Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

6O0M

crystal structure of BCL-2 F104L mutation with venetoclax

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
A0043066biological_processnegative regulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues24
Detailsbinding site for residue LBM A 301
ChainResidue
AARG12
ATRP144
AGLY145
AVAL148
AALA149
AGLU152
APHE153
AVAL156
AGLN190
APHE198
ATYR202
AALA100
APEG302
APEG305
AHOH405
AHOH446
AHOH458
AASP103
ALEU104
AARG107
APHE112
AMET115
AGLU136
AASN143

site_idAC2
Number of Residues3
Detailsbinding site for residue PEG A 302
ChainResidue
ATYR108
ALBM301
APEG303

site_idAC3
Number of Residues8
Detailsbinding site for residue PEG A 303
ChainResidue
AARG12
AMET16
AALA174
ALEU175
ATHR178
APEG302
AHOH423
AHOH433

site_idAC4
Number of Residues6
Detailsbinding site for residue PEG A 304
ChainResidue
AARG127
APHE130
AASN163
ATRP176
ATYR180
AHOH439

site_idAC5
Number of Residues4
Detailsbinding site for residue PEG A 305
ChainResidue
AARG12
AASP191
ALBM301
AHOH409

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues19
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. LFrDGv.NWGRIVAFFeFGG
ChainResidueDetails
ALEU137-GLY155

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WIqdnGGWDaFV
ChainResidueDetails
ATRP188-VAL199

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. VhltLRqAGDDLSRR
ChainResidueDetails
AVAL93-ARG107

site_idPS01260
Number of Residues21
DetailsBH4_1 Apoptosis regulator, Bcl-2 family BH4 motif signature. DNREIVmKYIHYKLSQRGYeW
ChainResidueDetails
AASP10-TRP30

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Cleavage; by caspase-3
ChainResidueDetails
AASP34

218853

数据于2024-04-24公开中

PDB statisticsPDBj update infoContact PDBjnumon