Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help
Search by PDB author
1A5Y
DownloadVisualize
BU of 1a5y by Molmil
PROTEIN TYROSINE PHOSPHATASE 1B CYSTEINYL-PHOSPHATE INTERMEDIATE
Descriptor: PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Pannifer, A.D.P, Flint, A.J, Tonks, N.K, Barford, D.
Deposit date:1998-02-19
Release date:1998-06-17
Last modified:2023-08-02
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Visualization of the cysteinyl-phosphate intermediate of a protein-tyrosine phosphatase by x-ray crystallography.
J.Biol.Chem., 273, 1998
3ZV2
DownloadVisualize
BU of 3zv2 by Molmil
Human protein-tyrosine phosphatase 1b C215A, S216A mutant
Descriptor: Tyrosine-protein phosphatase non-receptor type 1
Authors:Barford, D, Salmeen, A, Tonks, N.K.
Deposit date:2011-07-22
Release date:2011-08-31
Last modified:2023-12-20
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:Conformation-sensing antibodies stabilize the oxidized form of PTP1B and inhibit its phosphatase activity.
Cell, 147, 2011
5VF6
DownloadVisualize
BU of 5vf6 by Molmil
Crystal structure of single chain variable fragment (scFv45).
Descriptor: single chain variable fragment
Authors:Shrestha, O.K, Tocilj, A, Joshua-Tor, L, Tonks, N.K.
Deposit date:2017-04-06
Release date:2018-01-31
Last modified:2023-10-04
Method:X-RAY DIFFRACTION (1.635 Å)
Cite:Harnessing insulin- and leptin-induced oxidation of PTP1B for therapeutic development.
Nat Commun, 9, 2018
1H6G
DownloadVisualize
BU of 1h6g by Molmil
alpha-catenin M-domain
Descriptor: (4S)-2-METHYL-2,4-PENTANEDIOL, ALPHA-1 CATENIN, CALCIUM ION, ...
Authors:Yang, J, Dokurno, P, Tonks, N.K, Barford, D.
Deposit date:2001-06-14
Release date:2001-08-07
Last modified:2016-02-10
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Crystal Structure of the M-Fragment of Alpha-Catenin: Implications for Modulation of Cell Adhesion.
Embo J., 20, 2001
2HNQ
DownloadVisualize
BU of 2hnq by Molmil
CRYSTAL STRUCTURE OF HUMAN PROTEIN TYROSINE PHOSPHATASE 1B
Descriptor: PROTEIN-TYROSINE PHOSPHATASE-1B, TUNGSTATE(VI)ION
Authors:Barford, D, Flint, A.J, Tonks, N.K.
Deposit date:1994-09-28
Release date:1994-12-20
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.85 Å)
Cite:Crystal structure of human protein tyrosine phosphatase 1B.
Science, 263, 1994
2HNP
DownloadVisualize
BU of 2hnp by Molmil
CRYSTAL STRUCTURE OF HUMAN PROTEIN TYROSINE PHOSPHATASE 1B
Descriptor: PROTEIN-TYROSINE PHOSPHATASE-1B
Authors:Barford, D, Flint, A.J, Tonks, N.K.
Deposit date:1994-09-19
Release date:1994-12-20
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.85 Å)
Cite:Crystal structure of human protein tyrosine phosphatase 1B.
Science, 263, 1994
1G1H
DownloadVisualize
BU of 1g1h by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH A BIS-PHOSPHORYLATED PEPTIDE (ETD(PTR)(PTR)RKGGKGLL) FROM THE INSULIN RECEPTOR KINASE
Descriptor: BI-PHOSPHORYLATED PEPTIDE FROM THE INSULIN RECEPTOR KINASE, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Salmeen, A, Andersen, J.N, Myers, M.P, Tonks, N.K, Barford, D.
Deposit date:2000-10-11
Release date:2001-01-17
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.4 Å)
Cite:Molecular basis for the dephosphorylation of the activation segment of the insulin receptor by protein tyrosine phosphatase 1B.
