5P9N | |
5P9O | HUMANIZED RAT COMT IN COMPLEX WITH 7-FLUORO-5,6-BIS(4-FLUOROPHENYL)-8-HYDROXY-3H-QUINAZOLIN-4-ONE | Descriptor: | Catechol O-methyltransferase, 7-fluoranyl-5,6-bis(4-fluorophenyl)-8-oxidanyl-3~{H}-quinazolin-4-one, S-ADENOSYL-L-HOMOCYSTEINE, ... | Authors: | Ehler, A., Lerner, C., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-03-21 | Method: | X-RAY DIFFRACTION (1.1 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5P9P | |
5P9Q | HUMANIZED RAT COMT IN COMPLEX WITH 6-(2,4-DIMETHYL-1,3-THIAZOL-5-YL)-8-HYDROXY-3H-QUINAZOLIN-4-ONE | Descriptor: | Catechol O-methyltransferase, MAGNESIUM ION, CHLORIDE ION, ... | Authors: | Ehler, A., Jakob-Roetne, R., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-02-21 | Method: | X-RAY DIFFRACTION (1.63 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5P9R | |
5P9S | |
5P9T | |
5P9U | |
5P9V | |
5P9W | RAT CATECHOL O-METHYLTRANSFERASE IN COMPLEX WITH 4'-FLUORO-4,5-DIHYDROXY-N-{[(1R,2R)-2-{(2S,4R,5R)-4-HYDROXY-5-[6-(METHYLAMINO)-9H-PURIN-9-YL]OXOLAN-2-YL}CYCLOPROPYL]METHYL}[1,1'-BIPHENYL]-3-CARBOXAMIDE | Descriptor: | Catechol O-methyltransferase, MAGNESIUM ION, CHLORIDE ION, ... | Authors: | Ehler, A., Lerner, C., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-03-21 | Method: | X-RAY DIFFRACTION (1.43 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5P9X | HUMANIZED RAT CATECHOL O-METHYLTRANSFERASE IN COMPLEX WITH N-[1-[(2R,3S,4R,5R)-5-(6-AMINOPURIN-9-YL)-3,4-DIHYDROXYOXOLAN-2-YL]PROPAN-2-YL]-5-(4-FLUOROPHENYL)-2,3-DIHYDROXYBENZAMIDE | Descriptor: | Catechol O-methyltransferase, MAGNESIUM ION, CHLORIDE ION, ... | Authors: | Ehler, A., Lerner, C., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-02-21 | Method: | X-RAY DIFFRACTION (1.12 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5P9Y | HUMANIZED RAT CATECHOL O-METHYLTRANSFERASE IN COMPLEX WITH 6-(4-FLUOROPHENYL)-8-HYDROXY-3-(5-PYRROLO[3,2-C]PYRIDIN-1-YLPENTYL)QUINAZOLIN-4-ONE | Descriptor: | Catechol O-methyltransferase, MAGNESIUM ION, 6-(4-fluorophenyl)-8-oxidanyl-3-(5-pyrrolo[3,2-c]pyridin-1-ylpentyl)quinazolin-4-one, ... | Authors: | Ehler, A., Lerner, C., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-02-21 | Method: | X-RAY DIFFRACTION (1.2 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5P9Z | |
5PA0 | |
5PA1 | |
5PA2 | |
5PA3 | |
5PA4 | |
5PA5 | HUMANIZED RAT COMT IN COMPLEX WITH 6-(2,4-DIMETHYL-1,3-THIAZOL-5-YL)-8-HYDROXY-3H-QUINAZOLIN-4-ONE | Descriptor: | Catechol O-methyltransferase, MAGNESIUM ION, CHLORIDE ION, ... | Authors: | Ehler, A., Lerner, C., Rudolph, M.G. | Deposit date: | 2016-10-19 | Release date: | 2017-11-22 | Last modified: | 2018-02-21 | Method: | X-RAY DIFFRACTION (1.63 Å) | Cite: | Crystal Structure of a COMT complex To be published
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5PA6 | |
5PA7 | |