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5CH4
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BU of 5ch4 by Molmil
Peptide-Bound State of Thermus thermophilus SecYEG
分子名称: Protein translocase subunit SecE, Protein translocase subunit SecY, Putative preprotein translocase, ...
著者Tanaka, Y, Sugano, Y, Takemoto, M, Kusakizako, T, Kumazaki, K, Ishitani, R, Nureki, O, Tsukazaki, T.
登録日2015-07-10
公開日2015-11-25
最終更新日2023-11-08
実験手法X-RAY DIFFRACTION (3.64 Å)
主引用文献Crystal Structures of SecYEG in Lipidic Cubic Phase Elucidate a Precise Resting and a Peptide-Bound State.
Cell Rep, 13, 2015
6LEO
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BU of 6leo by Molmil
Crystal structure of thiosulfate transporter YeeE from Spirochaeta thermophila
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Sulf_transp domain-containing protein, THIOSULFATE
著者Tanaka, Y, Tsukazaki, T, Yoshikaie, K, Takeuchi, A, Uchino, S, Sugano, Y.
登録日2019-11-26
公開日2020-09-02
最終更新日2020-09-30
実験手法X-RAY DIFFRACTION (2.52 Å)
主引用文献Crystal structure of a YeeE/YedE family protein engaged in thiosulfate uptake.
Sci Adv, 6, 2020
6LEP
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BU of 6lep by Molmil
Crystal structure of thiosulfate transporter YeeE inactive mutant - C91A
分子名称: (2R)-2,3-dihydroxypropyl (9Z)-octadec-9-enoate, Sulf_transp domain-containing protein, THIOSULFATE
著者Tanaka, Y, Tsukazaki, T, Yoshikaie, K, Sugano, Y, Takeuchi, A, Uchino, S.
登録日2019-11-26
公開日2020-09-02
最終更新日2024-04-03
実験手法X-RAY DIFFRACTION (2.6 Å)
主引用文献Crystal structure of a YeeE/YedE family protein engaged in thiosulfate uptake.
Sci Adv, 6, 2020
6COT
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BU of 6cot by Molmil
CSP2-d10
分子名称: Competence-stimulating peptide type 2
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2018-09-19
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6COV
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BU of 6cov by Molmil
CSP2-l14
分子名称: Competence-stimulating peptide type 2
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2018-09-19
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6COO
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BU of 6coo by Molmil
CSP1-E1A
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6COR
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BU of 6cor by Molmil
CSP1-F11A
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6CJ8
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BU of 6cj8 by Molmil
CSP1
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-02-26
公開日2018-08-29
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6COU
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BU of 6cou by Molmil
CSP2-E1Ad10
分子名称: Competence-stimulating peptide type 2
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2018-09-19
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6OLD
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BU of 6old by Molmil
CSP1-cyc(Dap6E10)
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2019-04-16
公開日2020-01-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Designing cyclic competence-stimulating peptide (CSP) analogs with pan-group quorum-sensing inhibition activity inStreptococcus pneumoniae.
Proc.Natl.Acad.Sci.USA, 117, 2020
6OC4
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BU of 6oc4 by Molmil
CSP1-cyc(Dab6E10)
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2019-03-21
公開日2020-01-08
最終更新日2020-02-05
実験手法SOLUTION NMR
主引用文献Designing cyclic competence-stimulating peptide (CSP) analogs with pan-group quorum-sensing inhibition activity inStreptococcus pneumoniae.
Proc.Natl.Acad.Sci.USA, 117, 2020
6OBW
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BU of 6obw by Molmil
CSP1-cyc(K6D10)
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2019-03-21
公開日2020-01-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Designing cyclic competence-stimulating peptide (CSP) analogs with pan-group quorum-sensing inhibition activity inStreptococcus pneumoniae.
Proc.Natl.Acad.Sci.USA, 117, 2020
6OC2
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BU of 6oc2 by Molmil
CSP1-cyc(Orn6D10)
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2019-03-21
公開日2020-01-08
最終更新日2023-06-14
実験手法SOLUTION NMR
主引用文献Designing cyclic competence-stimulating peptide (CSP) analogs with pan-group quorum-sensing inhibition activity inStreptococcus pneumoniae.
