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7R50
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BU of 7r50 by Molmil
Crystal structure of GMP reductase from mycobacterium smegmatis in complex with GMP.
Descriptor: GUANOSINE-5'-MONOPHOSPHATE, Inosine-5-monophosphate dehydrogenase guaB1
Authors:Dolezal, M, Klima, M, Pichova, I.
Deposit date:2022-02-09
Release date:2022-04-27
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.5 Å)
Cite:The mycobacterial guaB1 gene encodes a guanosine 5'-monophosphate reductase with a cystathionine-beta-synthase domain.
Febs J., 289, 2022
7QGT
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BU of 7qgt by Molmil
Crystal structure of human cystathionine beta-synthase (delta516-525) in complex with AOAA.
Descriptor: 4'-DEOXY-4'-ACETYLYAMINO-PYRIDOXAL-5'-PHOSPHATE, Cystathionine beta-synthase, PROTOPORPHYRIN IX CONTAINING FE, ...
Authors:Hutchin, A, Kopec, J, Majtan, T, Zuhra, K, Szabo, C.
Deposit date:2021-12-10
Release date:2022-10-19
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.691 Å)
Cite:H 2 S biogenesis by cystathionine beta-synthase: mechanism of inhibition by aminooxyacetic acid and unexpected role of serine.
Cell.Mol.Life Sci., 79, 2022
7QEM
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BU of 7qem by Molmil
bacterial IMPDH chimera
Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase
Authors:Labesse, G, Gelin, M, Gedeon, A, Haouz, A, Munier-Lehmann, H.
Deposit date:2021-12-03
Release date:2023-06-14
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (3.09 Å)
Cite:Insight into the role of the Bateman domain at the molecular and physiological levels through engineered IMP dehydrogenases.
Protein Sci., 32, 2023
7QDX
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BU of 7qdx by Molmil
bacterial IMPDH chimera
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, Inosine-5'-monophosphate dehydrogenase, MAGNESIUM ION
Authors:Labesse, G, Gelin, M, Munier-Lehmann, H, Gedeon, A, Haouz, A.
Deposit date:2021-11-30
Release date:2023-06-14
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.9 Å)
Cite:Insight into the role of the Bateman domain at the molecular and physiological levels through engineered IMP dehydrogenases.
Protein Sci., 32, 2023
7QBJ
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BU of 7qbj by Molmil
bacterial IMPDH chimera
Descriptor: Inosine-5'-monophosphate dehydrogenase
Authors:Labesse, G, Gelin, M, Munier-Lehmann, H, Gedeon, A, Haouz, A.
Deposit date:2021-11-19
Release date:2023-05-31
Last modified:2024-02-07
Method:X-RAY DIFFRACTION (2.27 Å)
Cite:Insight into the role of the Bateman domain at the molecular and physiological levels through engineered IMP dehydrogenases.
Protein Sci., 32, 2023
7PMZ
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BU of 7pmz by Molmil
Crystal structure of Streptomyces coelicolor guaB (IMP dehydrogenase) bound to ATP and ppGpp at 2.0 A resolution
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5',3'-TETRAPHOSPHATE, Inosine-5'-monophosphate dehydrogenase, ...
Authors:Fernandez-Justel, D, Revuelta, J.L, Buey, R.M.
Deposit date:2021-09-04
Release date:2022-05-11
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.03 Å)
Cite:Diversity of mechanisms to control bacterial GTP homeostasis by the mutually exclusive binding of adenine and guanine nucleotides to IMP dehydrogenase.
Protein Sci., 31, 2022
7PJI
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BU of 7pji by Molmil
Crystal structure of Pseudomonas aeruginosa guaB (IMP dehydrogenase) bound to ATP and GDP at 1.65A resolution
Descriptor: ACETATE ION, ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-DIPHOSPHATE, ...
Authors:Fernandez-Justel, D, Buey, R.M.
Deposit date:2021-08-24
Release date:2022-07-06
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (1.65 Å)
Cite:Diversity of mechanisms to control bacterial GTP homeostasis by the mutually exclusive binding of adenine and guanine nucleotides to IMP dehydrogenase.
