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2JDJ
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BU of 2jdj by Molmil
crystal structure of HapK from Hahella chejuensis
分子名称: GLYCEROL, ISOPROPYL ALCOHOL, REDY-LIKE PROTEIN, ...
著者Kang, B.S, Cho, H.J, Kim, K.J.
登録日2007-01-10
公開日2007-09-11
最終更新日2011-07-13
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural Insight of the Role of the Hahella Chejuensis Hapk Protein in Prodigiosin Biosynthesis.
Proteins, 70, 2008
7EHK
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BU of 7ehk by Molmil
Crystal structure of C107S mutant of FfIBP
分子名称: CHLORIDE ION, Ice-binding protein
著者Do, H, Lee, J.H.
登録日2021-03-29
公開日2022-03-02
最終更新日2023-11-29
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Importance of rigidity of ice-binding protein (FfIBP) for hyperthermal hysteresis activity and microbial survival.
Int.J.Biol.Macromol., 204, 2022
7KDT
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Human Tom70 in complex with SARS CoV2 Orf9b
分子名称: Mitochondrial import receptor subunit TOM70, ORF9b protein
著者QCRG Structural Biology Consortium
登録日2020-10-09
公開日2020-10-21
最終更新日2024-03-06
実験手法ELECTRON MICROSCOPY (3.05 Å)
主引用文献Comparative host-coronavirus protein interaction networks reveal pan-viral disease mechanisms.
Science, 370, 2020
8EL2
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BU of 8el2 by Molmil
SARS-CoV-2 RBD bound to neutralizing antibody Fab ICO-hu23
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, Fab ICO-hu23 Heavy Chain, Fab ICO-hu23 Light Chain, ...
著者Besaw, J.E, Kuo, A, Morizumi, T, Ernst, O.P.
登録日2022-09-22
公開日2023-07-19
最終更新日2023-10-25
実験手法X-RAY DIFFRACTION (2.89 Å)
主引用文献Broadly neutralizing humanized SARS-CoV-2 antibody binds to a conserved epitope on Spike and provides antiviral protection through inhalation-based delivery in non-human primates.
Plos Pathog., 19, 2023
4XB2
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BU of 4xb2 by Molmil
Hyperthermophilic archaeal homoserine dehydrogenase mutant in complex with NADPH
分子名称: 319aa long hypothetical homoserine dehydrogenase, L-HOMOSERINE, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Sakuraba, H, Inoue, S, Yoneda, K, Ohshima, T.
登録日2014-12-16
公開日2015-07-15
最終更新日2023-11-15
実験手法X-RAY DIFFRACTION (2.43 Å)
主引用文献Crystal Structures of a Hyperthermophilic Archaeal Homoserine Dehydrogenase Suggest a Novel Cofactor Binding Mode for Oxidoreductases.
Sci Rep, 5, 2015
4XB1
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BU of 4xb1 by Molmil
Hyperthermophilic archaeal homoserine dehydrogenase in complex with NADPH
分子名称: (4S)-2-METHYL-2,4-PENTANEDIOL, 319aa long hypothetical homoserine dehydrogenase, NADPH DIHYDRO-NICOTINAMIDE-ADENINE-DINUCLEOTIDE PHOSPHATE, ...
著者Sakuraba, H, Inoue, S, Yoneda, K, Ohshima, T.
登録日2014-12-16
公開日2015-07-15
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of a Hyperthermophilic Archaeal Homoserine Dehydrogenase Suggest a Novel Cofactor Binding Mode for Oxidoreductases.
Sci Rep, 5, 2015
4B18
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BU of 4b18 by Molmil
The crystal structure of human Importin alpha 5 with TERT NLS peptide
分子名称: IMPORTIN SUBUNIT ALPHA-1, TELOMERASE REVERSE TRANSCRIPTASE
著者Kim, K.L, Yoo, J.H, Cho, H.S.
