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5ZBZ

Crystal structure of the DEAD domain of Human eIF4A with sanguinarine

Summary for 5ZBZ
Entry DOI10.2210/pdb5zbz/pdb
DescriptorEukaryotic initiation factor 4A-I, 13-methyl[1,3]benzodioxolo[5,6-c][1,3]dioxolo[4,5-i]phenanthridin-13-ium, MALONATE ION, ... (4 entities in total)
Functional Keywordseukaryotic translation initiation factor 4a, sanguinarine, inhibitor, translation, hydrolase
Biological sourceHomo sapiens (Human)
Total number of polymer chains1
Total formula weight25360.47
Authors
Ding, Y.,Ding, L. (deposition date: 2018-02-14, release date: 2019-02-20, Last modification date: 2023-11-22)
Primary citationJiang, C.,Tang, Y.,Ding, L.,Tan, R.,Li, X.,Lu, J.,Jiang, J.,Cui, Z.,Tang, Z.,Li, W.,Cao, Z.,Schneider-Poetsch, T.,Jiang, W.,Luo, C.,Ding, Y.,Liu, J.,Dang, Y.
Targeting the N Terminus of eIF4AI for Inhibition of Its Catalytic Recycling.
Cell Chem Biol, 26:1417-1426.e5, 2019
Cited by
PubMed: 31402318
DOI: 10.1016/j.chembiol.2019.07.010
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.30860259206 Å)
Structure validation

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