisome proliferator-activated receptor gamma coactivator 1-alpha
著者Matsui, Y, Hiroyuki, H.
登録日2011-07-05
公開日2011-08-24
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.6 Å)
主引用文献Pharmacology and in Vitro Profiling of a Novel Peroxisome Proliferator-Activated Receptor gamma Ligand, Cerco-A
Biol.Pharm.Bull., 34, 2011
3B20
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Crystal structure of Glyceraldehyde-3-Phosphate Dehydrogenase complexed with NADfrom Synechococcus elongatus"
分子名称: Glyceraldehyde 3-phosphate dehydrogenase (NADP+), NICOTINAMIDE-ADENINE-DINUCLEOTIDE, SULFATE ION
著者Matsumura, H, Kai, A, Maeda, T, Inoue, T.
登録日2011-07-17
公開日2012-01-11
最終更新日2024-03-13
実験手法X-RAY DIFFRACTION (2.398 Å)
主引用文献Structure Basis for the Regulation of Glyceraldehyde-3-Phosphate Dehydrogenase Activity via the Intrinsically Disordered Protein CP12.
Structure, 19, 2011
3BLB
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Crystal structure of Golgi Mannosidase II in complex with swainsonine at 1.3 Angstrom resolution
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, 1S-8AB-OCTAHYDRO-INDOLIZIDINE-1A,2A,8B-TRIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Kuntz, D.A, Rose, D.R.
登録日2007-12-10
公開日2008-01-08
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Golgi Mannosidase II in complex with swainsonine at 1.3 Angstrom.
To Be Published
3BUD
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BU of 3bud by Molmil
Golgi mannosidase II D204A catalytic nucleophile mutant with an empty active site
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-mannosidase 2, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-02
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008
3BVX
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GOLGI MANNOSIDASE II D204A catalytic nucleophile mutant complex with Methyl (2-deoxy-2-acetamido-beta-D-glucopyranosyl)-(1->2)-(alpha-D-mannopyranosyl)- (1->3)-[(alpha-D-mannopyranosyl)-(1->6)-(alpha-D-mannopyranosyl)-(1->6)]-beta-D-mannopyranoside
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)-alpha-D-mannopyranose-(1-6)]methyl beta-D-mannopyranoside, Alpha-mannosidase 2, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-07
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.1 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008
3S1Y
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AMP-C BETA-LACTAMASE (PSEUDOMONAS AERUGINOSA) in complex with a beta-lactamase inhibitor
分子名称: Beta-lactamase, CHLORIDE ION, ISOPROPYL ALCOHOL, ...
著者Scapin, G, Lu, J, Fitzgerald, P.M.D, Sharma, N.
登録日2011-05-16
公開日2011-06-29
最終更新日2013-06-26
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Side chain SAR of bicyclic Beta-lactamase inhibitors (BLIs). 2. N-Alkylated and open chain analogs of MK-8712
Bioorg.Med.Chem.Lett., 21, 2011
3BUI
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Golgi mannosidase II D204A catalytic nucleophile mutant complex with Tris
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, Alpha-mannosidase 2, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-02
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.25 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008
3BVT
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GOLGI MANNOSIDASE II D204A catalytic nucleophile mutant complex with Methyl (alpha-D-mannopyranosyl)-(1->3)-S-alpha-D-mannopyranoside
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-07
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008
3BWS
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BU of 3bws by Molmil
Crystal structure of the leptospiral antigen Lp49
分子名称: SULFATE ION, protein Lp49
著者Giuseppe, P.O, Neves, F.O, Nascimento, A.L.T.O, Guimaraes, B.G.
登録日2008-01-10
公開日2008-10-07
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (1.99 Å)
主引用文献The leptospiral antigen Lp49 is a two-domain protein with putative protein binding function
J.Struct.Biol., 163, 2008
3U2S
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BU of 3u2s by Molmil
Crystal Structure of PG9 Fab in Complex with V1V2 Region from HIV-1 strain ZM109
分子名称: (R,R)-2,3-BUTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Envelope glycoprotein gp120, ...
著者McLellan, J.S, Pancera, M, Kwong, P.D.
登録日2011-10-04
公開日2011-11-30
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (1.797 Å)
主引用文献Structure of HIV-1 gp120 V1/V2 domain with broadly neutralizing antibody PG9.
Nature, 480, 2011
2ZJ7
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Crystal structure of D157A mutant of Pseudomonas sp. MIS38 lipase
分子名称: CALCIUM ION, Lipase, ZINC ION
著者Angkawidjaja, C, Kuwahara, K, Kanaya, S.
登録日2008-02-29
公開日2008-12-02
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.21 Å)
主引用文献Importance of the Ca2+-binding sites in the N-catalytic domain of a family I.3 lipase for activity and stability
Protein Eng.Des.Sel., 21, 2008
3AIN
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BU of 3ain by Molmil
R267G mutant of a HSL-like carboxylesterase from Sulfolobus tokodaii
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, 303aa long hypothetical esterase, ...
著者Angkawidjaja, C, Kanaya, S.
登録日2010-05-16
公開日2011-06-08
最終更新日2012-09-05
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Structure and stability of a thermostable carboxylesterase from the thermoacidophilic archaeon Sulfolobustokodaii
Febs J., 279, 2012
3AIO
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R267K mutant of a HSL-like carboxylesterase from Sulfolobus tokodaii
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, (4S)-2-METHYL-2,4-PENTANEDIOL, 303aa long hypothetical esterase, ...