Protein Sci., 31, 2022
7RGQ
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BU of 7rgq by Molmil
HUMAN RETINAL VARIANT IMPDH1(546) TREATED WITH GTP, ATP, IMP, NAD+; INTERFACE-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-15
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (3.9 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RGI
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BU of 7rgi by Molmil
HUMAN RETINAL VARIANT IMPDH1(546) TREATED WITH GTP, ATP, IMP, NAD+; INTERFACE-CENTERED
Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase 1, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-15
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (3.6 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RGD
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BU of 7rgd by Molmil
HUMAN RETINAL VARIANT IMPDH1(595) TREATED WITH GTP, ATP, IMP, NAD+, OCTAMER-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-15
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (3 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RGL
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BU of 7rgl by Molmil
HUMAN RETINAL VARIANT IMPDH1(546) TREATED WITH ATP, IMP, NAD+, INTERFACE-CENTERED
Descriptor: INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase 1, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-15
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.4 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RGM
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BU of 7rgm by Molmil
HUMAN RETINAL VARIANT IMPDH1(546) TREATED WITH ATP, IMP, NAD+, OCTAMER-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, Inosine-5'-monophosphate dehydrogenase 1, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-15
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.8 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RFI
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BU of 7rfi by Molmil
HUMAN RETINAL VARIANT IMPDH1(595) TREATED WITH GTP, ATP, IMP, NAD+, INTERFACE-CENTERED
Descriptor: GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, Isoform 5 of Inosine-5'-monophosphate dehydrogenase 1, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-14
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.6 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RFE
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BU of 7rfe by Molmil
HUMAN IMPDH1 TREATED WITH GTP, IMP, AND NAD+; INTERFACE-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-14
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.6 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RFH
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BU of 7rfh by Molmil
HUMAN RETINAL VARIANT IMPDH1(595) TREATED WITH ATP, OCTAMER-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, Isoform 5 of Inosine-5'-monophosphate dehydrogenase 1
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-14
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (3.7 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RFF
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BU of 7rff by Molmil
HUMAN RETINAL VARIANT IMPDH1(595) TREATED WITH ATP; INTERFACE-CENTERED
Descriptor: Isoform 5 of Inosine-5'-monophosphate dehydrogenase 1
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-14
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.7 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RFG
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BU of 7rfg by Molmil
HUMAN IMPDH1 TREATED WITH GTP, IMP, AND NAD+ OCTAMER-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, GUANOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-14
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.6 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RER
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BU of 7rer by Molmil
HUMAN IMPDH1 TREATED WITH ATP, IMP, AND NAD+
Descriptor: INOSINIC ACID, Isoform 5 of Inosine-5'-monophosphate dehydrogenase 1, NICOTINAMIDE-ADENINE-DINUCLEOTIDE
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-13
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (2.6 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7RES
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BU of 7res by Molmil
HUMAN IMPDH1 TREATED WITH ATP, IMP, AND NAD+, OCTAMER-CENTERED
Descriptor: ADENOSINE-5'-TRIPHOSPHATE, INOSINIC ACID, Isoform 5 of Inosine-5'-monophosphate dehydrogenase 1, ...
Authors:Burrell, A.L, Kollman, J.M.
Deposit date:2021-07-13
Release date:2022-01-12
Last modified:2022-02-02
Method:ELECTRON MICROSCOPY (3.05 Å)
Cite:IMPDH1 retinal variants control filament architecture to tune allosteric regulation.
Nat.Struct.Mol.Biol., 29, 2022
7OY9
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BU of 7oy9 by Molmil
Crystal structure of GMP reductase from mycobacterium smegmatis.
Descriptor: Guanosine 5'-monophosphate reductase
Authors:Dolezal, M, Klima, M, Pichova, I.
Deposit date:2021-06-24
Release date:2022-04-27
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.8 Å)
Cite:The mycobacterial guaB1 gene encodes a guanosine 5'-monophosphate reductase with a cystathionine-beta-synthase domain.
