Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5T2G

mPI3Kd IN COMPLEX WITH 7i

Summary for 5T2G
Entry DOI10.2210/pdb5t2g/pdb
DescriptorPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform, 4-[3-azanyl-6-[1-methyl-5-(1-phenylcyclopropyl)-1,2,4-triazol-3-yl]pyrazin-2-yl]pyrazole-1-carboxamide (3 entities in total)
Functional Keywordsmi3kd, inhibitor, transferase
Biological sourceMus musculus (Mouse)
Cellular locationCytoplasm : O35904
Total number of polymer chains1
Total formula weight108168.03
Authors
Petersen, J.,Terstige, I.,Perry, M.,Svensson, T.,Tyrchan, C.,Lindmark, H.,Oster, L. (deposition date: 2016-08-23, release date: 2017-04-19)
Primary citationTerstiege, I.,Perry, M.,Petersen, J.,Tyrchan, C.,Svensson, T.,Lindmark, H.,Oster, L.
Discovery of triazole aminopyrazines as a highly potent and selective series of PI3K delta inhibitors.
Bioorg. Med. Chem. Lett., 27:679-687, 2017
Cited by
PubMed: 28017532
DOI: 10.1016/j.bmcl.2016.11.004
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.55 Å)
Structure validation

217705

PDB entries from 2024-03-27

PDB statisticsPDBj update infoContact PDBjnumon