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1MT8

Viability of a drug-resistant HIV-1 protease mutant: structural insights for better antiviral therapy

GO(遺伝子オントロジー)由来の情報
鎖名GO(遺伝子オントロジー)id名前空間内容
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
PDBデータベースに由来する情報
site_idAC1
残基数3
詳細BINDING SITE FOR RESIDUE ACT B 501
鎖名残基
APRO1
BHIS69
BLYS70

site_idAC2
残基数4
詳細BINDING SITE FOR RESIDUE ACT B 503
鎖名残基
AARG14
AGLY16
BARG14
BGLY16

site_idAC3
残基数2
詳細BINDING SITE FOR RESIDUE ACT P 508
鎖名残基
PALA2
PARG3

site_idAC4
残基数22
詳細BINDING SITE FOR CHAIN P OF CAPSID-P2 SUBSTRATE PEPTIDE OF HIV-1 GAG POLYPROTEIN
鎖名残基
AARG8
AASN25
AGLY27
AALA28
AASP29
AASP30
AGLY48
AGLY49
AILE50
AILE84
BASN25
BGLY27
BALA28
BASP29
BASP30
BILE47
BGLY48
BGLY49
BPRO81
PACT508
PHOH510
PHOH512

SwissProt/UniProtに記載されている蛋白質分子機能情報
site_idSWS_FT_FI1
残基数2
詳細SITE: Cleavage; by viral protease => ECO:0000250
鎖名残基詳細
AGLY78
BGLY78

site_idSWS_FT_FI2
残基数2
詳細MOD_RES: Phosphotyrosine; by host => ECO:0000250
鎖名残基詳細
AGLY78
BGLY78

217705

件を2024-03-27に公開中

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