Febs J., 289, 2022
7MYJ
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BU of 7myj by Molmil
Structure of full length human AMPK (a2b1g1) in complex with a small molecule activator MSG011
Descriptor: (5S,6R,7R,9R,13cR,14R,16aS)-6-methoxy-5-methyl-7-(methylamino)-6,7,8,9,14,15,16,16a-octahydro-5H,13cH-5,9-epoxy-4b,9a,1 5-triazadibenzo[b,h]cyclonona[1,2,3,4-jkl]cyclopenta[e]-as-indacen-14-ol, 5'-AMP-activated protein kinase catalytic subunit alpha-2, 5'-AMP-activated protein kinase subunit beta-1, ...
Authors:Ovens, A.J, Gee, Y.S, Ling, N.X.Y, Waters, N.J, Yu, D, Scott, J.W, Parker, M.W, Hoffman, N.J, Kemp, B.E, Baell, J.B, Oakhill, J.S, Langendorf, C.G.
Deposit date:2021-05-21
Release date:2022-06-29
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.95 Å)
Cite:Structure-function analysis of the AMPK activator SC4 and identification of a potent pan AMPK activator.
Biochem.J., 479, 2022
7OJ1
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BU of 7oj1 by Molmil
Bacillus subtilis IMPDH in complex with Ap4A
Descriptor: BIS(ADENOSINE)-5'-TETRAPHOSPHATE, Inosine-5'-monophosphate dehydrogenase, MAGNESIUM ION
Authors:Giammarinaro, P.I, Bange, G.
Deposit date:2021-05-13
Release date:2022-09-14
Last modified:2024-01-31
Method:X-RAY DIFFRACTION (2.44 Å)
Cite:Diadenosine tetraphosphate regulates biosynthesis of GTP in Bacillus subtilis.
Nat Microbiol, 7, 2022
7MSU
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BU of 7msu by Molmil
Crystal structure of an archaeal CNNM, MtCorB, CBS-pair domain in complex with Mg2+-ATP
Descriptor: 1,2-ETHANEDIOL, ADENOSINE-5'-TRIPHOSPHATE, Hemolysin, ...
Authors:Chen, Y.S, Gehring, K.
Deposit date:2021-05-12
Release date:2021-06-16
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (2.07 Å)
Cite:Crystal structure of an archaeal CorB magnesium transporter.
Nat Commun, 12, 2021
7M74
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BU of 7m74 by Molmil
ATP-bound AMP-activated protein kinase
Descriptor: 5'-AMP-activated protein kinase catalytic subunit alpha-1, 5'-AMP-activated protein kinase subunit beta-2, 5'-AMP-activated protein kinase subunit gamma-1, ...
Authors:Yan, Y, Mukherjee, S, Harikumar, K.G, Strutzenberg, T, Zhou, X.E, Powell, S.K, Xu, T, Sheldon, R, Lamp, J, Brunzelle, J.S, Radziwon, K, Ellis, A, Novick, S.J, Vega, I.E, Jones, R, Miller, L.J, Xu, H.E, Griffin, P.R, Kossiakoff, A.A, Melcher, K.
Deposit date:2021-03-26
Release date:2021-12-15
Last modified:2021-12-22
Method:ELECTRON MICROSCOPY (3.93 Å)
Cite:Structure of an AMPK complex in an inactive, ATP-bound state.
Science, 373, 2021
7M1U
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BU of 7m1u by Molmil
Crystal structure of an archaeal CNNM, MtCorB, R235L mutant with C-terminal deletion
Descriptor: Hemolysin, contains CBS domains
Authors:Chen, Y.S, Kozlov, G, Gehring, K.
Deposit date:2021-03-15
Release date:2021-06-16
Last modified:2023-10-18
Method:X-RAY DIFFRACTION (3.8 Å)
Cite:Crystal structure of an archaeal CorB magnesium transporter.
Nat Commun, 12, 2021

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PDB entries from 2024-03-27

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