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PDB: 6 件

5HF3
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BU of 5hf3 by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 201D with 14-3-3sigma
分子名称: 14-3-3 protein sigma, modified Tau peptide
著者Bartel, M, Milroy, L.G, Brunsveld, L, Ottmann, C.
登録日2016-01-06
公開日2016-01-27
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Stabilizer-Guided Inhibition of Protein-Protein Interactions.
Angew.Chem.Int.Ed.Engl., 54, 2015
4Y3B
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BU of 4y3b by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 201D with 14-3-3sigma
分子名称: (2S)-2-(2-methoxyethyl)pyrrolidine, 14-3-3 protein sigma, ARG-THR-PRO-SEP-LEU-PRO-THR-[H][C@@]1(C(C2=CC=CC=C2)C3=CC=CC=C3)CCCN1C
著者Bartel, M, Milroy, L.G, Brunsveld, L, Ottmann, C.
登録日2015-02-10
公開日2015-12-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.8 Å)
主引用文献Stabilizer-Guided Inhibition of Protein-Protein Interactions.
Angew.Chem.Int.Ed.Engl., 54, 2015
4Y32
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BU of 4y32 by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 109B with 14-3-3sigma
分子名称: (2S)-2-(2-methoxyethyl)pyrrolidine, 14-3-3 protein sigma, ARG-THR-PRO-SEP-LEU-PRO-CNC(C(C)O)C(=O)N1CCCC1CCOC
著者Bartel, M, Milroy, L, Bier, D, Brunsveld, L, Ottmann, C.
登録日2015-02-10
公開日2015-12-23
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Stabilizer-Guided Inhibition of Protein-Protein Interactions.
Angew.Chem.Int.Ed.Engl., 54, 2015
4Y5I
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BU of 4y5i by Molmil
Crystal structure of C-terminal modified Tau peptide-hybrid 126B with 14-3-3sigma
分子名称: 14-3-3 protein sigma, CHLORIDE ION, Microtubule-associated protein tau
著者Leysen, S, Bartel, M, Milroy, L, Brunsveld, L, Ottmann, C.
登録日2015-02-11
公開日2016-01-13
最終更新日2024-01-10
実験手法X-RAY DIFFRACTION (1.4 Å)
主引用文献Stabilizer-Guided Inhibition of Protein-Protein Interactions.
Angew.Chem.Int.Ed.Engl., 54, 2015
5BTV
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BU of 5btv by Molmil
Crystal structure of human 14-3-3 sigma in complex with a Tau-protein peptide surrounding pS324
分子名称: 14-3-3 protein sigma, CALCIUM ION, CHLORIDE ION, ...
著者Ottmann, C, Schumacher, B, Bartel, M.
登録日2015-06-03
公開日2016-07-20
最終更新日2019-03-13
実験手法X-RAY DIFFRACTION (1.7 Å)
主引用文献Involvement of 14-3-3 in tubulin instability and impaired axon development is mediated by Tau.
Faseb J., 29, 2015
3UX0
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BU of 3ux0 by Molmil
Crystal structure of human 14-3-3 sigma in complex with TASK-3 peptide and stabilizer Fusicoccin H
分子名称: (4R,5R,6R,6aS,9S,9aE,10aR)-5-hydroxy-9-(hydroxymethyl)-6,10a-dimethyl-3-(propan-2-yl)-1,2,4,5,6,6a,7,8,9,10a-decahydrodicyclopenta[a,d][8]annulen-4-yl alpha-D-gulopyranoside, 14-3-3 protein sigma, CHLORIDE ION, ...
著者Thiel, P, Bartel, M, Anders, C, Higuchi, Y, Schumacher, B, Kato, N, Ottmann, C.
登録日2011-12-03
公開日2013-01-02
最終更新日2013-05-01
実験手法X-RAY DIFFRACTION (1.75 Å)
主引用文献A semisynthetic fusicoccane stabilizes a protein-protein interaction and enhances the expression of k(+) channels at the cell surface.
Chem.Biol., 20, 2013

224201

件を2024-08-28に公開中

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