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PDB: 5628 件

4NQ4
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Bacillus cereus Zn-dependent metallo-beta-lactamase at pH 7
分子名称: Beta-lactamase 2, POTASSIUM ION, ZINC ION
著者Gonzalez, J.M, Gonzalez, M.M, Vila, A.J.
登録日2013-11-23
公開日2014-11-26
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.67 Å)
主引用文献Inhibition of metallo-lactamases with bicyclic compounds
TO BE PUBLISHED
4NFP
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Crystal Structure Analysis of the 16mer GCAGNCUUAAGUCUGC containing 8-aza-7-deaza-7-ethynyl Adenosine
分子名称: FORMAMIDE, GCAG(A7E)CUUAAGUCUGC
著者Beal, P.A, Fisher, A.J, Phelps, K.J, Ibarra-Soza, J.M, Zheng, Y.
登録日2013-10-31
公開日2014-07-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Click Modification of RNA at Adenosine: Structure and Reactivity of 7-Ethynyl- and 7-Triazolyl-8-aza-7-deazaadenosine in RNA.
Acs Chem.Biol., 9, 2014
4NFQ
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Crystal Structure Analysis of the 16mer GCAGNCUUAAGUCUGC containing 7-triazolyl-8-aza-7-deazaadenosine
分子名称: GCAG(7AT)CUUAAGUCUGC
著者Beal, P.A, Fisher, A.J, Phelps, K.J, Ibarra-Soza, J.M, Zheng, Y.
登録日2013-10-31
公開日2014-07-02
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Click Modification of RNA at Adenosine: Structure and Reactivity of 7-Ethynyl- and 7-Triazolyl-8-aza-7-deazaadenosine in RNA.
Acs Chem.Biol., 9, 2014
1P6A
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STRUCTURAL BASIS FOR VARIATION IN ADENOVIRUS AFFINITY FOR THE CELLULAR RECEPTOR CAR (S489Y MUTANT)
分子名称: Coxsackievirus and adenovirus receptor, Fiber protein
著者Howitt, J, Bewley, M.C, Graziano, V, Flanagan, J.M, Freimuth, P.
登録日2003-04-29
公開日2004-05-11
最終更新日2018-08-22
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural basis for variation in adenovirus affinity for the cellular coxsackievirus and adenovirus receptor.
J.Biol.Chem., 278, 2003
4QNH
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Calcium-calmodulin (T79D) complexed with the calmodulin binding domain from a small conductance potassium channel SK2-a
分子名称: CALCIUM ION, Calmodulin, SULFATE ION, ...
著者Zhang, M, Pascal, J.M, Logothetis, D.E, Zhang, J.F.
登録日2014-06-17
公開日2014-08-06
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.02 Å)
主引用文献Selective phosphorylation modulates the PIP2 sensitivity of the CaM-SK channel complex.
Nat.Chem.Biol., 10, 2014
1G10
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TOLUENE-4-MONOOXYGENASE CATALYTIC EFFECTOR PROTEIN NMR STRUCTURE
分子名称: TOLUENE-4-MONOOXYGENASE CATALYTIC EFFECTOR
著者Hemmi, H, Studts, J.M, Chae, Y.K, Song, J, Markley, J.L, Fox, B.G.
登録日2000-10-10
公開日2001-05-09
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献Solution structure of the toluene 4-monooxygenase effector protein (T4moD).
Biochemistry, 40, 2001
4MX1
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Structure of ricin A chain bound with 2-amino-4-oxo-N-(2-(3-phenylureido)ethyl)-3,4-dihydropteridine-7-carboxamide
分子名称: 2-amino-4-oxo-N-{2-[(phenylcarbamoyl)amino]ethyl}-3,4-dihydropteridine-7-carboxamide, MALONIC ACID, Ricin A chain, ...
著者Robertus, J.D, Wiget, P.A, Manzano, L.A, Pruet, J.M, Gao, G, Saito, R, Jasheway, K.R, Monzingo, A.F, Anslyn, E.V.
登録日2013-09-25
公開日2014-01-15
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.59 Å)
主引用文献Sulfur incorporation generally improves Ricin inhibition in pterin-appended glycine-phenylalanine dipeptide mimics.
Bioorg.Med.Chem.Lett., 23, 2013
4N4A
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Cystal structure of Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1
分子名称: Cap-specific mRNA (nucleoside-2'-O-)-methyltransferase 1
著者Smietanski, M, Werener, M, Purta, E, Kaminska, K.H, Stepinski, J, Darzynkiewicz, E, Nowotny, M, Bujnicki, J.M.
登録日2013-10-08
公開日2014-01-22
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (2.35 Å)
主引用文献Structural analysis of human 2'-O-ribose methyltransferases involved in mRNA cap structure formation.
