6B4X
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6B53
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6BZ4
| Human IgG1 lacking complement-dependent cytotoxicity: hu3S193 Fc mutant K322A | 分子名称: | 1,2-ETHANEDIOL, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)-[alpha-D-mannopyranose-(1-3)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Farrugia, W, Burvenich, I.G.J, Scott, A.M, Ramsland, P.A. | 登録日 | 2017-12-22 | 公開日 | 2018-06-13 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.4 Å) | 主引用文献 | Global conformational changes in IgG-Fc upon mutation of the FcRn-binding site are not associated with altered antibody-dependent effector functions. Biochem. J., 475, 2018
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7SJB
| Crystal structure of dehaloperoxidase B in complex with alpha-terpinene | 分子名称: | 1-methyl-4-(propan-2-yl)cyclohexa-1,3-diene, Dehaloperoxidase B, GLYCEROL, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Malewschik, T, Yun, D. | 登録日 | 2021-10-17 | 公開日 | 2022-11-23 | 最終更新日 | 2023-10-18 | 実験手法 | X-RAY DIFFRACTION (1.718 Å) | 主引用文献 | The Multifunctional Globin Dehaloperoxidase as a Biocatalyst in the Oxidation of Monoterpenes To Be Published
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7SJE
| Crystal structure of dehaloperoxidase B in complex with p-cymene | 分子名称: | 1-methyl-4-(1-methylethyl)benzene, Dehaloperoxidase B, OXYGEN MOLECULE, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Malewschik, T, Yun, D. | 登録日 | 2021-10-17 | 公開日 | 2022-11-23 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.72 Å) | 主引用文献 | The Multifunctional Globin Dehaloperoxidase as a Biocatalyst in the Oxidation of Monoterpenes To Be Published
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7SJD
| Crystal structure of dehaloperoxidase B in complex with terpinolene | 分子名称: | 1-methyl-4-(propan-2-ylidene)cyclohex-1-ene, Dehaloperoxidase B, GLYCEROL, ... | 著者 | Ghiladi, R.A, de Serrano, V.S, Yun, D, Malewschik, T. | 登録日 | 2021-10-17 | 公開日 | 2022-11-23 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.703 Å) | 主引用文献 | The Multifunctional Globin Dehaloperoxidase as a Biocatalyst in the Oxidation of Monoterpenes To Be Published
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6BBS
| Joint X-ray/neutron structure of human carbonic anhydrase II in complex with brinzolamide | 分子名称: | (+)-4-ETHYLAMINO-3,4-DIHYDRO-2-(METHOXY)PROPYL-2H-THIENO[3,2-E]-1,2-THIAZINE-6-SULFONAMIDE-1,1-DIOXIDE, Carbonic anhydrase 2, ZINC ION | 著者 | Kovalevsky, A, Aggarwal, M, McKenna, R. | 登録日 | 2017-10-19 | 公開日 | 2018-02-28 | 最終更新日 | 2024-03-13 | 実験手法 | NEUTRON DIFFRACTION (2 Å), X-RAY DIFFRACTION | 主引用文献 | "To Be or Not to Be" Protonated: Atomic Details of Human Carbonic Anhydrase-Clinical Drug Complexes by Neutron Crystallography and Simulation. Structure, 26, 2018
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5V4E
| Engineered human IgG Fc domain glyco801 (Fc801) | 分子名称: | 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-2)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-[alpha-L-fucopyranose-(1-6)]2-acetamido-2-deoxy-beta-D-glucopyranose, ... | 著者 | Yan, W, Marshall, N, Zhang, Y.J. | 登録日 | 2017-03-09 | 公開日 | 2017-06-21 | 最終更新日 | 2020-07-29 | 実験手法 | X-RAY DIFFRACTION (3.216 Å) | 主引用文献 | IgG Fc domains that bind C1q but not effector Fc gamma receptors delineate the importance of complement-mediated effector functions. Nat. Immunol., 18, 2017
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6C92
| The structure of MppP soaked with the product 2-ketoarginine | 分子名称: | (4S)-5-carbamimidamido-4-hydroxy-2-oxopentanoic acid, (E)-N~2~-({3-hydroxy-2-methyl-5-[(phosphonooxy)methyl]pyridin-4-yl}methylidene)-L-arginine, PLP-Dependent L-Arginine Hydroxylase MppP | 著者 | Han, L, Silvaggi, N.R. | 登録日 | 2018-01-25 | 公開日 | 2018-09-05 | 最終更新日 | 2023-11-15 | 実験手法 | X-RAY DIFFRACTION (1.834 Å) | 主引用文献 | Streptomyces wadayamensis MppP is a PLP-Dependent Oxidase, Not an Oxygenase. Biochemistry, 57, 2018
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6C9B
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5WA2
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6CQK
