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1X81

Farnesyl transferase structure of Jansen compound

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0008318molecular_functionprotein prenyltransferase activity
A0018342biological_processprotein prenylation
B0003824molecular_functioncatalytic activity
B0004311molecular_functionfarnesyltranstransferase activity
B0004659molecular_functionprenyltransferase activity
B0004660molecular_functionprotein farnesyltransferase activity
B0005515molecular_functionprotein binding
B0005875cellular_componentmicrotubule associated complex
B0005965cellular_componentprotein farnesyltransferase complex
B0006629biological_processlipid metabolic process
B0008270molecular_functionzinc ion binding
B0008283biological_processcell population proliferation
B0008284biological_processpositive regulation of cell population proliferation
B0008285biological_processnegative regulation of cell population proliferation
B0008318molecular_functionprotein prenyltransferase activity
B0010035biological_processresponse to inorganic substance
B0014070biological_processresponse to organic cyclic compound
B0016740molecular_functiontransferase activity
B0018343biological_processprotein farnesylation
B0034097biological_processresponse to cytokine
B0042060biological_processwound healing
B0042277molecular_functionpeptide binding
B0045787biological_processpositive regulation of cell cycle
B0046872molecular_functionmetal ion binding
B0048144biological_processfibroblast proliferation
B0048145biological_processregulation of fibroblast proliferation
B0048146biological_processpositive regulation of fibroblast proliferation
B0051770biological_processpositive regulation of nitric-oxide synthase biosynthetic process
PDBデータベースに由来する情報
site_idAC1
残基数4
詳細BINDING SITE FOR RESIDUE ZN B 2
鎖名残基
BJAN1
BASP297
BCYS299
BHIS362

site_idAC2
残基数6
詳細BINDING SITE FOR RESIDUE JAN B 1
鎖名残基
BTYR361
BZN2
BTRP102
BTRP106
BASP297
BASP359

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数3
詳細BINDING:
鎖名残基詳細
BHIS248
BARG291
BTYR300

site_idSWS_FT_FI2
残基数3
詳細BINDING: BINDING => ECO:0000269|PubMed:18844669, ECO:0000269|PubMed:20056542, ECO:0000269|PubMed:9065406
鎖名残基詳細
BASP297
BCYS299
BHIS362

site_idSWS_FT_FI3
残基数1
詳細SITE: Important for selectivity against geranylgeranyl diphosphate => ECO:0000250|UniProtKB:P49356
鎖名残基詳細
BTRP102

CSAにおける酵素触媒機能の情報
site_idMCSA1
残基数9
詳細M-CSA 484
鎖名残基詳細
BHIS248electrostatic stabiliser
BARG291electrostatic stabiliser
BLYS294electrostatic stabiliser
BASP297metal ligand
BCYS299metal ligand
BTYR300electrostatic stabiliser
BASP352metal ligand
BASP359electrostatic stabiliser
BHIS362metal ligand

218853

件を2024-04-24に公開中

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