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4A1Z

Eg5-1

Summary for 4A1Z
Entry DOI10.2210/pdb4a1z/pdb
Related1II6 1Q0B 1X88 1YRS 2FKY 2FL2 2FL6 2G1Q 2GM1 2UYI 2UYM 2WOG 2X2R 2X7C 2X7D 2X7E 2XAE
DescriptorKINESIN-LIKE PROTEIN KIF11, MAGNESIUM ION, NITRATE ION, ... (5 entities in total)
Functional Keywordsmotor protein
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm: P52732
Total number of polymer chains2
Total formula weight83106.27
Authors
Talapatra, S.K.,Kozielski, F. (deposition date: 2011-09-20, release date: 2012-10-31, Last modification date: 2023-12-20)
Primary citationTalapatra, S.K.,Anthony, N.G.,Mackay, S.P.,Kozielski, F.
The Mitotic Kinesin Eg5 Overcomes Inhibition to the Phase I/II Clinical Candidate Sb743921 by an Allosteric Resistance Mechanism.
J.Med.Chem., 56:6317-, 2013
Cited by
PubMed: 23875972
DOI: 10.1021/JM4006274
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (2.8 Å)
Structure validation

217705

건을2024-03-27부터공개중

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