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1PO1

POLIOVIRUS (TYPE 1, MAHONEY) IN COMPLEX WITH R80633, AN INHIBITOR OF VIRAL REPLICATION

1PO1 の概要
エントリーDOI10.2210/pdb1po1/pdb
分子名称POLIOVIRUS TYPE 1 MAHONEY, (METHYLPYRIDAZINE PIPERIDINE BUTYLOXYPHENYL)ETHYLACETATE, MYRISTIC ACID, ... (7 entities in total)
機能のキーワードpoliovirus, picornavirus coat protein, anti-viral drugs, hydrolase, thiol protease, icosahedral virus, virus
由来する生物種Human poliovirus 1
詳細
細胞内の位置Capsid protein VP0: Virion. Capsid protein VP4: Virion. Capsid protein VP2: Virion. Capsid protein VP3: Virion. Capsid protein VP1: Virion. Protein 2B: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 2C: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 3A: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Protein 3AB: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . Viral protein genome-linked: Virion. Protease 3C: Host cytoplasm. Protein 3CD: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side . RNA-directed RNA polymerase: Host cytoplasmic vesicle membrane ; Peripheral membrane protein ; Cytoplasmic side : P03300 P03300 P03300
タンパク質・核酸の鎖数5
化学式量合計98568.21
構造登録者
Hiremath, C.N.,Filman, D.J.,Grant, R.A.,Hogle, J.M. (登録日: 1997-01-08, 公開日: 1997-12-03, 最終更新日: 2023-08-09)
主引用文献Hiremath, C.N.,Filman, D.J.,Grant, R.A.,Hogle, J.M.
Ligand-induced conformational changes in poliovirus-antiviral drug complexes.
Acta Crystallogr.,Sect.D, 53:558-570, 1997
Cited by
PubMed: 15299887
DOI: 10.1107/S0907444997000954
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (2.9 Å)
構造検証レポート
Validation report summary of 1po1
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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