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3UZC

Thermostabilised Adenosine A2A receptor in complex with 4-(3-amino-5-phenyl-1,2,4-triazin-6-yl)-2-chlorophenol

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0001609molecular_functionG protein-coupled adenosine receptor activity
A0001973biological_processG protein-coupled adenosine receptor signaling pathway
A0004930molecular_functionG protein-coupled receptor activity
A0007186biological_processG protein-coupled receptor signaling pathway
A0016020cellular_componentmembrane
PDBデータベースに由来する情報
site_idAC1
残基数9
詳細BINDING SITE FOR RESIDUE T4E A 330
鎖名残基
AVAL84
ALEU85
APHE168
ALEU249
AHIS250
AASN253
AILE274
AALA277
AHIS278

UniProtにおけるモチーフ・データベースPROSITEからの機能情報
site_idPS00237
残基数17
詳細G_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. SSIfSLLAIAIDRYIaI
鎖名残基詳細
ASER90-ILE106

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数52
詳細TOPO_DOM: Extracellular => ECO:0000269|PubMed:18832607
鎖名残基詳細
AMET1-SER7
ASER67-CYS77
AASN144-PRO173
ACYS259-PRO266

site_idSWS_FT_FI2
残基数24
詳細TRANSMEM: Helical; Name=1
鎖名残基詳細
AVAL8-TRP32

site_idSWS_FT_FI3
残基数63
詳細TOPO_DOM: Cytoplasmic => ECO:0000269|PubMed:18832607
鎖名残基詳細
ALEU33-ASN42
AASP101-ARG120
AARG199-SER234

site_idSWS_FT_FI4
残基数23
詳細TRANSMEM: Helical; Name=2
鎖名残基詳細
ATYR43-ILE66

site_idSWS_FT_FI5
残基数22
詳細TRANSMEM: Helical; Name=3
鎖名残基詳細
ALEU78-ILE100

site_idSWS_FT_FI6
残基数22
詳細TRANSMEM: Helical; Name=4
鎖名残基詳細
AALA121-TRP143

site_idSWS_FT_FI7
残基数24
詳細TRANSMEM: Helical; Name=5
鎖名残基詳細
AMET174-LEU198

site_idSWS_FT_FI8
残基数23
詳細TRANSMEM: Helical; Name=6
鎖名残基詳細
AALA235-PHE258

site_idSWS_FT_FI9
残基数23
詳細TRANSMEM: Helical; Name=7
鎖名残基詳細
ALEU267-TYR290

site_idSWS_FT_FI10
残基数4
詳細BINDING: BINDING => ECO:0000269|PubMed:21593763, ECO:0007744|PDB:2YDO
鎖名残基詳細
AGLU169
AASN253
AALA277
AHIS278

site_idSWS_FT_FI11
残基数1
詳細CARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
鎖名残基詳細
AASN154

218853

件を2024-04-24に公開中

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