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6E3G

Structure of RORgt in complex with a novel agonist.

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 601
ChainResidue
AMET313
ATRP317
ALEU391
AGLY392
AARG482
BGLN434

site_idAC2
Number of Residues17
Detailsbinding site for residue HOJ A 602
ChainResidue
AHIS323
ALEU324
AVAL361
AMET365
AALA368
APHE377
APHE378
AGLU379
APHE388
ALEU391
AILE400
AHIS479
AHOH708
AHOH769
AGLN286
ATRP317
ACYS320

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO B 601
ChainResidue
AGLN434
BMET313
BLEU391
BGLY392
BCYS393
BARG482

site_idAC4
Number of Residues15
Detailsbinding site for residue HOJ B 602
ChainResidue
BGLN286
BTRP317
BCYS320
BHIS323
BLEU324
BVAL361
BPHE377
BPHE378
BGLU379
BPHE388
BLEU391
BILE400
BHIS479
BHOH707
BHOH810

218500

数据于2024-04-17公开中

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