登録日2012-07-08
公開日2013-09-04
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Akt-Mediated Phosphorylation Increases the Binding Affinity of Htert for Importin Alpha to Promote Nuclear Translocation.
J.Cell.Sci., 128, 2015
6NE5
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BU of 6ne5 by Molmil
Discovery of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors that Demonstrate in vivo Activity in Mouse Xenograft Models of Human Cancer
分子名称: 3-[(4R)-7-chloro-10-[3-(4-chloro-3,5-dimethylphenoxy)propyl]-4-methyl-1-oxo-6-(1,3,5-trimethyl-1H-pyrazol-4-yl)-3,4-dihydropyrazino[1,2-a]indol-2(1H)-yl]-1-methyl-1H-indole-5-carboxylic acid, Induced myeloid leukemia cell differentiation protein Mcl-1
著者Zhao, B.
登録日2018-12-17
公開日2019-04-17
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.85 Å)
主引用文献Discovery of Potent Myeloid Cell Leukemia-1 (Mcl-1) Inhibitors That Demonstrate in Vivo Activity in Mouse Xenograft Models of Human Cancer.
J.Med.Chem., 62, 2019
6KID
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BU of 6kid by Molmil
Crystal structure of human leucyl-tRNA synthetase, ATP-bound form
分子名称: ADENOSINE-5'-TRIPHOSPHATE, LEUCINE, Leucine--tRNA ligase, ...
著者Kim, S, Son, J, Kim, S, Hwang, K.Y.
登録日2019-07-18
公開日2021-01-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Leucine-sensing mechanism of leucyl-tRNA synthetase 1 for mTORC1 activation.
Cell Rep, 35, 2021
6KQY
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BU of 6kqy by Molmil
Crystal structure of human leucyl-tRNA synthetase, Leucine-bound form
分子名称: LEUCINE, Leucine--tRNA ligase, cytoplasmic, ...
著者Kim, S, Son, J, Kim, S, Hwang, K.Y.
登録日2019-08-20
公開日2021-01-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.3 Å)
主引用文献Leucine-sensing mechanism of leucyl-tRNA synthetase 1 for mTORC1 activation.
Cell Rep, 35, 2021
6KR7
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BU of 6kr7 by Molmil
Crystal structure of methylated human leucyl-tRNA synthetase, Leu-AMS-bound form
分子名称: 5'-O-(L-leucylsulfamoyl)adenosine, LEUCINE, Leucine--tRNA ligase, ...
著者Kim, S, Son, J, Kim, S, Hwang, K.Y.
登録日2019-08-21
公開日2021-01-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (4 Å)
主引用文献Leucine-sensing mechanism of leucyl-tRNA synthetase 1 for mTORC1 activation.
Cell Rep, 35, 2021
8K55
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BU of 8k55 by Molmil
Crystal structure of sulfur transferase from Frondihabitans sp. PAMC28461 crystallized in the P1 space group
分子名称: sulfur transferase
著者Nguyen, D.L, Do, H.
登録日2023-07-21
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2 Å)
主引用文献Structural and functional characterization of sulfurtransferase from Frondihabitans sp. PAMC28461.
Plos One, 19, 2024
8K57
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Crystal structure of sulfur transferase from Frondihabitans sp. PAMC28461 crystallized in the I21 space group
分子名称: sulfur transferase
著者Nguyen, D.L, Do, H.
登録日2023-07-21
公開日2024-04-24
実験手法X-RAY DIFFRACTION (2.38 Å)
主引用文献Structural and functional characterization of sulfurtransferase from Frondihabitans sp. PAMC28461.
Plos One, 19, 2024
6KIE
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BU of 6kie by Molmil
Crystal structure of human leucyl-tRNA synthetase, Leu-AMS-bound form
分子名称: 5'-O-(L-leucylsulfamoyl)adenosine, LEUCINE, Leucine--tRNA ligase, ...
著者Kim, S, Son, J, Kim, S, Hwang, K.Y.
