6PET
Crystal structure of 8-hydroxychromene compound 30 bound to estrogen receptor alpha
PDBデータベースに由来する情報
site_id | AC1 |
残基数 | 10 |
詳細 | binding site for residue G9J D 601 |
鎖名 | 残基 |
D | LEU346 |
D | LEU525 |
D | THR347 |
D | ALA350 |
D | GLU353 |
D | LEU387 |
D | ARG394 |
D | ILE424 |
D | GLY521 |
D | HIS524 |
site_id | AC2 |
残基数 | 12 |
詳細 | binding site for residue ODY A 601 |
鎖名 | 残基 |
A | LEU346 |
A | LEU349 |
A | ALA350 |
A | ASP351 |
A | GLU353 |
A | TRP383 |
A | MET421 |
A | ILE424 |
A | GLY521 |
A | HIS524 |
A | LEU525 |
A | VAL533 |
site_id | AC3 |
残基数 | 11 |
詳細 | binding site for residue G9J C 601 |
鎖名 | 残基 |
C | LEU346 |
C | THR347 |
C | ALA350 |
C | GLU353 |
C | LEU387 |
C | ARG394 |
C | PHE404 |
C | MET421 |
C | ILE424 |
C | HIS524 |
C | HOH715 |
site_id | AC4 |
残基数 | 12 |
詳細 | binding site for residue ODY B 601 |
鎖名 | 残基 |
B | LEU346 |
B | THR347 |
B | LEU349 |
B | ALA350 |
B | ASP351 |
B | GLU353 |
B | LEU387 |
B | LEU391 |
B | MET421 |
B | GLY521 |
B | HIS524 |
B | LEU525 |
site_id | AC5 |
残基数 | 4 |
詳細 | binding site for residue DMS B 602 |
鎖名 | 残基 |
B | LEU320 |
B | GLU323 |
B | TRP393 |
B | GLY442 |
SwissProt/UniProtに記載されている蛋白質分子機能情報
site_id | SWS_FT_FI1 |
残基数 | 4 |
詳細 | MOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106 |
鎖名 | 残基 | 詳細 |
D | TYR537 | |
A | TYR537 | |
C | TYR537 | |
B | TYR537 |
site_id | SWS_FT_FI2 |
残基数 | 4 |
詳細 | LIPID: S-palmitoyl cysteine => ECO:0000250 |
鎖名 | 残基 | 詳細 |
D | CYS447 | |
A | CYS447 | |
C | CYS447 | |
B | CYS447 |