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6WGN
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BU of 6wgn by Molmil
Crystal structure of K-Ras(G12D) GppNHp bound to cyclic peptide ligand KD2
Descriptor: Cyclic Peptide KD2, GTPase KRas, MAGNESIUM ION, ...
Authors:Zhang, Z, Gao, R, Hu, Q, Peacock, H, Peacock, D.M, Shokat, K.M, Suga, H.
Deposit date:2020-04-06
Release date:2020-10-14
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (1.601 Å)
Cite:GTP-State-Selective Cyclic Peptide Ligands of K-Ras(G12D) Block Its Interaction with Raf.
Acs Cent.Sci., 6, 2020
8TLR
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BU of 8tlr by Molmil
Crystal Structure of human HRAS G12C covalently bound to AMG 510
Descriptor: AMG 510 (bound form), GTPase HRas, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Morstein, J, Guiley, K.Z, Shokat, K.M.
Deposit date:2023-07-27
Release date:2024-07-31
Method:X-RAY DIFFRACTION (1.70003951 Å)
Cite:Targeting Ras-, Rho-, and Rab-Family GTPases via a Conserved Cryptic Pocket
To Be Published

224201

건을2024-08-28부터공개중

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