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2WTW

Aurora-A Inhibitor Structure (2nd crystal form)

Summary for 2WTW
Entry DOI10.2210/pdb2wtw/pdb
Related1MQ4 1MUO 1OL5 1OL6 1OL7 2BMC 2C6D 2C6E 2J4Z 2J50 2W1C 2W1D 2W1E 2W1F 2W1G 2WQE 2WTV
DescriptorSERINE/THREONINE-PROTEIN KINASE 6 AURORA/IPL1-RELATED KINASE 1, BREAST TUMOR-AMPLIFIED KINASE, AURORA-A, AURORA-RELATED KINASE 1, HARK1, 4-{[9-CHLORO-7-(2,6-DIFLUOROPHENYL)-5H-PYRIMIDO[5,4-D][2]BENZAZEPIN-2-YL]AMINO}BENZOIC ACID (2 entities in total)
Functional Keywordskinase, cell cycle, transferase, phosphoprotein, protein kinase
Biological sourceHOMO SAPIENS (HUMAN)
Cellular locationCytoplasm, cytoskeleton, centrosome: O14965
Total number of polymer chains1
Total formula weight33469.68
Authors
Kosmopoulou, M.,Bayliss, R. (deposition date: 2009-09-24, release date: 2010-01-26, Last modification date: 2023-12-20)
Primary citationDodson, C.A.,Kosmopoulou, M.,Richards, M.W.,Atrash, B.,Bavetsias, V.,Blagg, J.,Bayliss, R.
Crystal Structure of an Aurora-A Mutant that Mimics Aurora-B Bound to Mln8054: Insights Into Selectivity and Drug Design.
Biochem.J., 427:19-, 2010
Cited by
PubMed: 20067443
DOI: 10.1042/BJ20091530
PDB entries with the same primary citation
Experimental method
X-RAY DIFFRACTION (3.302 Å)
Structure validation

217705

数据于2024-03-27公开中

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