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5MME

Crystal structure of CREBBP bromodomain complexd with US46C

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
B0004402molecular_functionhistone acetyltransferase activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 8Q6 A 1201
ChainResidue
ALEU1109
AHOH1374
AHOH1377
AHOH1414
BLEU1120
B8Q61201
APRO1110
AGLN1113
AVAL1115
ALEU1120
AASN1168
AARG1173
AHOH1318
AHOH1322

site_idAC2
Number of Residues11
Detailsbinding site for residue 8Q6 B 1201
ChainResidue
A8Q61201
AHOH1377
BLEU1109
BPRO1110
BLEU1120
BASN1168
BARG1173
BVAL1174
BHOH1308
BHOH1342
BHOH1399

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

218853

數據於2024-04-24公開中

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