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8PX7
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BU of 8px7 by Molmil
Structure of Bacterial Multidrug Efflux transporter AcrB, solved at wavelength 3.02 A
Descriptor: Multidrug efflux pump subunit AcrB
Authors:El Omari, K, Duman, R, Mykhaylyk, V, Orr, C, Qu, F, Beis, K, Wagner, A.
Deposit date:2023-07-22
Release date:2023-10-25
Method:X-RAY DIFFRACTION (3.4 Å)
Cite:Experimental phasing opportunities for macromolecular crystallography at very long wavelengths.
Commun Chem, 6, 2023
7WLV
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BU of 7wlv by Molmil
Crystal Structure of the Multidrug effulx transporter BpeF from Burkholderia pseudomallei.
Descriptor: DODECYL-BETA-D-MALTOSIDE, Efflux pump membrane transporter
Authors:Kato, T, Hung, L.-W, Yamashita, E, Okada, U, Terwilliger, T.C, Murakami, S.
Deposit date:2022-01-13
Release date:2023-07-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (3 Å)
Cite:Crystal structures of multidrug efflux transporters from Burkholderia pseudomallei suggest details of transport mechanism.
Proc.Natl.Acad.Sci.USA, 120, 2023
7WLS
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BU of 7wls by Molmil
Crystal structure of the multidrug efflux transporter BpeB from Burkholderia pseudomallei
Descriptor: Efflux pump membrane transporter, TETRAETHYLENE GLYCOL, UNDECYL-MALTOSIDE
Authors:Kato, T, Hung, L.-W, Yamashita, E, Okada, U, Terwilliger, T.C, Murakami, S.
Deposit date:2022-01-13
Release date:2023-07-19
Last modified:2023-11-29
Method:X-RAY DIFFRACTION (2.94 Å)
Cite:Crystal structures of multidrug efflux transporters from Burkholderia pseudomallei suggest details of transport mechanism.
Proc.Natl.Acad.Sci.USA, 120, 2023
8GK0
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BU of 8gk0 by Molmil
Multi-drug efflux pump RE-CmeB bound with Erythromycin
Descriptor: ERYTHROMYCIN A, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2023-03-16
Release date:2023-06-07
Last modified:2023-10-04
Method:ELECTRON MICROSCOPY (3.44 Å)
Cite:Cryo-Electron Microscopy Structures of a Campylobacter Multidrug Efflux Pump Reveal a Novel Mechanism of Drug Recognition and Resistance.
Microbiol Spectr, 11, 2023
8GJL
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BU of 8gjl by Molmil
multi-drug efflux pump RE-CmeB bound with Ciprofloxacin
Descriptor: 1-CYCLOPROPYL-6-FLUORO-4-OXO-7-PIPERAZIN-1-YL-1,4-DIHYDROQUINOLINE-3-CARBOXYLIC ACID, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2023-03-16
Release date:2023-05-31
Last modified:2023-10-04
Method:ELECTRON MICROSCOPY (3.44 Å)
Cite:Cryo-Electron Microscopy Structures of a Campylobacter Multidrug Efflux Pump Reveal a Novel Mechanism of Drug Recognition and Resistance.
Microbiol Spectr, 11, 2023
8GK4
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BU of 8gk4 by Molmil
Multi-drug efflux pump RE-CmeB bound with Chloramphenicol
Descriptor: CHLORAMPHENICOL, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2023-03-17
Release date:2023-05-31
Last modified:2023-10-04
Method:ELECTRON MICROSCOPY (3.12 Å)
Cite:Cryo-Electron Microscopy Structures of a Campylobacter Multidrug Efflux Pump Reveal a Novel Mechanism of Drug Recognition and Resistance.
Microbiol Spectr, 11, 2023
8GJJ
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BU of 8gjj by Molmil
Multi-drug efflux pump RE-CmeB Apo form
Descriptor: Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2023-03-15
Release date:2023-05-31
Last modified:2023-10-04
Method:ELECTRON MICROSCOPY (3.08 Å)
Cite:Cryo-Electron Microscopy Structures of a Campylobacter Multidrug Efflux Pump Reveal a Novel Mechanism of Drug Recognition and Resistance.
Microbiol Spectr, 11, 2023
8GJK
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BU of 8gjk by Molmil
Multi-drug efflux pump RE-CmeB bound with ampicillin
Descriptor: (2R,4S)-2-[(R)-{[(2R)-2-amino-2-phenylacetyl]amino}(carboxy)methyl]-5,5-dimethyl-1,3-thiazolidine-4-carboxylic acid, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2023-03-16
Release date:2023-05-31
Last modified:2023-10-04
Method:ELECTRON MICROSCOPY (3.16 Å)
Cite:Cryo-Electron Microscopy Structures of a Campylobacter Multidrug Efflux Pump Reveal a Novel Mechanism of Drug Recognition and Resistance.