登録日2019-07-18
公開日2021-01-27
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.15 Å)
主引用文献Leucine-sensing mechanism of leucyl-tRNA synthetase 1 for mTORC1 activation.
Cell Rep, 35, 2021
3VQR
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BU of 3vqr by Molmil
Structure of a dye-linked L-proline dehydrogenase mutant from the aerobic hyperthermophilic archaeon, Aeropyrum pernix
分子名称: 1,2-ETHANEDIOL, ACETATE ION, FLAVIN-ADENINE DINUCLEOTIDE, ...
著者Sakuraba, H, Ohshima, T, Satomura, T, Yoneda, K.
登録日2012-03-29
公開日2012-04-25
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.01 Å)
主引用文献Crystal Structure of Novel Dye-linked L-Proline Dehydrogenase from Hyperthermophilic Archaeon Aeropyrum pernix
J.Biol.Chem., 287, 2012
4RSU
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BU of 4rsu by Molmil
Crystal structure of the light and hvem complex
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, CHLORIDE ION, GLYCEROL, ...
著者Liu, W, Ramagoal, U.A, Himmel, D, Bonanno, J.B, Nathenson, S.G, Almo, S.C, Atoms-to-Animals: The Immune Function Network (IFN), New York Structural Genomics Research Consortium (NYSGRC)
登録日2014-11-11
公開日2015-02-04
最終更新日2023-09-20
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献HVEM structures and mutants reveal distinct functions of binding to LIGHT and BTLA/CD160.
J.Exp.Med., 218, 2021
1A57
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BU of 1a57 by Molmil
THE THREE-DIMENSIONAL STRUCTURE OF A HELIX-LESS VARIANT OF INTESTINAL FATTY ACID BINDING PROTEIN, NMR, 20 STRUCTURES
分子名称: INTESTINAL FATTY ACID-BINDING PROTEIN
著者Steele, R.A, Emmert, D.A, Kao, J, Hodsdon, M.E, Frieden, C, Cistola, D.P.
登録日1998-02-20
公開日1998-05-27
最終更新日2024-05-22
実験手法SOLUTION NMR
主引用文献The three-dimensional structure of a helix-less variant of intestinal fatty acid-binding protein.
Protein Sci., 7, 1998
7MSJ
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BU of 7msj by Molmil
The crystal structure of mouse HVEM
分子名称: SULFATE ION, Tumor necrosis factor receptor superfamily member 14
著者Liu, W, Ramagopal, U, Garrett-Thompson, S.C, Fedorov, E, Bonanno, J.B, Almo, S.C.
登録日2021-05-11
公開日2021-10-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (2.1 Å)
主引用文献HVEM structures and mutants reveal distinct functions of binding to LIGHT and BTLA/CD160.
J.Exp.Med., 218, 2021
7MSG
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BU of 7msg by Molmil
The crystal structure of LIGHT in complex with HVEM and CD160
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, CD160 antigen, soluble form,Tumor necrosis factor receptor superfamily member 14, ...
著者Liu, W, Ramagopal, U, Garrett-Thompson, S.C, Fedorov, E, Bonanno, J.B, Almo, S.C.
登録日2021-05-11
公開日2021-10-27
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (3.5 Å)
主引用文献HVEM structures and mutants reveal distinct functions of binding to LIGHT and BTLA/CD160.
J.Exp.Med., 218, 2021
7LJX
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BU of 7ljx by Molmil
Oxidized rat cytochrome c mutant (K53Q)
分子名称: Cytochrome c, somatic, HEME C, ...
著者Huttemann, M, Edwards, B.F.P, Brunzelle, J.S, Vaishnav, A.
登録日2021-02-01
公開日2021-05-12
最終更新日2023-10-18
実験手法X-RAY DIFFRACTION (1.31 Å)
主引用文献Lysine 53 Acetylation of Cytochrome c in Prostate Cancer: Warburg Metabolism and Evasion of Apoptosis.