Nat Commun, 5, 2014
4QQV
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Extracellular domains of mouse IL-3 beta receptor
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Interleukin-3 receptor class 2 subunit beta
著者Jackson, C.J, Young, I.G, Murphy, J.M, Carr, P.D, Ewens, C.L, Dai, J, Ollis, D.L.
登録日2014-06-30
公開日2014-09-03
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.45 Å)
主引用文献Crystal structure of the mouse interleukin-3 beta-receptor: insights into interleukin-3 binding and receptor activation.
Biochem.J., 463, 2014
4QYY
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Discovery of Novel, Dual Mechanism ERK Inhibitors by Affinity Selection Screening of an Inactive Kinase State
分子名称: (3R)-1-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-N-(3-chloro-4-hydroxyphenyl)pyrrolidine-3-carboxamide, Mitogen-activated protein kinase 1, SULFATE ION
著者Deng, Y, Shipps, G.W, Cooper, A, English, J.M, Annis, D.A, Carr, D, Nan, Y, Wang, T, Zhu, Y.H, Chuang, C, Dayananth, P, Hruza, A.W, Xiao, L, Jin, W, Kirschmeier, P, Windsor, W.T, Samatar, A.A.
登録日2014-07-26
公開日2014-11-12
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.65 Å)
主引用文献Discovery of Novel, Dual Mechanism ERK Inhibitors by Affinity Selection Screening of an Inactive Kinase.
J.Med.Chem., 57, 2014
4R6W
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Plasmodium falciparum phosphoethanolamine methyltransferase D128A mutant in complex with S-adenosylhomocysteine and phosphocholine
分子名称: PHOSPHOCHOLINE, Phosphoethanolamine N-methyltransferase, S-ADENOSYL-L-HOMOCYSTEINE
著者Lee, S.G, Jez, J.M.
登録日2014-08-26
公開日2014-10-08
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (1.5894 Å)
主引用文献An Alternative Mechanism for the Methylation of Phosphoethanolamine Catalyzed by Plasmodium falciparum Phosphoethanolamine Methyltransferase.
J.Biol.Chem., 289, 2014
3IWZ
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The c-di-GMP Responsive Global Regulator CLP Links Cell-Cell Signaling to Virulence Gene Expression in Xanthomonas campestris
分子名称: Catabolite activation-like protein
著者Chin, K.H, Tu, Z.L, Tseng, Y.H, Dow, J.M, Wang, A.H.J, Chou, S.H.
登録日2009-09-03
公開日2009-12-15
最終更新日2024-03-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献The cAMP receptor-like protein CLP is a novel c-di-GMP receptor linking cell-cell signaling to virulence gene expression in Xanthomonas campestris.
J.Mol.Biol., 396, 2010
4R1Q
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Crystal Structure of Thermophilic Geobacillus kaustophilus L-Arabinose isomerase in complex with L-arabitol
分子名称: L-arabinitol, L-arabinose isomerase, MANGANESE (II) ION
著者Choi, J.M, Lee, Y.J, Lee, D.W, Lee, S.H.
登録日2014-08-07
公開日2015-08-12
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.248 Å)
主引用文献Crystal Structure of Thermophilic L-Arabinose Isomerase with L-Arabitol from Geobacillus kaustophilus
to be published
4R2Y
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Crystal structure of APC11 RING domain
分子名称: Anaphase-promoting complex subunit 11, ZINC ION
著者Brown, N.G, Watson, E.R, Weissmann, F, Jarvis, M.A, Vanderlinden, R, Grace, C.R.R, Frye, J.J, Dube, P, Qiao, R, Petzold, G, Cho, S.E, Alsharif, O, Bao, J, Zheng, J, Nourse, A, Kurinov, I, Peters, J.M, Stark, H, Schulman, B.A.
登録日2014-08-13
公開日2014-10-29
最終更新日2024-02-28
実験手法X-RAY DIFFRACTION (1.755 Å)
主引用文献Mechanism of Polyubiquitination by Human Anaphase-Promoting Complex: RING Repurposing for Ubiquitin Chain Assembly.
Mol.Cell, 56, 2014
4R79
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Mos1 transposase paired-end complex with left transposon end
分子名称: MANGANESE (II) ION, Mariner Mos1 transposase, SULFATE ION, ...
著者Richardson, J.M.
登録日2014-08-27
公開日2015-04-22
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3.1 Å)
主引用文献Structural Basis for the Inverted Repeat Preferences of mariner Transposases.
J.Biol.Chem., 290, 2015
4R0E
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Crystal Structure of the Poliovirus RNA-Dependent RNA Polymerase Low-Fidelity Mutant 3Dpol H273R
分子名称: RNA-directed RNA polymerase
著者Marcotte, L.L, Gohara, D.W, Filman, D.J, Hogle, J.M.