Microbiol Spectr, 11, 2023
8FFK
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BU of 8ffk by Molmil
Klebsiella pneumoniae AcrB multidrug efflux pump apo form
Descriptor: Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-12-08
Release date:2023-04-05
Last modified:2023-07-12
Method:ELECTRON MICROSCOPY (2.82 Å)
Cite:Cryo-EM Structures of the Klebsiella pneumoniae AcrB Multidrug Efflux Pump.
Mbio, 14, 2023
8FFS
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BU of 8ffs by Molmil
Erythromycin bound Klebsiella pneumoniae AcrB multidrug efflux pump
Descriptor: ERYTHROMYCIN A, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-12-09
Release date:2023-04-05
Last modified:2023-07-12
Method:ELECTRON MICROSCOPY (2.96 Å)
Cite:Cryo-EM Structures of the Klebsiella pneumoniae AcrB Multidrug Efflux Pump.
Mbio, 14, 2023
8F4R
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BU of 8f4r by Molmil
Gentamicin bound aminoglycoside efflux pump AcrD
Descriptor: (2R,3R,4R,5R)-2-((1S,2S,3R,4S,6R)-4,6-DIAMINO-3-((2R,3R,6S)-3-AMINO-6-(AMINOMETHYL)-TETRAHYDRO-2H-PYRAN-2-YLOXY)-2-HYDR OXYCYCLOHEXYLOXY)-5-METHYL-4-(METHYLAMINO)-TETRAHYDRO-2H-PYRAN-3,5-DIOL, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-11-11
Release date:2022-12-28
Last modified:2023-03-08
Method:ELECTRON MICROSCOPY (3.06 Å)
Cite:Cryo-EM Structures of AcrD Illuminate a Mechanism for Capturing Aminoglycosides from Its Central Cavity.
Mbio, 14, 2023
8F3E
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BU of 8f3e by Molmil
Trimer of aminoglycoside efflux pump AcrD
Descriptor: Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-11-10
Release date:2022-12-28
Last modified:2023-03-08
Method:ELECTRON MICROSCOPY (3.09 Å)
Cite:Cryo-EM Structures of AcrD Illuminate a Mechanism for Capturing Aminoglycosides from Its Central Cavity.
Mbio, 14, 2023
8F56
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BU of 8f56 by Molmil
Dimer of aminoglycoside efflux pump AcrD treated with gentamicin
Descriptor: Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-11-11
Release date:2022-12-28
Last modified:2023-03-08
Method:ELECTRON MICROSCOPY (2.98 Å)
Cite:Cryo-EM Structures of AcrD Illuminate a Mechanism for Capturing Aminoglycosides from Its Central Cavity.
Mbio, 14, 2023
8F4N
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BU of 8f4n by Molmil
Dimer of aminoglycoside efflux pump AcrD
Descriptor: Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2022-11-11
Release date:2022-12-28
Last modified:2023-03-08
Method:ELECTRON MICROSCOPY (2.95 Å)
Cite:Cryo-EM Structures of AcrD Illuminate a Mechanism for Capturing Aminoglycosides from Its Central Cavity.
Mbio, 14, 2023
8DEW
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BU of 8dew by Molmil
Cryo-electron microscopy structure of Neisseria gonorrhoeae multidrug efflux pump MtrD with LL-37 complex
Descriptor: Antibacterial peptide LL-37, Efflux pump membrane transporter, PHOSPHATIDYLETHANOLAMINE
Authors:Lyu, M, Yu, E.W.
Deposit date:2022-06-21
Release date:2022-09-14
Last modified:2022-11-09
Method:ELECTRON MICROSCOPY (2.89 Å)
Cite:Structural Basis of Peptide-Based Antimicrobial Inhibition of a Resistance-Nodulation-Cell Division Multidrug Efflux Pump.
Microbiol Spectr, 10, 2022
8DEV
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BU of 8dev by Molmil
Cryo-electron microscopy structure of Neisseria gonorrhoeae multidrug efflux pump MtrD with colistin complex
Descriptor: Colistin, Efflux pump membrane transporter, PHOSPHATIDYLETHANOLAMINE
Authors:Lyu, M, Yu, E.W.
Deposit date:2022-06-21
Release date:2022-09-14
Last modified:2022-11-09
Method:ELECTRON MICROSCOPY (3.08 Å)
Cite:Structural Basis of Peptide-Based Antimicrobial Inhibition of a Resistance-Nodulation-Cell Division Multidrug Efflux Pump.
Microbiol Spectr, 10, 2022
8DEU
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BU of 8deu by Molmil
Cryo-electron microscopy structure of Neisseria gonorrhoeae multidrug efflux pump MtrD with CASP peptide complex
Descriptor: CASP peptide, Efflux pump membrane transporter, PHOSPHATIDYLETHANOLAMINE
Authors:Lyu, M, Yu, E.W.
