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2OC0

Structure of NS3 complexed with a ketoamide inhibitor SCh491762

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0006508biological_processproteolysis
A0008236molecular_functionserine-type peptidase activity
A0019087biological_processtransformation of host cell by virus
C0006508biological_processproteolysis
C0008236molecular_functionserine-type peptidase activity
C0019087biological_processtransformation of host cell by virus
PDBデータベースに由来する情報
site_idAC1
残基数4
詳細BINDING SITE FOR RESIDUE ZN A 901
鎖名残基
ACYS97
ACYS99
ACYS145
AHOH1000

site_idAC2
残基数4
詳細BINDING SITE FOR RESIDUE ZN C 902
鎖名残基
CCYS97
CCYS99
CCYS145
CHOH915

site_idAC3
残基数3
詳細BINDING SITE FOR RESIDUE BME A 801
鎖名残基
AILE17
ATHR38
ACYS16

site_idAC4
残基数12
詳細BINDING SITE FOR RESIDUE HU1 A 999
鎖名残基
AGLN41
AHIS57
AILE132
ALYS136
AGLY137
ASER138
ASER139
APHE154
AARG155
AALA156
AALA157
ACYS159

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細ACT_SITE: Charge relay system; for serine protease NS3 activity => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000269|PubMed:8386278, ECO:0000305|PubMed:8861917
鎖名残基詳細
AHIS57
CHIS57

site_idSWS_FT_FI2
残基数2
詳細ACT_SITE: Charge relay system; for serine protease NS3 activity => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000305|PubMed:8861917
鎖名残基詳細
AASP81
CASP81

site_idSWS_FT_FI3
残基数2
詳細ACT_SITE: Charge relay system; for serine protease NS3 activity => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000269|PubMed:8248148, ECO:0000269|PubMed:8386278, ECO:0000305|PubMed:8861917
鎖名残基詳細
ASER139
CSER139

site_idSWS_FT_FI4
残基数4
詳細BINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000269|PubMed:21507982, ECO:0007744|PDB:1A1R, ECO:0007744|PDB:1N1L, ECO:0007744|PDB:1RGQ, ECO:0007744|PDB:2A4R, ECO:0007744|PDB:2F9V, ECO:0007744|PDB:2O8M, ECO:0007744|PDB:2OBQ, ECO:0007744|PDB:2OC0, ECO:0007744|PDB:2OC1, ECO:0007744|PDB:2OC7, ECO:0007744|PDB:2OC8, ECO:0007744|PDB:2OIN, ECO:0007744|PDB:2XNI
鎖名残基詳細
ACYS97
ACYS99
CCYS97
CCYS99

site_idSWS_FT_FI5
残基数2
詳細BINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000269|PubMed:21507982, ECO:0007744|PDB:1N1L, ECO:0007744|PDB:1RGQ, ECO:0007744|PDB:2A4R, ECO:0007744|PDB:2F9V, ECO:0007744|PDB:2O8M, ECO:0007744|PDB:2OBQ, ECO:0007744|PDB:2OC0, ECO:0007744|PDB:2OC1, ECO:0007744|PDB:2OC7, ECO:0007744|PDB:2OC8, ECO:0007744|PDB:2OIN, ECO:0007744|PDB:2XNI
鎖名残基詳細
ACYS145
CCYS145

site_idSWS_FT_FI6
残基数2
詳細BINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU01166, ECO:0000269|PubMed:21507982
鎖名残基詳細
AHIS149
CHIS149

CSAにおける酵素触媒機能の情報
site_idMCSA2
残基数4
詳細M-CSA 776
鎖名残基詳細
CHIS57proton shuttle (general acid/base)
CASP81electrostatic stabiliser
CGLY137electrostatic stabiliser
CSER139covalently attached, electrostatic stabiliser

site_idMCSA1
残基数4
詳細M-CSA 776
鎖名残基詳細
AHIS57proton shuttle (general acid/base)
AASP81electrostatic stabiliser
AGLY137electrostatic stabiliser
ASER139covalently attached, electrostatic stabiliser

217705

件を2024-03-27に公開中

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