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-Structure paper
Title | Development of Dimethylisoxazole-Attached Imidazo[1,2- a ]pyridines as Potent and Selective CBP/P300 Inhibitors. |
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Journal, issue, pages | J. Med. Chem., Vol. 64, Page 5787-5801, Year 2021 |
Publish date | Nov 12, 2020 (structure data deposition date) |
![]() | Muthengi, A. / Wimalasena, V.K. / Yosief, H.O. / Bikowitz, M.J. / Sigua, L.H. / Wang, T. / Li, D. / Gaieb, Z. / Dhawan, G. / Liu, S. ...Muthengi, A. / Wimalasena, V.K. / Yosief, H.O. / Bikowitz, M.J. / Sigua, L.H. / Wang, T. / Li, D. / Gaieb, Z. / Dhawan, G. / Liu, S. / Erickson, J. / Amaro, R.E. / Schonbrunn, E. / Qi, J. / Zhang, W. |
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Methods | X-ray diffraction |
Resolution | 1.7 Å |
Structure data | ![]() PDB-7kpy: |
Chemicals | ![]() ChemComp-EDO: ![]() ChemComp-WU1: ![]() ChemComp-HOH: |
Source |
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![]() | TRANSCRIPTION / epigenetics / inhibitor / drug development / multi domain proteins |