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3KXM

Crystal structure of Z. mays CK2 kinase alpha subunit in complex with the inhibitor K74

Summary for 3KXM
Entry DOI10.2210/pdb3kxm/pdb
Related1zoh 2oxx 3KXG 3KXH 3KXJ 3KXN
DescriptorCasein kinase II subunit alpha, N-methyl-2-[(4,5,6,7-tetrabromo-1-methyl-1H-benzimidazol-2-yl)sulfanyl]acetamide (3 entities in total)
Functional Keywordsprotein kinase ck2-inhibitor complex, atp-binding, kinase, nucleotide-binding, serine/threonine-protein kinase, transferase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
Biological sourceZea mays (maize)
Total number of polymer chains1
Total formula weight39224.28
Authors
Papinutto, E.,Franchin, C.,Battistutta, R. (deposition date: 2009-12-03, release date: 2010-11-17, Last modification date: 2024-02-21)
Primary citationSarno, S.,Papinutto, E.,Franchin, C.,Bain, J.,Elliott, M.,Meggio, F.,Kazimierczuk, Z.,Orzeszko, A.,Zanotti, G.,Battistutta, R.,Pinna, L.A.
ATP site-directed inhibitors of protein kinase CK2: an update.
Curr Top Med Chem, 11:1340-1351, 2011
Cited by
PubMed: 21513497
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (1.75 Å)
Structure validation

217157

건을2024-03-13부터공개중

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