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1H07

CDK2 in complex with a disubstituted 4, 6-bis anilino pyrimidine CDK4 inhibitor

Experimental procedure
Experimental methodSINGLE WAVELENGTH
Source typeSYNCHROTRON
Source detailsSRS BEAMLINE PX9.6
Synchrotron siteSRS
BeamlinePX9.6
Temperature [K]100
Detector technologyIMAGE PLATE
Collection date1998-05-15
DetectorMARRESEARCH
Spacegroup nameP 21 21 21
Unit cell lengths53.323, 71.543, 72.550
Unit cell angles90.00, 90.00, 90.00
Refinement procedure
Resolution32.350 - 1.850
Rwork0.210
R-free0.23500
Structure solution methodMOLECULAR REPLACEMENT
RMSD bond length0.006
RMSD bond angle22.400

*

Data reduction softwareMOSFLM
Data scaling softwareSCALA
Phasing softwareAMoRE
Refinement softwareCNX (2000.1)
Data quality characteristics
 OverallOuter shell
Low resolution limit [Å]32.3501.950
High resolution limit [Å]1.8501.850
Rmerge0.0960.191
Total number of observations53065

*

Number of reflections21455
<I/σ(I)>10.24.7
Completeness [%]87.7

*

71.6
Redundancy2.52.1
Crystallization Conditions
crystal IDmethodpHtemperaturedetails
1unknown

*

7Lawrie, A.M., (1997) Nat.Struct.Biol., 4, 796.

*

217705

數據於2024-03-27公開中

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