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2X9E

HUMAN MPS1 IN COMPLEX WITH NMS-P715

Entity
Entity IDChain IDDescriptionTypeChain lengthFormula weightNumber of moleculesDB Name (Accession)Biological sourceDescriptive keywords
1ADUAL SPECIFICITY PROTEIN KINASE TTKpolymer31736239.71UniProt (P33981)
Pfam (PF00069)
In PDB
HOMO SAPIENS (HUMAN)MPS1, PHOSPHOTYROSINE PICKED THREONINE-PROTEIN KINASE, PYT
2AN-(2,6-DIETHYLPHENYL)-1-METHYL-8-({4-[(1-METHYLPIPERIDIN-4-YL)CARBAMOYL]-2-(TRIFLUOROMETHOXY)PHENYL}AMINO)-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDEnon-polymer676.71Chemie (SVE)
3waterwater18.02Chemie (HOH)
Sequence modifications
A: 514 - 828 (UniProt: P33981)
PDBExternal DatabaseDetails
Gly 512-expression tag
Pro 513-expression tag
Sequence viewer
Contents of the asymmetric unit
PolymersNumber of chains1
Total formula weight36239.7
Non-Polymers*Number of molecules1
Total formula weight676.7
All*Total formula weight36916.4
*Water molecules are not included.

217157

数据于2024-03-13公开中

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