Mol.Cell, 6, 2000
1G1G
DownloadVisualize
BU of 1g1g by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH A MONO-PHOSPHORYLATED PEPTIDE (ETDY(PTR)RKGGKGLL) FROM THE INSULIN RECEPTOR KINASE
Descriptor: MONO-PHOSPHORYLATED PEPTIDE FROM THE INSULIN RECEPTOR KINASE, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Salmeen, A, Andersen, J.N, Myers, M.P, Tonks, N.K, Barford, D.
Deposit date:2000-10-11
Release date:2001-01-17
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:Molecular basis for the dephosphorylation of the activation segment of the insulin receptor by protein tyrosine phosphatase 1B.
Mol.Cell, 6, 2000
1G1F
DownloadVisualize
BU of 1g1f by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH A TRI-PHOSPHORYLATED PEPTIDE (RDI(PTR)ETD(PTR)(PTR)RK) FROM THE INSULIN RECEPTOR KINASE
Descriptor: PROTEIN TYROSINE PHOSPHATASE 1B, TRI-PHOSPHORYLATED PEPTIDE FROM THE INSULIN RECEPTOR KINASE
Authors:Salmeen, A, Andersen, J.N, Myers, M.P, Tonks, N.K, Barford, D.
Deposit date:2000-10-11
Release date:2001-01-17
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2 Å)
Cite:Molecular basis for the dephosphorylation of the activation segment of the insulin receptor by protein tyrosine phosphatase 1B.
Mol.Cell, 6, 2000
1RPM
DownloadVisualize
BU of 1rpm by Molmil
HUMAN RECEPTOR PROTEIN TYROSINE PHOSPHATASE MU, DOMAIN 1
Descriptor: RECEPTOR PROTEIN TYROSINE PHOSPHATASE MU
Authors:Hoffmann, K.M.V, Tonks, N.K, Barford, D.
Deposit date:1997-09-11
Release date:1998-04-01
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:The crystal structure of domain 1 of receptor protein-tyrosine phosphatase mu.
J.Biol.Chem., 272, 1997
1OEM
DownloadVisualize
BU of 1oem by Molmil
PTP1B with the catalytic cysteine oxidized to a sulfenyl-amide bond
Descriptor: PROTEIN-TYROSINE PHOSPHATASE, NON-RECEPTOR TYPE 1
Authors:Salmeen, A, Andersen, J.N, Myers, M.P, Meng, T.C, Hinks, J.A, Tonks, N.K, Barford, D.
Deposit date:2003-03-28
Release date:2003-06-12
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (1.8 Å)
Cite:Redox Regulation of Protein Tyrosine Phosphatase Involves a Sulfenyl-Amide Intermediate
Nature, 423, 2003
1OEO
DownloadVisualize
BU of 1oeo by Molmil
PTP1B with the catalytic cysteine oxidized to sulfonic acid
Descriptor: PROTEIN-TYROSINE PHOSPHATASE, NON-RECEPTOR TYPE 1
Authors:Salmeen, A, Andersen, J.N, Myers, M.P, Meng, T.C, Hinks, J.A, Tonks, N.K, Barford, D.
Deposit date:2003-03-28
Release date:2003-06-12
Last modified:2023-12-13
Method:X-RAY DIFFRACTION (2.15 Å)
Cite:Redox Regulation of Protein Tyrosine Phosphatase Involves a Sulfenyl-Amide Intermediate
Nature, 423, 2003
1OHE
DownloadVisualize
BU of 1ohe by Molmil
Structure of cdc14b phosphatase with a peptide ligand
Descriptor: CDC14B2 PHOSPHATASE, PEPTIDE LIGAND
Authors:Gray, C.H, Good, V.M, Tonks, N.K, Barford, D.
