2WIP
STRUCTURE OF CDK2-CYCLIN A COMPLEXED WITH 8-ANILINO-1-METHYL-4,5-DIHYDRO- 1H-PYRAZOLO[4,3-H] QUINAZOLINE-3-CARBOXYLIC ACID
Entity
Entity ID | Chain ID | Description | Type | Chain length | Formula weight | Number of molecules | DB Name (Accession) | Biological source | Descriptive keywords |
1 | A, C | CELL DIVISION PROTEIN KINASE 2 | polymer | 309 | 35251.9 | 2 | UniProt (P24941) Pfam (PF00069) In PDB | HOMO SAPIENS (HUMAN) | P33 PROTEIN KINASE |
2 | B, D | CYCLIN-A2 | polymer | 265 | 30279.0 | 2 | UniProt (P20248) Pfam (PF00134) Pfam (PF02984) In PDB | HOMO SAPIENS (HUMAN) | CYCLIN-A, CYCLIN A2 |
3 | A, C | 1-methyl-8-(phenylamino)-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxylic acid | non-polymer | 321.3 | 2 | Chemie (P49) | |||
4 | D | SULFATE ION | non-polymer | 96.1 | 1 | Chemie (SO4) | |||
5 | water | water | 18.0 | 172 | Chemie (HOH) |
Sequence modifications
A, C: -4 - 0 (PDB: 2WIP)
A, C: 299 - 304 (PDB: 2WIP)
A, C: 1 - 298 (UniProt: P24941)
B, D: 168 - 172 (PDB: 2WIP)
B, D: 173 - 432 (UniProt: P20248)
A, C: 299 - 304 (PDB: 2WIP)
A, C: 1 - 298 (UniProt: P24941)
B, D: 168 - 172 (PDB: 2WIP)
B, D: 173 - 432 (UniProt: P20248)
Sequence viewer
Contents of the asymmetric unit
Polymers | Number of chains | 4 |
Total formula weight | 131061.7 | |
Non-Polymers* | Number of molecules | 3 |
Total formula weight | 738.7 | |
All* | Total formula weight | 131800.4 |