Deposit date:2022-06-21
Release date:2022-09-14
Last modified:2022-11-09
Method:ELECTRON MICROSCOPY (2.95 Å)
Cite:Structural Basis of Peptide-Based Antimicrobial Inhibition of a Resistance-Nodulation-Cell Division Multidrug Efflux Pump.
Microbiol Spectr, 10, 2022
7RR7
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BU of 7rr7 by Molmil
Multidrug efflux pump subunit AcrB
Descriptor: DODECANE, Multidrug efflux pump subunit AcrB, PHOSPHATIDYLETHANOLAMINE
Authors:Trinh, T.K.H, Cabezas, A, Catalano, C, Qiu, W, des Georges, A, Guo, Y.
Deposit date:2021-08-09
Release date:2022-08-17
Method:ELECTRON MICROSCOPY (3.05 Å)
Cite:Multidrug efflux pump subunit AcrB
To Be Published
7RR8
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BU of 7rr8 by Molmil
Multidrug efflux pump subunit AcrB
Descriptor: DODECANE, Multidrug efflux pump subunit AcrB, PHOSPHATIDYLETHANOLAMINE
Authors:Trinh, T.K.H, Cabezas, A, Catalano, C, Qiu, W, des Georges, A, Guo, Y.
Deposit date:2021-08-09
Release date:2022-08-17
Method:ELECTRON MICROSCOPY (3.51 Å)
Cite:Multidrug efflux pump subunit AcrB
To Be Published
7RR6
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BU of 7rr6 by Molmil
Multidrug efflux pump subunit AcrB
Descriptor: DODECANE, Multidrug efflux pump subunit AcrB, PHOSPHATIDYLETHANOLAMINE
Authors:Trinh, T.K.H, Cabezas, A, Catalano, C, Qiu, W, des Georges, A, Guo, Y.
Deposit date:2021-08-09
Release date:2022-08-17
Method:ELECTRON MICROSCOPY (3.1 Å)
Cite:Multidrug efflux pump subunit AcrB
To Be Published
7O3M
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BU of 7o3m by Molmil
Crystal Structure of AcrB Single Mutant - 1
Descriptor: DODECYL-BETA-D-MALTOSIDE, Efflux pump membrane transporter
Authors:Ababou, A.
Deposit date:2021-04-02
Release date:2022-04-13
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (3.551 Å)
Cite:Crystal Structure of AcrB Single Mutant - 1
To Be Published
7O3L
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BU of 7o3l by Molmil
Crystal Structure of AcrB Double Mutant
Descriptor: DODECYL-BETA-D-MALTOSIDE, Efflux pump membrane transporter
Authors:Ababou, A.
Deposit date:2021-04-02
Release date:2022-04-13
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (3.526 Å)
Cite:Crystal Structure of AcrB Double Mutant
To Be Published
7O3N
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BU of 7o3n by Molmil
Crystal Structure of AcrB Single Mutant - 2
Descriptor: DODECYL-BETA-D-MALTOSIDE, Efflux pump membrane transporter
Authors:Ababou, A.
Deposit date:2021-04-02
Release date:2022-04-13
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (3.561 Å)
Cite:Crystal Structure of AcrB Single Mutant - 2
To Be Published
7RY3
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BU of 7ry3 by Molmil
Multidrug Efflux pump AdeJ with TP-6076 bound
Descriptor: (4S,4aS,5aR,12aS)-4-(diethylamino)-3,10,12,12a-tetrahydroxy-1,11-dioxo-8-[(2S)-pyrrolidin-2-yl]-7-(trifluoromethyl)-1,4,4a,5,5a,6,11,12a-octahydrotetracene-2-carboxamide, Efflux pump membrane transporter
Authors:Zhang, Z.
Deposit date:2021-08-24
Release date:2022-02-02
Last modified:2022-12-07
Method:ELECTRON MICROSCOPY (2.91 Å)
Cite:An Analysis of the Novel Fluorocycline TP-6076 Bound to Both the Ribosome and Multidrug Efflux Pump AdeJ from Acinetobacter baumannii.
Mbio, 13, 2022
7OUK
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BU of 7ouk by Molmil
BDM88855 inhibitor bound to the transmembrane domain of AcrB
Descriptor: (2S)-3-hydroxypropane-1,2-diyl didecanoate, (2S)-3-{[(R)-(2-aminoethoxy)(hydroxy)phosphoryl]oxy}-2-hydroxypropyl hexadecanoate, 1,2-ETHANEDIOL, ...
Authors:Tam, H.K, Foong, W.E, Pos, K.M.
Deposit date:2021-06-12
Release date:2021-12-29
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.6 Å)
Cite:Pyridylpiperazine-based allosteric inhibitors of RND-type multidrug efflux pumps.
Nat Commun, 13, 2022

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PDB entries from 2024-03-27

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