Cells, 10, 2021
4CQG
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BU of 4cqg by Molmil
The crystal structure of MPK38 in complex with OTSSP167, an orally- administrative MELK selective inhibitor
分子名称: 1-[6-(3,5-dichloro-4-hydroxyphenyl)-4-({trans-4-[(dimethylamino)methyl]cyclohexyl}amino)-1,5-naphthyridin-3-yl]ethanone, Maternal embryonic leucine zipper kinase, SULFATE ION
著者Cho, Y.S, Kang, Y.J, Cho, H.S.
登録日2014-02-17
公開日2014-07-09
最終更新日2023-12-20
実験手法X-RAY DIFFRACTION (2.57 Å)
主引用文献The crystal structure of MPK38 in complex with OTSSP167, an orally administrative MELK selective inhibitor.
Biochem.Biophys.Res.Commun., 447, 2014
3F82
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Crystal structure of the tyrosine kinase domain of the hepatocyte growth factor receptor C-MET in complex with N-(4-(2-amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
分子名称: N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorophenyl}-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide, hepatocyte growth factor receptor
著者Sack, J.
登録日2008-11-11
公開日2009-03-31
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.5 Å)
主引用文献Discovery of N-(4-(2-Amino-3-chloropyridin-4-yloxy)-3-fluorophenyl)-4-ethoxy-1-(4-fluorophenyl)-2-oxo-1,2-dihydropyridine-3-carboxamide (BMS-777607), a Selective and Orally Efficacious Inhibitor of the Met Kinase Superfamily
J.Med.Chem., 52, 2009
5WS3
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BU of 5ws3 by Molmil
Crystal structures of human orexin 2 receptor bound to the selective antagonist EMPA determined by serial femtosecond crystallography at SACLA
分子名称: N-ethyl-2-[(6-methoxypyridin-3-yl)-(2-methylphenyl)sulfonyl-amino]-N-(pyridin-3-ylmethyl)ethanamide, OLEIC ACID, Orexin receptor type 2,GlgA glycogen synthase,Orexin receptor type 2, ...
著者Suno, R, Kimura, K, Nakane, T, Yamashita, K, Wang, J, Fujiwara, T, Yamanaka, Y, Im, D, Tsujimoto, H, Sasanuma, M, Horita, S, Hirokawa, T, Nango, E, Tono, K, Kameshima, T, Hatsui, T, Joti, Y, Yabashi, M, Shimamoto, K, Yamamoto, M, Rosenbaum, D.M, Iwata, S, Shimamura, T, Kobayashi, T.
登録日2016-12-05
公開日2017-12-13
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Crystal Structures of Human Orexin 2 Receptor Bound to the Subtype-Selective Antagonist EMPA.
Structure, 26, 2018
6LKS
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Effects of zinc ion on oligomerization and pH stability of influenza virus hemagglutinin
分子名称: 2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-[alpha-D-mannopyranose-(1-6)]beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-2)-alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ...
著者Seok, J, Kim, K.
登録日2019-12-20
公開日2020-10-21
最終更新日2023-11-22
実験手法X-RAY DIFFRACTION (3.24 Å)
主引用文献Divalent cation-induced conformational changes of influenza virus hemagglutinin.
Sci Rep, 10, 2020
8FVJ
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BU of 8fvj by Molmil
Dimeric form of HIV-1 Vif in complex with human CBF-beta, ELOB, ELOC, and CUL5
分子名称: Core-binding factor subunit beta, Cullin-5, Elongin-B, ...
著者Ito, F, Alvarez-Cabrera, A.L, Zhou, Z.H, Chen, X.S.
登録日2023-01-19
公開日2023-09-06
最終更新日2024-05-01
実験手法ELECTRON MICROSCOPY (3.54 Å)
主引用文献Structural basis of HIV-1 Vif-mediated E3 ligase targeting of host APOBEC3H.
Nat Commun, 14, 2023

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