7M6M
Full length alpha1 Glycine receptor in presence of 32uM Tetrahydrocannabinol
Summary for 7M6M
Entry DOI | 10.2210/pdb7m6m/pdb |
EMDB information | 23700 |
Descriptor | Glycine receptor subunit alphaZ1, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, (6aR,10aR)-6,6,9-trimethyl-3-pentyl-6a,7,8,10a-tetrahydro-6H-benzo[c]chromen-1-ol (3 entities in total) |
Functional Keywords | ions ligands receptors, glycine receptor recombinant proteins, membrane protein |
Biological source | Danio rerio (zebrafish) |
Total number of polymer chains | 5 |
Total formula weight | 257802.87 |
Authors | Kumar, A.,Chakrapani, S. (deposition date: 2021-03-26, release date: 2022-08-03, Last modification date: 2022-09-07) |
Primary citation | Kumar, A.,Kindig, K.,Rao, S.,Zaki, A.M.,Basak, S.,Sansom, M.S.P.,Biggin, P.C.,Chakrapani, S. Structural basis for cannabinoid-induced potentiation of alpha1-glycine receptors in lipid nanodiscs. Nat Commun, 13:4862-4862, 2022 Cited by PubMed: 35982060DOI: 10.1038/s41467-022-32594-5 PDB entries with the same primary citation |
Experimental method | ELECTRON MICROSCOPY (3.09 Å) |
Structure validation
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