Deposit date:2003-05-24
Release date:2003-07-24
Last modified:2019-05-08
Method:X-RAY DIFFRACTION (2.2 Å)
Cite:The Structure of the Cell Cycle Protein Cdc14 Reveals a Proline-Directed Protein Phosphatase
Embo J., 22, 2003
1OHD
DownloadVisualize
BU of 1ohd by Molmil
structure of cdc14 in complex with tungstate
Descriptor: CDC14B2 PHOSPHATASE, TUNGSTATE(VI)ION
Authors:Gray, C.H, Good, V.M, Tonks, N.K, Barford, D.
Deposit date:2003-05-24
Release date:2003-07-24
Last modified:2019-05-08
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:The Structure of the Cell Cycle Protein Cdc14 Reveals a Proline-Directed Protein Phosphatase
Embo J., 22, 2003
1OHC
DownloadVisualize
BU of 1ohc by Molmil
Structure of the proline directed phosphatase cdc14
Descriptor: CDC14B2 PHOSPHATASE
Authors:Gray, C.H, Good, V.M, Tonks, N.K, Barford, D.
Deposit date:2003-05-24
Release date:2003-07-24
Last modified:2019-05-08
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The Structure of the Cell Cycle Protein Cdc14 Reveals a Proline-Directed Protein Phosphatase
Embo J., 22, 2003
1AAX
DownloadVisualize
BU of 1aax by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH TWO BIS(PARA-PHOSPHOPHENYL)METHANE (BPPM) MOLECULES
Descriptor: 4-PHOSPHONOOXY-PHENYL-METHYL-[4-PHOSPHONOOXY]BENZEN, MAGNESIUM ION, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Puius, Y.A, Zhao, Y, Sullivan, M, Lawrence, D, Almo, S.C, Zhang, Z.-Y.
Deposit date:1997-01-16
Release date:1998-03-04
Last modified:2023-08-02
Method:X-RAY DIFFRACTION (1.9 Å)
Cite:Identification of a second aryl phosphate-binding site in protein-tyrosine phosphatase 1B: a paradigm for inhibitor design.
Proc.Natl.Acad.Sci.USA, 94, 1997
3HB0
DownloadVisualize
BU of 3hb0 by Molmil
Structure of edeya2 complexed with bef3
Descriptor: BERYLLIUM TRIFLUORIDE ION, Eyes absent homolog 2 (Drosophila), MAGNESIUM ION
Authors:Jung, S.K, Jeong, D.G, Ryu, S.E, Kim, S.J.
Deposit date:2009-05-03
Release date:2009-12-01
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:Crystal structure of ED-Eya2: insight into dual roles as a protein tyrosine phosphatase and a transcription factor
Faseb J., 24, 2010
3HB1
DownloadVisualize
BU of 3hb1 by Molmil
Crystal structure of ed-eya2 complexed with Alf3
Descriptor: ALUMINUM FLUORIDE, Eyes absent homolog 2 (Drosophila), MAGNESIUM ION
Authors:Jung, S.K, Jeong, D.G, Ryu, S.E, Kim, S.J.
Deposit date:2009-05-03
Release date:2009-12-01
Last modified:2023-11-01
Method:X-RAY DIFFRACTION (2.51 Å)
Cite:Crystal structure of ED-Eya2: insight into dual roles as a protein tyrosine phosphatase and a transcription factor
Faseb J., 24, 2010
4Y14
DownloadVisualize
BU of 4y14 by Molmil
Structure of protein tyrosine phosphatase 1B complexed with inhibitor (PTP1B:CPT157633)
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, 3-bromo-4-[difluoro(phosphono)methyl]-N-methyl-Nalpha-(methylsulfonyl)-L-phenylalaninamide, CHLORIDE ION, ...
Authors:Choy, M.S, Connors, C, Page, R, Peti, W.
Deposit date:2015-02-06
Release date:2015-08-05
Last modified:2023-09-27
Method:X-RAY DIFFRACTION (1.898 Å)
Cite:PTP1B inhibition suggests a therapeutic strategy for Rett syndrome.