登録日2014-07-30
公開日2014-11-12
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (3 Å)
主引用文献Structural Dynamics as a Contributor to Error-prone Replication by an RNA-dependent RNA Polymerase.
J.Biol.Chem., 289, 2014
4R0R
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Ebolavirus GP Prehairpin Intermediate Mimic
分子名称: eboIZN21
著者Clinton, T.R, Weinstock, M.T, Jacobsen, M.T, Szabo-Fresnais, N, Pandya, M.J, Whitby, F.G, Herbert, A.S, Prugar, L.I, McKinnon, R, Hill, C.P, Welch, B.D, Dye, J.M, Eckert, D.M, Kay, M.S.
登録日2014-08-01
公開日2014-10-22
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Design and characterization of ebolavirus GP prehairpin intermediate mimics as drug targets.
Protein Sci., 24, 2015
4R1O
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Crystal Structure of Thermophilic Geobacillus kaustophilus L-Arabinose isomerase
分子名称: L-arabinose isomerase
著者Choi, J.M, Lee, Y.J, Lee, D.W, Lee, S.H.
登録日2014-08-07
公開日2015-08-12
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.401 Å)
主引用文献Crystal Structure of Thermophilic apo L-Arabinose Isomerase from Geobacillus kaustophilus
to be published
4R27
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Crystal structure of beta-glycosidase BGL167
分子名称: Glycoside hydrolase
著者Park, S.J, Choi, J.M, Kyeong, H.H, Kim, S.G, Kim, H.S.
登録日2014-08-09
公開日2015-05-27
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.03 Å)
主引用文献Rational design of a beta-glycosidase with high regiospecificity for triterpenoid tailoring
Chembiochem, 16, 2015
1K38
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CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-2
分子名称: Beta-lactamase OXA-2, FORMIC ACID
著者Kerff, F, Fonze, E, Bouillenne, F, Frere, J.M, Charlier, P.
登録日2001-10-02
公開日2003-06-24
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (1.5 Å)
主引用文献CRYSTAL STRUCTURE OF THE CLASS D BETA-LACTAMASE OXA-2
To be Published
4E2K
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The structure of the S. aureus DnaG RNA Polymerase Domain
分子名称: BENZAMIDINE, DNA primase
著者Rymer, R.U, Solorio, F.A, Clement, C, Corn, J.E, Wang, J.D, Berger, J.M.
登録日2012-03-08
公開日2012-08-01
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (2.15 Å)
主引用文献Binding Mechanism of Metal-NTP Substrates and Stringent-Response Alarmones to Bacterial DnaG-Type Primases.
Structure, 20, 2012
8PUJ
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The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: COB(II)INAMIDE, HYDROXIDE ION, SODIUM ION, ...
著者Whittaker, J, Martinez-Felices, J.M, Guskov, A, Slotboom, D.J.
登録日2023-07-17
公開日2024-07-24
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献The surface-exposed lipo-protein of BtuG3 in complex with cyanocobinamide.
To Be Published
8PTF
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The surface-exposed lipo-protein of BtuG2 in complex with cyanocobalamin.
分子名称: COB(II)INAMIDE, SODIUM ION, YncE family protein, ...
著者Whittaker, J, Felices Martinez, J.M, Guskov, A, Slotboom, D.J.
登録日2023-07-14
公開日2024-07-24
実験手法X-RAY DIFFRACTION (1.95 Å)
主引用文献The surface-exposed lipo-protein of BtuG1 in complex with cyanocobinamide.
To Be Published
1AR6
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P1/MAHONEY POLIOVIRUS, DOUBLE MUTANT V1160I +P1095S
分子名称: MYRISTIC ACID, P1/MAHONEY POLIOVIRUS, SPHINGOSINE
著者Wien, M.W, Curry, S, Filman, D.J, Hogle, J.M.
登録日1997-08-11
公開日1997-12-03
最終更新日2023-08-09
実験手法X-RAY DIFFRACTION (2.9 Å)
主引用文献Structural studies of poliovirus mutants that overcome receptor defects.
Nat.Struct.Biol., 4, 1997
4EEU
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Crystal structure of phiLOV2.1
分子名称: FLAVIN MONONUCLEOTIDE, Phototropin-2
著者Hitomi, K, Christie, J.M, Arvai, A.S, Hartfield, K.A, Pratt, A.J, Tainer, J.A, Getzoff, E.D.
登録日2012-03-28
公開日2012-05-16
最終更新日2023-09-13
実験手法X-RAY DIFFRACTION (1.4068 Å)
主引用文献Structural Tuning of the Fluorescent Protein iLOV for Improved Photostability.
J.Biol.Chem., 287, 2012

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件を2024-08-28に公開中

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