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PDB: 1 件

5I5Z
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CDK8-CYCC IN COMPLEX WITH 8-(1-Methyl-2,2-dioxo-2,3-dihydro-1H-2l6-benzo[c]isothiazol-5-yl)-[1,6]naphthyridine-2-carboxylic acid methylamide
分子名称: Cyclin-C, Cyclin-dependent kinase 8, FORMIC ACID, ...
著者Musil, D, Blagg, J, Mallinger, A.
登録日2016-02-15
公開日2016-04-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献2,8-Disubstituted-1,6-Naphthyridines and 4,6-Disubstituted-Isoquinolines with Potent, Selective Affinity for CDK8/19.
Acs Med.Chem.Lett., 7, 2016

224201

件を2024-08-28に公開中

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