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5H85

Crystal structure of the bromodomain of human CREBBP in complex with UO37D

Experimental procedure
実験手法SINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsSLS BEAMLINE X06DA
Synchrotron siteSLS
BeamlineX06DA
Temperature [K]100
Detector technologyPIXEL
Collection date2015-04-27
DetectorDECTRIS PILATUS 2M-F
Wavelength(s)1.00002
Spacegroup nameP 21 21 21
格子定数 [Å]24.413, 45.314, 104.660
格子定数 [度]90.00, 90.00, 90.00
精密化法
残基41.584 - 1.701
R因子0.163
Rwork0.161
R-free0.19850
Structure solution methodMOLECULAR REPLACEMENT
Starting model (for MR)4nr5
結合長の平均二乗偏差(RMSD) [Å]0.006
結合角の平均二乗偏差(RMSD) [度]0.832
Data reduction softwareXDS
Data scaling softwareSCALA (3.3.22)
Phasing softwarePHASER (2.5.7)
Refinement softwarePHENIX
Quality characteristics
 OverallInner shellOuter shell
分解能 [Å] (低)52.33045.3141.790
分解能 [Å] (高)1.7015.3801.700
Rmerge_l_obs0.0340.400
Rmeas0.077
Rpim0.0220.0100.128
Total number of observations151242594516287
独立反射数13297
<I/σ(I)>24.353.15.7
完全性 [%]98.899.893.9
冗長性11.411.69.1
結晶化条件
結晶ID方法pH温度溶液条件
1VAPOR DIFFUSION, HANGING DROP7.52770.15M KSCN, 20% PEG 3350, 10% EtGly

217705

件を2024-03-27に公開中

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