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2VV2

hPPARgamma Ligand binding domain in complex with 5-HEPA

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 5HE A 1476
ChainResidue
AILE281
AHIS449
ALEU453
ATYR473
ACYS285
ASER289
AHIS323
ATYR327
ALEU330
ASER342
APHE363
AMET364

site_idAC2
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 5HE B 1476
ChainResidue
BILE281
BCYS285
BARG288
BGLU291
BLEU333
BLEU340
BSER342
BGLU343
BMET364
B5HE1477

site_idAC3
Number of Residues10
DetailsBINDING SITE FOR RESIDUE 5HE B 1477
ChainResidue
BLEU228
BPHE282
BCYS285
BARG288
BGLU295
BILE326
BMET329
BLEU333
BPHE363
B5HE1476

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000269|PubMed:9744270, ECO:0007744|PDB:2PRG
ChainResidueDetails
BTHR316
BLEU353
ATHR316
ALEU353

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin) => ECO:0000269|PubMed:36737649
ChainResidueDetails
ASER254
BSER254

218500

数据于2024-04-17公开中

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