Proc.Natl.Acad.Sci.USA, 117, 2020
6COQ
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BU of 6coq by Molmil
CSP1-K6A
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
6COP
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BU of 6cop by Molmil
CSP1-R3A
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2024-05-15
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018
7OAJ
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BU of 7oaj by Molmil
Crystal structure of pseudokinase CASK in complex with compound 7
分子名称: 1,2-ETHANEDIOL, 4-(cyclopentylamino)-2-[(3,4-dichlorophenyl)methylamino]-N-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (1.93 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAI
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BU of 7oai by Molmil
Crystal structure of pseudokinase CASK in complex with PFE-PKIS12
分子名称: 1,2-ETHANEDIOL, 4-(Cyclopentylamino)-2-[(2,5-dichlorophenyl)methylamino]-N-[3-(2-oxo-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.3 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAK
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BU of 7oak by Molmil
Crystal structure of pseudokinase CASK in complex with compound 26
分子名称: 1,2-ETHANEDIOL, 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclopentylamino)-N-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.23 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAL
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BU of 7oal by Molmil
Crystal structure of pseudokinase CASK in complex with compound 25
分子名称: 1,2-ETHANEDIOL, 2-[[2,5-bis(bromanyl)-4-methyl-phenyl]methylamino]-4-(cyclohexylamino)-N-[3-(2-oxidanylidene-1,3-oxazolidin-3-yl)propyl]pyrimidine-5-carboxamide, Peripheral plasma membrane protein CASK
著者Chaikuad, A, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.17 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
7OAM
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BU of 7oam by Molmil
Kinase domain of MERTK in complex with compound 8
分子名称: 1,2-ETHANEDIOL, 2-[[2,5-bis(fluoranyl)phenyl]methylamino]-4-(cyclopentylamino)-N-[3-(2-oxidanylidenepyrrolidin-1-yl)propyl]pyrimidine-5-carboxamide, Tyrosine-protein kinase Mer
著者Schroeder, M, Russ, N, Knapp, S, Structural Genomics Consortium (SGC)
登録日2021-04-19
公開日2021-05-19
最終更新日2024-01-31
実験手法X-RAY DIFFRACTION (2.65 Å)
主引用文献Design and Development of a Chemical Probe for Pseudokinase Ca 2+ /calmodulin-Dependent Ser/Thr Kinase.
J.Med.Chem., 64, 2021
6V1N
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BU of 6v1n by Molmil
CSP1-E1A-cyc(Dap6E10)
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2019-11-20
公開日2020-01-08
最終更新日2020-02-05
実験手法SOLUTION NMR
主引用文献Designing cyclic competence-stimulating peptide (CSP) analogs with pan-group quorum-sensing inhibition activity inStreptococcus pneumoniae.
Proc.Natl.Acad.Sci.USA, 117, 2020
6DDR
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BU of 6ddr by Molmil
Crystal Structure Analysis of the Epitope of an Anti-MICA Antibody
分子名称: Anti-MICA Fab fragment heavy chain clone 13A9, Anti-MICA Fab fragment light chain clone 13A9, GLYCEROL, ...
著者Matsumoto, M.L.
登録日2018-05-10
公開日2018-10-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.9 Å)
主引用文献High-resolution glycosylation site-engineering method identifies MICA epitope critical for shedding inhibition activity of anti-MICA antibodies.
MAbs, 11, 2019
6DDM
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BU of 6ddm by Molmil
Crystal Structure Analysis of the Epitope of an Anti-MICA Antibody
分子名称: Anti-MICA Fab fragment heavy chain clone 1D5, Anti-MICA Fab fragment light chain clone 1D5, MHC class I polypeptide-related sequence A
著者Matsumoto, M.L.
登録日2018-05-10
公開日2018-10-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (1.3 Å)
主引用文献High-resolution glycosylation site-engineering method identifies MICA epitope critical for shedding inhibition activity of anti-MICA antibodies.
MAbs, 11, 2019
6DDV
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BU of 6ddv by Molmil
Crystal Structure Analysis of the Epitope of an Anti-MICA Antibody
分子名称: Anti-MICA Fab fragment heavy chain clone 6E1, Anti-MICA Fab fragment light chain clone 6E1, MHC class I chain-related protein A
著者Matsumoto, M.L.
登録日2018-05-10
公開日2018-10-24
最終更新日2023-10-11
実験手法X-RAY DIFFRACTION (2.05 Å)
主引用文献High-resolution glycosylation site-engineering method identifies MICA epitope critical for shedding inhibition activity of anti-MICA antibodies.
MAbs, 11, 2019
6COW
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BU of 6cow by Molmil
CSP1
分子名称: Competence-stimulating peptide type 1
著者Yang, Y.
登録日2018-03-12
公開日2018-08-29
最終更新日2024-05-01
実験手法SOLUTION NMR
主引用文献Structural Characterization of Competence-Stimulating Peptide Analogues Reveals Key Features for ComD1 and ComD2 Receptor Binding in Streptococcus pneumoniae.
Biochemistry, 57, 2018

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