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5UVX

BRD4 Bromodomain 2 with A-1359643

Summary for 5UVX
Entry DOI10.2210/pdb5uvx/pdb
Related5UVS 5UVT 5UVU 5UVV 5UVW 5UVY 5UVZ
DescriptorBromodomain-containing protein 4, N-[3-(6-methyl-7-oxo-6,7-dihydro-1H-pyrrolo[2,3-c]pyridin-4-yl)-4-phenoxyphenyl]methanesulfonamide (3 entities in total)
Functional Keywordshelix bundle, signaling protein-inhibitor complex, signaling protein/inhibitor
Biological sourceHomo sapiens (Human)
Cellular locationNucleus: O60885
Total number of polymer chains2
Total formula weight26432.78
Authors
Park, C.H. (deposition date: 2017-02-20, release date: 2017-06-21, Last modification date: 2024-03-06)
Primary citationPark, C.H.
BRD4 Bromodomain 2 with A-1359643
To Be Published,
Experimental method
X-RAY DIFFRACTION (1.53 Å)
Structure validation

218853

數據於2024-04-24公開中

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