著者Angkawidjaja, C, Kanaya, S.
登録日2010-05-16
公開日2011-06-08
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Structure and stability of a thermostable carboxylesterase from the thermoacidophilic archaeon Sulfolobustokodaii
Febs J., 279, 2012
3AM6
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Crystal structure of the proton pumping rhodopsin AR2 from marine alga Acetabularia acetabulum
分子名称: CHOLESTEROL, RETINAL, rhodopsin-2
著者Wada, T, Yokoyama, S.
登録日2010-08-16
公開日2011-07-06
最終更新日2011-12-07
実験手法X-RAY DIFFRACTION (3.2 Å)
主引用文献Crystal structure of the eukaryotic light-driven proton-pumping rhodopsin, Acetabularia rhodopsin II, from marine alga
J.Mol.Biol., 411, 2011
3AH6
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Remarkable improvement of the heat stability of CutA1 from E.coli by rational protein designing
分子名称: Divalent-cation tolerance protein cutA
著者Matsuura, Y, Tanaka, T, Bagautdinov, B, Kunishima, N, Yutani, K.
登録日2010-04-15
公開日2010-08-11
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.4 Å)
主引用文献Remarkable improvement in the heat stability of CutA1 from Escherichia coli by rational protein design
J.Biochem., 148, 2010
3AID
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BU of 3aid by Molmil
A NEW CLASS OF HIV-1 PROTEASE INHIBITOR: THE CRYSTALLOGRAPHIC STRUCTURE, INHIBITION AND CHEMICAL SYNTHESIS OF AN AMINIMIDE PEPTIDE ISOSTERE
分子名称: BENZOYLAMINO-BENZYL-METHYL-[2-HYDROXY-3-[1-METHYL-ETHYL-OXY-N-FORMAMIDYL]-4-PHENYL-BUTYL]-AMMONIUM, HUMAN IMMUNODEFICIENCY VIRUS PROTEASE
著者Rutenber, E.E, Stroud, R.M.
登録日1997-05-15
公開日1997-09-17
最終更新日2024-05-22
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献A new class of HIV-1 protease inhibitor: the crystallographic structure, inhibition and chemical synthesis of an aminimide peptide isostere.
Bioorg.Med.Chem., 4, 1996
2Z21
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Crystal Structure of a five site mutated Cyanovirin-N
分子名称: Cyanovirin-N
著者Fromme, R, Katilene, Z, Fromme, P, Ghirlanda, G.
登録日2007-05-17
公開日2007-07-31
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献A Monovalent Mutant of Cyanovirin-N Provides Insight into the Role of Multiple Interactions with gp120 for Antiviral Activity.
Biochemistry, 46, 2007
3BUB
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BU of 3bub by Molmil
Golgi alpha-mannosidase II with an empty active site
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-mannosidase 2, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-02
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.38 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008
3U4E
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Crystal Structure of PG9 Fab in Complex with V1V2 Region from HIV-1 strain CAP45
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, PG9 Heavy Chain, PG9 Light Chain, ...
著者Gorman, J, McLellan, J, Pancera, M, Kwong, P.D.
登録日2011-10-07
公開日2011-11-30
最終更新日2023-12-06
実験手法X-RAY DIFFRACTION (2.185 Å)
主引用文献Structure of HIV-1 gp120 V1/V2 domain with broadly neutralizing antibody PG9.
Nature, 480, 2011
2ZPN
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The crystal structure of Saccharomyces cerevisiae Atg8- Atg19(412-415) complex
分子名称: Autophagy-related protein 8, SULFATE ION, Saccharomyces cerevisiae Atg19(412-415)
著者Noda, N.N, Inagaki, F.
登録日2008-07-17
公開日2008-12-09
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.7 Å)
主引用文献Structural basis of target recognition by Atg8/LC3 during selective autophagy
Genes Cells, 13, 2008
2ZQB
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Crystal structure of a psychrotrophic RNaseHI variant with sextuple thermostabilizing mutations
分子名称: Ribonuclease HI, SULFATE ION
著者Angkawidjaja, C, Kanaya, S.
登録日2008-08-07
公開日2009-06-23
最終更新日2023-11-01
実験手法X-RAY DIFFRACTION (2.49 Å)
主引用文献Destabilization of psychrotrophic RNase HI in a localized fashion as revealed by mutational and X-ray crystallographic analyses
Febs J., 276, 2009
3BVU
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GOLGI MANNOSIDASE II D204A catalytic nucleophile mutant complex with Methyl(alpha-D-mannopyranosyl)-(1->3)-S-[(alpha-D-mannopyranosyl)-(1->6)]-alpha-D-mannopyranoside
分子名称: (4R)-2-METHYLPENTANE-2,4-DIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose, Alpha-mannosidase 2, ...
著者Kuntz, D.A, Rose, D.R.
登録日2008-01-07
公開日2008-07-01
最終更新日2023-08-30
実験手法X-RAY DIFFRACTION (1.12 Å)
主引用文献Probing the substrate specificity of Golgi alpha-mannosidase II by use of synthetic oligosaccharides and a catalytic nucleophile mutant.
J.Am.Chem.Soc., 130, 2008

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