J.Clin.Invest., 125, 2015
1BZH
DownloadVisualize
BU of 1bzh by Molmil
Cyclic peptide inhibitor of human PTP1B
Descriptor: PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE 1B INHIBITOR), PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE 1B)
Authors:Groves, M.R, Yao, Z.J, Burke Jr, T.R, Barford, D.
Deposit date:1998-10-28
Release date:1999-02-16
Last modified:2023-11-15
Method:X-RAY DIFFRACTION (2.1 Å)
Cite:Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics.
Biochemistry, 37, 1998
1BZC
DownloadVisualize
BU of 1bzc by Molmil
HUMAN PTP1B CATALYTIC DOMAIN COMPLEXED WITH TPI
Descriptor: 4-CARBAMOYL-4-{[6-(DIFLUORO-PHOSPHONO-METHYL)-NAPHTHALENE-2-CARBONYL]-AMINO}-BUTYRIC ACID, PROTEIN (PROTEIN-TYROSINE-PHOSPHATASE)
Authors:Groves, M.R, Yao, Z.J, Jr Burke, T.R, Barford, D.
Deposit date:1998-10-27
Release date:1999-02-16
Last modified:2023-08-09
Method:X-RAY DIFFRACTION (2.35 Å)
Cite:Structural basis for inhibition of the protein tyrosine phosphatase 1B by phosphotyrosine peptide mimetics.
Biochemistry, 37, 1998
1PTV
DownloadVisualize
BU of 1ptv by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH PHOSPHOTYROSINE
Descriptor: O-PHOSPHOTYROSINE, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Barford, D, Jia, Z.
Deposit date:1995-04-21
Release date:1996-08-01
Last modified:2024-02-14
Method:X-RAY DIFFRACTION (2.3 Å)
Cite:Structural basis for phosphotyrosine peptide recognition by protein tyrosine phosphatase 1B.
Science, 268, 1995
1PTT
DownloadVisualize
BU of 1ptt by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH PHOSPHOTYROSINE-CONTAINING TETRA-PEPTIDE (AC-DEPYL-NH2)
Descriptor: PHOSPHOTYROSINE-CONTAINING TETRA-PEPTIDE, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Barford, D, Jia, Z.
Deposit date:1995-04-21
Release date:1996-08-01
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Structural basis for phosphotyrosine peptide recognition by protein tyrosine phosphatase 1B.
Science, 268, 1995
1PTU
DownloadVisualize
BU of 1ptu by Molmil
CRYSTAL STRUCTURE OF PROTEIN TYROSINE PHOSPHATASE 1B COMPLEXED WITH PHOSPHOTYROSINE-CONTAINING HEXA-PEPTIDE (DADEPYL-NH2)
Descriptor: PHOSPHOTYROSINE-CONTAINING HEXA-PEPTIDE, PROTEIN TYROSINE PHOSPHATASE 1B
Authors:Barford, D, Jia, Z.
Deposit date:1995-04-21
Release date:1996-08-01
Last modified:2021-11-03
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Structural basis for phosphotyrosine peptide recognition by protein tyrosine phosphatase 1B.
Science, 268, 1995
1SUG
DownloadVisualize
BU of 1sug by Molmil
1.95 A structure of apo protein tyrosine phosphatase 1B
Descriptor: 2-AMINO-2-HYDROXYMETHYL-PROPANE-1,3-DIOL, GLYCEROL, Protein-tyrosine phosphatase, ...
Authors:Pedersen, A.K, Peters, G.H, Moller, K.B, Iversen, L.F, Kastrup, J.S.
Deposit date:2004-03-26
Release date:2004-09-07
Last modified:2023-08-23
Method:X-RAY DIFFRACTION (1.95 Å)
Cite:Water-molecule network and active-site flexibility of apo protein tyrosine phosphatase 1B.
Acta Crystallogr.,Sect.D, 60, 2004

 

12>

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon