7FBP
FXIIa-cMCoFx1 complex
Summary for 7FBP
Entry DOI | 10.2210/pdb7fbp/pdb |
Descriptor | Coagulation factor XIIa light chain, cMCoFx1, 2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-3)-alpha-D-mannopyranose-(1-3)-beta-D-mannopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose-(1-4)-2-acetamido-2-deoxy-beta-D-glucopyranose, ... (4 entities in total) |
Functional Keywords | serine protease, inhibitor, macrocyclic peptide, cyclotide, blood clotting |
Biological source | Homo sapiens (Human) More |
Total number of polymer chains | 2 |
Total formula weight | 30738.48 |
Authors | Sengoku, T.,Liu, W.,de Veer, S.J.,Huang, Y.H.,Okada, C.,Zdenek, C.N.,Fry, B.G.,Swedberg, J.E.,Passioura, T.,Craik, D.J.,Suga, H.,Ogata, K. (deposition date: 2021-07-12, release date: 2021-11-10, Last modification date: 2023-11-29) |
Primary citation | Liu, W.,de Veer, S.J.,Huang, Y.H.,Sengoku, T.,Okada, C.,Ogata, K.,Zdenek, C.N.,Fry, B.G.,Swedberg, J.E.,Passioura, T.,Craik, D.J.,Suga, H. An Ultrapotent and Selective Cyclic Peptide Inhibitor of Human beta-Factor XIIa in a Cyclotide Scaffold. J.Am.Chem.Soc., 143:18481-18489, 2021 Cited by PubMed: 34723512DOI: 10.1021/jacs.1c07574 PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (1.99 Å) |
Structure validation
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