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2YCW

TURKEY BETA1 ADRENERGIC RECEPTOR WITH STABILISING MUTATIONS AND BOUND ANTAGONIST CARAZOLOL

Summary for 2YCW
Entry DOI10.2210/pdb2ycw/pdb
Related1DEP 2VT4 2Y00 2Y01 2Y02 2Y03 2Y04 2YCX 2YCY 2YCZ
DescriptorBETA-1 ADRENERGIC RECEPTOR, (2S)-1-(9H-Carbazol-4-yloxy)-3-(isopropylamino)propan-2-ol, HEGA-10, ... (4 entities in total)
Functional Keywordsgpcr, receptor, transducer, antagonist bound form, integral membrane protein, g-protein coupled receptor, thermostabilising point mutations, seven-helix receptor, 7tm receptor
Biological sourceMELEAGRIS GALLOPAVO (TURKEY)
Total number of polymer chains2
Total formula weight74045.38
Authors
Moukhametzianov, R.,Warne, T.,Edwards, P.C.,Serrano-Vega, M.J.,Leslie, A.G.W.,Tate, C.G.,Schertler, G.F.X. (deposition date: 2011-03-17, release date: 2011-06-01, Last modification date: 2023-12-20)
Primary citationMoukhametzianov, R.,Warne, T.,Edwards, P.C.,Serrano-Vega, M.J.,Leslie, A.G.,Tate, C.G.,Schertler, G.F.
Two Distinct Conformations of Helix 6 Observed in Antagonist-Bound Structures of a Beta-1- Adrenergic Receptor.
Proc.Natl.Acad.Sci.USA, 108:8228-, 2011
Cited by
PubMed: 21540331
DOI: 10.1073/PNAS.1100185108
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3 Å)
Structure validation

217705

數據於2024-03-27公開中

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