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6FQK

GluA2(flop) S729C ligand binding core dimer bound to ZK200775 at 1.98 Angstrom resolution

Summary for 6FQK
Entry DOI10.2210/pdb6fqk/pdb
DescriptorGlutamate receptor 2,Glutamate receptor 2, {[7-morpholin-4-yl-2,3-dioxo-6-(trifluoromethyl)-3,4-dihydroquinoxalin-1(2H)-yl]methyl}phosphonic acid (3 entities in total)
Functional Keywordsampar receptor, ligand binding domain, competitive antagonist, cross-linked dimer, membrane protein
Biological sourceRattus norvegicus (Norway Rat)
More
Total number of polymer chains2
Total formula weight61652.41
Authors
Coombs, I.D.,Soto, D.,Gold, M.G.,Farrant, M.F.,Cull-Candy, S.G. (deposition date: 2018-02-14, release date: 2019-03-13, Last modification date: 2019-10-02)
Primary citationCoombs, I.D.,Soto, D.,McGee, T.P.,Gold, M.G.,Farrant, M.,Cull-Candy, S.G.
Homomeric GluA2(R) AMPA receptors can conduct when desensitized.
Nat Commun, 10:4312-4312, 2019
Cited by
PubMed: 31541113
DOI: 10.1038/s41467-019-12280-9
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.98010442598 Å)
Structure validation

217705

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