6PMB
TRK-A IN COMPLEX WITH LIGAND 1a
Summary for 6PMB
Entry DOI | 10.2210/pdb6pmb/pdb |
Related | 6PMA |
Descriptor | High affinity nerve growth factor receptor, 2-[5,7-dimethyl-2-(pyridin-3-yl)[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-N-[3-(trifluoromethyl)phenyl]acetamide (3 entities in total) |
Functional Keywords | trk-a kinase domain, transferase |
Biological source | Homo sapiens (Human) |
Total number of polymer chains | 1 |
Total formula weight | 35775.14 |
Authors | Subramanian, G.,Brown, D.G. (deposition date: 2019-07-01, release date: 2020-02-26, Last modification date: 2024-03-13) |
Primary citation | Subramanian, G.,Vairagoundar, R.,Bowen, S.J.,Roush, N.,Zachary, T.,Javens, C.,Williams, T.,Janssen, A.,Gonzales, A. Synthetic inhibitor leads of human tropomyosin receptor kinase A ( h TrkA). Rsc Med Chem, 11:370-377, 2020 Cited by PubMed: 33479642DOI: 10.1039/c9md00554d PDB entries with the same primary citation |
Experimental method | X-RAY DIFFRACTION (2.81 Å) |
Structure validation
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