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1Q8U

The Catalytic Subunit of cAMP-dependent Protein Kinase in Complex with Rho-kinase Inhibitor H-1152P

1Q8U の概要
エントリーDOI10.2210/pdb1q8u/pdb
関連するPDBエントリー1Q8T 1Q8W
分子名称cAMP-dependent protein kinase, alpha-catalytic subunit, cAMP-dependent protein kinase inhibitor, alpha form, (S)-2-METHYL-1-[(4-METHYL-5-ISOQUINOLINE)SULFONYL]-HOMOPIPERAZINE, ... (5 entities in total)
機能のキーワードkinase-inhibitor-complex, phosphotransferase/inhibitor, camp, phosphorylation, serine/threonine-protein kinase, atp-binding, pka, rho-kinase, transferase-transferase inhibitor complex, transferase/transferase inhibitor
由来する生物種Bos taurus (cattle)
詳細
細胞内の位置Cytoplasm: P00517
タンパク質・核酸の鎖数2
化学式量合計43973.06
構造登録者
Breitenlechner, C.,Gassel, M.,Hidaka, H.,Kinzel, V.,Huber, R.,Engh, R.A.,Bossemeyer, D. (登録日: 2003-08-22, 公開日: 2003-12-16, 最終更新日: 2011-07-13)
主引用文献Breitenlechner, C.,Gassel, M.,Hidaka, H.,Kinzel, V.,Huber, R.,Engh, R.A.,Bossemeyer, D.
Protein kinase A in complex with Rho-kinase inhibitors Y-27632, Fasudil, and H-1152P: structural basis of selectivity.
Structure, 11:1595-1607, 2003
Cited by
PubMed: 14656443
DOI: 10.1016/j.str.2003.11.002
主引用文献が同じPDBエントリー
実験手法
X-RAY DIFFRACTION (1.9 Å)
構造検証レポート
Validation report summary of 1q8u
検証レポート(詳細版)ダウンロードをダウンロード

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件を2024-03-27に公開中

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