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9Q5B

Crystal Structure of Human P38 alpha MAPK in Complex with MW01-21-114SRM

This is a non-PDB format compatible entry.
Summary for 9Q5B
Entry DOI10.2210/pdb9q5b/pdb
DescriptorMitogen-activated protein kinase 14, 4-[3-(4-FLUOROPHENYL)-1H-PYRAZOL-4-YL]PYRIDINE, (3P)-6-chloro-3-(naphthalen-2-yl)-4-(pyridin-4-yl)pyridazine, ... (5 entities in total)
Functional Keywordsp38 alpha mapk, mw01-25-195srm, transferase
Biological sourceHomo sapiens (human)
Total number of polymer chains1
Total formula weight42182.80
Authors
Minasov, G.,Brunzelle, J.S.,Roy, S.M.,Watterson, D.M.,Shuvalova, L. (deposition date: 2025-08-20, release date: 2025-09-17)
Primary citationMinasov, G.,Brunzelle, J.S.,Roy, S.M.,Watterson, D.M.,Shuvalova, L.
Crystal Structure of Human P38 alpha MAPK in Complex with MW01-21-114SRM
To Be Published,
Experimental method
X-RAY DIFFRACTION (2.05 Å)
Structure validation

245663

数据于2025-12-03公开中

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