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5FTQ

Crystal structure of the ALK kinase domain in complex with Cmpd 17

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004672molecular_functionprotein kinase activity
A0004713molecular_functionprotein tyrosine kinase activity
A0004714molecular_functiontransmembrane receptor protein tyrosine kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
A0007169biological_processtransmembrane receptor protein tyrosine kinase signaling pathway
A0016020cellular_componentmembrane
PDBデータベースに由来する情報
site_idAC1
残基数18
詳細BINDING SITE FOR RESIDUE U4W A 2402
鎖名残基
ALEU1122
AGLY1202
AASP1203
AARG1253
AASN1254
ACYS1255
ALEU1256
AGLY1269
AASP1270
AHOH2103
APHE1127
AVAL1130
AALA1148
ALEU1196
AGLU1197
ALEU1198
AMET1199
AALA1200

site_idAC2
残基数3
詳細BINDING SITE FOR RESIDUE GOL A 2403
鎖名残基
APRO1351
ALYS1352
AHOH2309

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS00107
残基数29
詳細PROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGHGAFGEVYeGqvsgmpndpsplq.....VAVK
鎖名残基詳細
ALEU1122-LYS1150

site_idPS00109
残基数13
詳細PROTEIN_KINASE_TYR Tyrosine protein kinases specific active-site signature. FIHrDIAARNCLL
鎖名残基詳細
APHE1245-LEU1257

site_idPS00239
残基数9
詳細RECEPTOR_TYR_KIN_II Receptor tyrosine kinase class II signature. DIYrasYYR
鎖名残基詳細
AASP1276-ARG1284

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数1
詳細ACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159, ECO:0000255|PROSITE-ProRule:PRU10028
鎖名残基詳細
AASP1249

site_idSWS_FT_FI2
残基数2
詳細BINDING:
鎖名残基詳細
AHIS1124
AGLU1197

site_idSWS_FT_FI3
残基数1
詳細BINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
鎖名残基詳細
ALYS1150

site_idSWS_FT_FI4
残基数1
詳細BINDING: BINDING => ECO:0000269|PubMed:20632993
鎖名残基詳細
AASP1270

site_idSWS_FT_FI5
残基数1
詳細MOD_RES: Phosphotyrosine => ECO:0000269|PubMed:16878150, ECO:0007744|PubMed:15592455
鎖名残基詳細
ATYR1096

site_idSWS_FT_FI6
残基数1
詳細MOD_RES: Phosphotyrosine => ECO:0007744|PubMed:15592455
鎖名残基詳細
ATYR1131

site_idSWS_FT_FI7
残基数1
詳細MOD_RES: Phosphotyrosine => ECO:0000269|PubMed:15938644
鎖名残基詳細
ATYR1278

217705

件を2024-03-27に公開中

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