| Crystal Structure of mitochondrial single-stranded DNA binding proteins from S. cerevisiae, Rim1 (Form1) | 分子名称: | SsDNA-binding protein essential for mitochondrial genome maintenance | 著者 | Singh, S.P, Kukshal, V, Bona, P.D, Lytle, A.K, Edwin, A, Galletto, R. | 登録日 | 2018-03-15 | 公開日 | 2018-05-30 | 最終更新日 | 2023-10-04 | 実験手法 | X-RAY DIFFRACTION (2.8 Å) | 主引用文献 | The mitochondrial single-stranded DNA binding protein from S. cerevisiae, Rim1, does not form stable homo-tetramers and binds DNA as a dimer of dimers. Nucleic Acids Res., 46, 2018
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7T9C
| Crystal structure of dehaloperoxidase B in complex with thymol | 分子名称: | 5-METHYL-2-(1-METHYLETHYL)PHENOL, Dehaloperoxidase B, GLYCEROL, ... | 著者 | de Serrano, V.S, Ghiladi, R.A, Malewschik, T, Yun, D. | 登録日 | 2021-12-18 | 公開日 | 2023-01-25 | 最終更新日 | 2023-10-25 | 実験手法 | X-RAY DIFFRACTION (1.73 Å) | 主引用文献 | The Multifunctional Globin Dehaloperoxidase as a Biocatalyst in the Oxidation of Monoterpenes To Be Published
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7UJD
| PSMD2 Structure bound to MC1 and Fab8/14 | 分子名称: | 26S proteasome non-ATPase regulatory subunit 2, ACY-PHE-PRO-ASP-VAL-SAR-LEU-HIS-ARG-TYR-TRP-GLY-TRP-ASP-CYS-GLY-NH2, Fab 14 HC CDRs, ... | 著者 | Johnson, M.C, Bashore, C, Ciferri, C, Dueber, E.C. | 登録日 | 2022-03-30 | 公開日 | 2023-01-11 | 実験手法 | ELECTRON MICROSCOPY (2.5 Å) | 主引用文献 | Targeted degradation via direct 26S proteasome recruitment. Nat.Chem.Biol., 19, 2023
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7UIH
| PSMD2 Structure | 分子名称: | 26S proteasome non-ATPase regulatory subunit 2, Fab 14 HC CDRs, Fab 14 LC CDRs, ... | 著者 | Johnson, M.C, Bashore, C, Ciferri, C, Dueber, E.C. | 登録日 | 2022-03-29 | 公開日 | 2023-01-11 | 最終更新日 | 2024-06-12 | 実験手法 | ELECTRON MICROSCOPY (3.1 Å) | 主引用文献 | Targeted degradation via direct 26S proteasome recruitment. Nat.Chem.Biol., 19, 2023
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8RDX
| PGGtase I in complex with probe BAY-6092 | 分子名称: | (5~{R})-5-(2-methoxyphenyl)-9-[(2~{R})-3,3,3-tris(fluoranyl)-2-methoxy-2-phenyl-propanoyl]-3,9-diazaspiro[5.5]undecan-2-one, CHLORIDE ION, DIPHOSPHATE, ... | 著者 | Steuber, H. | 登録日 | 2023-12-08 | 公開日 | 2024-02-14 | 最終更新日 | 2024-07-31 | 実験手法 | X-RAY DIFFRACTION (3.67 Å) | 主引用文献 | Discovery of YAP1/TAZ pathway inhibitors through phenotypic screening with potent anti-tumor activity via blockade of Rho-GTPase signaling. Cell Chem Biol, 31, 2024
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7LVT
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7NCJ
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7NCG
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7NCI
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7NCH
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7NCK
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7NCA
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8ORV
| Crystal structure of monkeypox virus poxin in complex with the STING agonist MD1203 | 分子名称: | 9-[(1~{S},6~{R},8~{R},9~{R},10~{R},15~{R},17~{R},18~{R})-8-(6-aminopurin-9-yl)-9,18-bis(fluoranyl)-3,12-bis(oxidanyl)-3,12-bis(oxidanylidene)-2,4,7,11,13-pentaoxa-3$l^{5},12$l^{5}-diphosphatricyclo[13.2.1.0^{6,10}]octadecan-17-yl]-1~{H}-purin-6-one, MPXVgp165 | 著者 | Duchoslav, V, Klima, M, Boura, E. | 登録日 | 2023-04-17 | 公開日 | 2023-12-20 | 最終更新日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (1.65 Å) | 主引用文献 | Fluorinated cGAMP analogs, which act as STING agonists and are not cleavable by poxins: Structural basis of their function. Structure, 32, 2024
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8P44
| Crystal structure of monkeypox virus poxin in complex with the STING agonist MD1202D | 分子名称: | 9-[(1~{S},3~{R},6~{R},8~{R},9~{R},10~{R},12~{R},15~{R},17~{R},18~{R})-8-(6-aminopurin-9-yl)-9,18-bis(fluoranyl)-3,12-bis(oxidanylidene)-3,12-bis(sulfanyl)-2,4,7,11,13-pentaoxa-3$l^{5},12$l^{5}-diphosphatricyclo[13.2.1.0^{6,10}]octadecan-17-yl]-1~{H}-purin-6-one, MPXVgp165 | 著者 | Duchoslav, V, Klima, M, Boura, E. | 登録日 | 2023-05-19 | 公開日 | 2023-12-20 | 最終更新日 | 2024-04-17 | 実験手法 | X-RAY DIFFRACTION (1.93 Å) | 主引用文献 | Fluorinated cGAMP analogs, which act as STING agonists and are not cleavable by poxins: Structural basis of their function. Structure, 32, 2024
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