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4LUV

Fragment-Based Discovery of a Potent Inhibitor of Replication Protein A Protein-Protein Interactions

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0005634cellular_componentnucleus
A0006260biological_processDNA replication
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE 1XS A 201
ChainResidue
AARG41
AMET57
AALA59
ATHR60
AASN85
AILE95
A1DZ202
AHOH312
AHOH391

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE 1DZ A 202
ChainResidue
AARG31
AILE33
ATHR34
AARG43
ASER55
AMET57
AVAL93
A1XS201

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N-acetylmethionine => ECO:0007744|PubMed:19413330, ECO:0007744|PubMed:22223895
ChainResidueDetails
AMET1

site_idSWS_FT_FI2
Number of Residues3
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:26474068
ChainResidueDetails
ALYS22
ALYS88

218853

數據於2024-04-24公開中

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